JP2011074063A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2011074063A5 JP2011074063A5 JP2010168639A JP2010168639A JP2011074063A5 JP 2011074063 A5 JP2011074063 A5 JP 2011074063A5 JP 2010168639 A JP2010168639 A JP 2010168639A JP 2010168639 A JP2010168639 A JP 2010168639A JP 2011074063 A5 JP2011074063 A5 JP 2011074063A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- salt
- carbon atoms
- general formula
- aminopyrazole derivative
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000004432 carbon atom Chemical group C* 0.000 claims description 35
- JVVRJMXHNUAPHW-UHFFFAOYSA-N 1h-pyrazol-5-amine Chemical class NC=1C=CNN=1 JVVRJMXHNUAPHW-UHFFFAOYSA-N 0.000 claims description 19
- 150000003839 salts Chemical class 0.000 claims description 17
- 125000000217 alkyl group Chemical group 0.000 claims description 14
- 125000003118 aryl group Chemical group 0.000 claims description 14
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims description 13
- 238000004519 manufacturing process Methods 0.000 claims description 11
- 125000003277 amino group Chemical group 0.000 claims description 10
- 125000000623 heterocyclic group Chemical group 0.000 claims description 9
- 125000003545 alkoxy group Chemical group 0.000 claims description 8
- 125000004104 aryloxy group Chemical group 0.000 claims description 8
- 125000003342 alkenyl group Chemical group 0.000 claims description 7
- 125000003282 alkyl amino group Chemical group 0.000 claims description 3
- 125000004414 alkyl thio group Chemical group 0.000 claims description 3
- 125000001769 aryl amino group Chemical group 0.000 claims description 3
- 125000005110 aryl thio group Chemical group 0.000 claims description 3
- 125000005843 halogen group Chemical group 0.000 claims description 3
- 150000001875 compounds Chemical class 0.000 claims 7
- 238000000034 method Methods 0.000 claims 4
- ZWEHNKRNPOVVGH-UHFFFAOYSA-N 2-Butanone Chemical compound CCC(C)=O ZWEHNKRNPOVVGH-UHFFFAOYSA-N 0.000 claims 3
- WFDIJRYMOXRFFG-UHFFFAOYSA-N Acetic anhydride Chemical compound CC(=O)OC(C)=O WFDIJRYMOXRFFG-UHFFFAOYSA-N 0.000 claims 3
- IKHGUXGNUITLKF-UHFFFAOYSA-N Acetaldehyde Chemical compound CC=O IKHGUXGNUITLKF-UHFFFAOYSA-N 0.000 claims 2
- CSCPPACGZOOCGX-UHFFFAOYSA-N Acetone Chemical compound CC(C)=O CSCPPACGZOOCGX-UHFFFAOYSA-N 0.000 claims 2
- 239000007789 gas Substances 0.000 claims 2
- FYSNRJHAOHDILO-UHFFFAOYSA-N thionyl chloride Chemical compound ClS(Cl)=O FYSNRJHAOHDILO-UHFFFAOYSA-N 0.000 claims 2
- FALRKNHUBBKYCC-UHFFFAOYSA-N 2-(chloromethyl)pyridine-3-carbonitrile Chemical compound ClCC1=NC=CC=C1C#N FALRKNHUBBKYCC-UHFFFAOYSA-N 0.000 claims 1
- NGNBDVOYPDDBFK-UHFFFAOYSA-N 2-[2,4-di(pentan-2-yl)phenoxy]acetyl chloride Chemical compound CCCC(C)C1=CC=C(OCC(Cl)=O)C(C(C)CCC)=C1 NGNBDVOYPDDBFK-UHFFFAOYSA-N 0.000 claims 1
- LGRFSURHDFAFJT-UHFFFAOYSA-N Phthalic anhydride Natural products C1=CC=C2C(=O)OC(=O)C2=C1 LGRFSURHDFAFJT-UHFFFAOYSA-N 0.000 claims 1
- WETWJCDKMRHUPV-UHFFFAOYSA-N acetyl chloride Chemical compound CC(Cl)=O WETWJCDKMRHUPV-UHFFFAOYSA-N 0.000 claims 1
- 239000012346 acetyl chloride Substances 0.000 claims 1
- 150000008065 acid anhydrides Chemical class 0.000 claims 1
- 125000003172 aldehyde group Chemical group 0.000 claims 1
- JHIWVOJDXOSYLW-UHFFFAOYSA-N butyl 2,2-difluorocyclopropane-1-carboxylate Chemical compound CCCCOC(=O)C1CC1(F)F JHIWVOJDXOSYLW-UHFFFAOYSA-N 0.000 claims 1
- 229910052799 carbon Inorganic materials 0.000 claims 1
- 125000004185 ester group Chemical group 0.000 claims 1
- 238000010438 heat treatment Methods 0.000 claims 1
- 150000002429 hydrazines Chemical class 0.000 claims 1
- 238000002955 isolation Methods 0.000 claims 1
- 125000000468 ketone group Chemical group 0.000 claims 1
- FPYJFEHAWHCUMM-UHFFFAOYSA-N maleic anhydride Chemical compound O=C1OC(=O)C=C1 FPYJFEHAWHCUMM-UHFFFAOYSA-N 0.000 claims 1
- 150000007522 mineralic acids Chemical class 0.000 claims 1
- 150000007524 organic acids Chemical class 0.000 claims 1
- 229940014800 succinic anhydride Drugs 0.000 claims 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2010168639A JP5789362B2 (ja) | 2009-09-04 | 2010-07-27 | ５−アミノピラゾール誘導体又はその塩の製造方法 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2009205354 | 2009-09-04 | ||
| JP2009205354 | 2009-09-04 | ||
| JP2010168639A JP5789362B2 (ja) | 2009-09-04 | 2010-07-27 | ５−アミノピラゾール誘導体又はその塩の製造方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2011074063A JP2011074063A (ja) | 2011-04-14 |
| JP2011074063A5 true JP2011074063A5 (enExample) | 2013-03-07 |
| JP5789362B2 JP5789362B2 (ja) | 2015-10-07 |
Family
ID=44018417
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010168639A Expired - Fee Related JP5789362B2 (ja) | 2009-09-04 | 2010-07-27 | ５−アミノピラゾール誘導体又はその塩の製造方法 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JP5789362B2 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2011201794A (ja) * | 2010-03-24 | 2011-10-13 | Fujifilm Corp | ５−アミノピラゾール誘導体及びその塩の製造方法 |
| JP6327369B2 (ja) | 2015-02-06 | 2018-05-23 | 日産自動車株式会社 | 自動変速機の制御装置 |
| CN111116416B (zh) * | 2019-12-30 | 2021-03-23 | 中国农业大学 | 一种β-氨基丙烯腈类化合物的制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4346097A (en) * | 1980-09-30 | 1982-08-24 | Warner-Lambert Company | Method for treating convulsions with pyrazole-4-carboxamide derivatives |
| US4393217A (en) * | 1981-01-12 | 1983-07-12 | American Cyanamid Company | Substituted phenyl-5-aminopyrazoles |
| ZA836003B (en) * | 1982-08-17 | 1984-07-25 | May & Baker Ltd | New tetrazine derivatives |
| JPS62158257A (ja) * | 1985-12-28 | 1987-07-14 | Konishiroku Photo Ind Co Ltd | ５−アミノピラゾ−ル−４−カルボキシレ−ト系化合物の製造方法 |
| US4826866A (en) * | 1987-11-02 | 1989-05-02 | A. H. Robins Company, Incorporated | 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics |
| JPH07206826A (ja) * | 1993-12-02 | 1995-08-08 | Fujisawa Pharmaceut Co Ltd | ５−アミノピラゾール誘導体の製造法 |
| US20070037987A1 (en) * | 2005-08-12 | 2007-02-15 | Chamberlin Kim S | Preparation of 4,5-diamino-1-(substituted)-pyrazole and acid addition salts thereof |
| JP5244369B2 (ja) * | 2006-11-10 | 2013-07-24 | 富士フイルム株式会社 | ５−アミノピラゾール誘導体の製造方法、アゾ色素 |
-
2010
- 2010-07-27 JP JP2010168639A patent/JP5789362B2/ja not_active Expired - Fee Related
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2015524409A5 (enExample) | ||
| JP6488359B2 (ja) | ベンズイミダゾール誘導体の製造方法 | |
| JP2015509939A5 (enExample) | ||
| RU2009105669A (ru) | Способ получения 3-замещенных 2-амино-5-галогенбензамидов | |
| JP2010502715A5 (enExample) | ||
| JP2010531876A5 (enExample) | ||
| WO2007102499A1 (ja) | ４－オキソキノリン化合物の製造方法 | |
| JP2015500335A5 (enExample) | ||
| JP2012515142A5 (enExample) | ||
| EP1945640A2 (en) | Process for the synthesis of 9-hydroxy risperidone (paliperidone) | |
| JP2012527489A5 (enExample) | ||
| JP2012517965A5 (enExample) | ||
| JP2013505273A5 (enExample) | ||
| JP2011074063A5 (enExample) | ||
| RU2012138410A (ru) | Соединение, содержащее кольцо пиридина, и способ получения галогенированного производного пиколина и производного тетразолилоксима | |
| JP2009532428A5 (enExample) | ||
| JP2008222606A5 (enExample) | ||
| JP2012131790A (ja) | ベンダムスチンアルキルエステル、ベンダムスチン、およびそれらの誘導体の製造のためのプロセス | |
| JP2008526918A5 (enExample) | ||
| JP6787331B2 (ja) | 酸ハライド溶液の製造方法、混合溶液、及びモノエステル化合物の製造方法 | |
| JP2015526507A (ja) | フルボキサミン遊離塩基の精製方法およびそれを用いた高純度フルボキサミンマレイン酸塩の製造方法 | |
| JP4701196B2 (ja) | ケイ素ルイス酸触媒、及びケイ素ルイス酸触媒を用いた反応方法 | |
| JP2008105970A (ja) | ジヒドロキノリン誘導体の製造方法及びその中間体 | |
| JPWO2017130871A1 (ja) | 酸ハライド溶液の製造方法、及びモノエステル化合物の製造方法 | |
| JP2015524846A5 (enExample) |