JP2010536719A5 - - Google Patents

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Publication number
JP2010536719A5
JP2010536719A5 JP2010520440A JP2010520440A JP2010536719A5 JP 2010536719 A5 JP2010536719 A5 JP 2010536719A5 JP 2010520440 A JP2010520440 A JP 2010520440A JP 2010520440 A JP2010520440 A JP 2010520440A JP 2010536719 A5 JP2010536719 A5 JP 2010536719A5
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JP
Japan
Prior art keywords
tumors
group
leukemia
head
chronic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010520440A
Other languages
English (en)
Japanese (ja)
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JP2010536719A (ja
Filing date
Publication date
Priority claimed from DE102007038957A external-priority patent/DE102007038957A1/de
Application filed filed Critical
Publication of JP2010536719A publication Critical patent/JP2010536719A/ja
Publication of JP2010536719A5 publication Critical patent/JP2010536719A5/ja
Pending legal-status Critical Current

Links

JP2010520440A 2007-08-17 2008-07-18 ６−チオキソピリダジン誘導体 Pending JP2010536719A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007038957A DE102007038957A1 (de) 2007-08-17 2007-08-17 6-Thioxo-pyridazinderivate
PCT/EP2008/005928 WO2009024221A1 (de) 2007-08-17 2008-07-18 6-thioxo-pyridazinderivate

Publications (2)

Publication Number Publication Date
JP2010536719A JP2010536719A (ja) 2010-12-02
JP2010536719A5 true JP2010536719A5 (enExample) 2011-09-08

Family

ID=40029265

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010520440A Pending JP2010536719A (ja) 2007-08-17 2008-07-18 ６−チオキソピリダジン誘導体

Country Status (7)

Country Link
US (1) US20110136819A1 (enExample)
EP (1) EP2176236A1 (enExample)
JP (1) JP2010536719A (enExample)
AU (1) AU2008290896A1 (enExample)
CA (1) CA2696472A1 (enExample)
DE (1) DE102007038957A1 (enExample)
WO (1) WO2009024221A1 (enExample)

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WO2012030633A1 (en) * 2010-08-31 2012-03-08 Merck Sharp & Dohme Corp. Tyrosine kinase inhibitors
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CA2915622C (en) 2013-06-21 2020-08-18 Zenith Epigenetics Corp. Novel substituted bicyclic compounds as bromodomain inhibitors
EA201690087A1 (ru) 2013-07-31 2016-08-31 Зенит Эпидженетикс Корп. Новые квиназолиноны как ингибиторы бромодомена
WO2016087936A1 (en) 2014-12-01 2016-06-09 Zenith Epigenetics Corp. Substituted pyridinones as bromodomain inhibitors
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CN107207474B (zh) 2014-12-11 2021-05-07 恒翼生物医药科技(上海)有限公司 被取代的杂环作为溴结构域抑制剂
JP2017538721A (ja) 2014-12-17 2017-12-28 ゼニス・エピジェネティクス・リミテッドＺｅｎｉｔｈ Ｅｐｉｇｅｎｅｔｉｃｓ Ｌｔｄ． ブロモドメインの阻害剤
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HUE063586T2 (hu) 2018-11-06 2024-01-28 Edgewise Therapeutics Inc Piridazinon-vegyületek és alkalmazásaik
KR20230124927A (ko) 2020-11-25 2023-08-28 아카제라 메디신즈, 인크. 핵산 전달을 위한 지질 나노입자, 및 관련 사용 방법
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