JP2010535738A5 - - Google Patents
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- Publication number
- JP2010535738A5 JP2010535738A5 JP2010519457A JP2010519457A JP2010535738A5 JP 2010535738 A5 JP2010535738 A5 JP 2010535738A5 JP 2010519457 A JP2010519457 A JP 2010519457A JP 2010519457 A JP2010519457 A JP 2010519457A JP 2010535738 A5 JP2010535738 A5 JP 2010535738A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- triazol
- ylamine
- trifluoromethyl
- methoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200701134 | 2007-08-08 | ||
| US95508107P | 2007-08-10 | 2007-08-10 | |
| PCT/EP2008/060307 WO2009019278A1 (en) | 2007-08-08 | 2008-08-06 | Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010535738A JP2010535738A (ja) | 2010-11-25 |
| JP2010535738A5 true JP2010535738A5 (https=) | 2011-09-15 |
Family
ID=39870242
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010519457A Abandoned JP2010535738A (ja) | 2007-08-08 | 2008-08-06 | ニコチン性アセチルコリン受容体の調節物質として有用な新規１，２，３−トリアゾール誘導体 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8110588B2 (https=) |
| EP (1) | EP2185529A1 (https=) |
| JP (1) | JP2010535738A (https=) |
| KR (1) | KR20100046179A (https=) |
| CN (1) | CN101796034A (https=) |
| AU (1) | AU2008285644A1 (https=) |
| CA (1) | CA2695812A1 (https=) |
| MX (1) | MX2010001135A (https=) |
| NZ (1) | NZ582520A (https=) |
| RU (1) | RU2010102994A (https=) |
| WO (1) | WO2009019278A1 (https=) |
| ZA (1) | ZA201000127B (https=) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110060017A1 (en) * | 2008-03-11 | 2011-03-10 | Neurosearch A/S | Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors |
| WO2010015583A1 (en) * | 2008-08-08 | 2010-02-11 | Neurosearch A/S | Novel diphenyl 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors |
| BRPI0917693A2 (pt) * | 2008-09-02 | 2016-05-17 | Neurosearch As | composto derivado de triazol, composição farmacêutica, e, uso de um derivado de triazol |
| ES2737429T3 (es) | 2009-10-07 | 2020-01-14 | Karo Pharma Ab | Pirazoles sustituidos como ligandos del receptor de estrógenos |
| SG192078A1 (en) | 2011-02-03 | 2013-08-30 | Lupin Ltd | Pyrrole derivatives used as modulators of alpha7 nachr |
| ES2594409T3 (es) | 2011-02-23 | 2016-12-20 | Lupin Limited | Derivados de heteroarilo como moduladores del nAChR á7 |
| WO2012131576A1 (en) | 2011-03-31 | 2012-10-04 | Lupin Limited | Pyrrole derivatives as nicotinic acetylcholine receptor modulators for use in the treatment of neurodegenerative disorders such as alzheimer's and parkinson's disease |
| FR2974365B1 (fr) * | 2011-04-20 | 2017-08-25 | Centre Nat De La Rech Scient (C N R S) | 1,2,3-triazoles 1,4-disubstituees, leurs procedes de preparation et leurs utilisations diagnostiques et therapeutiques |
| EP2729455B1 (en) | 2011-07-05 | 2016-09-14 | Lupin Limited | Biaryl derivatives as nachr modulators |
| GB201113538D0 (en) | 2011-08-04 | 2011-09-21 | Karobio Ab | Novel estrogen receptor ligands |
| NZ629453A (en) | 2012-03-06 | 2016-04-29 | Lupin Ltd | Thiazole derivatives as alpha 7 nachr modulators |
| US20150299178A1 (en) | 2012-11-12 | 2015-10-22 | Lupin Limited | Thiazole Derivatives as Alpha 7 NACHR Modulators |
| US9617211B2 (en) | 2013-01-16 | 2017-04-11 | Lupin Limited | Pyrrole derivatives as alpha 7 nAChR modulators |
| US9617210B2 (en) | 2013-03-13 | 2017-04-11 | Lupin Limited | Pyrrole derivatives as alpha 7 NACHR modulators |
| TW201446243A (zh) | 2013-06-03 | 2014-12-16 | Lupin Ltd | 4-(5-(4-氯苯基)-2-(2-環丙基乙醯基)-1,4-二甲基-1氫-吡咯-3-基)苯磺醯胺作為α7尼古丁乙醯膽鹼受體調節劑 |
| AU2014282886A1 (en) | 2013-06-17 | 2015-12-17 | Lupin Limited | Pyrrole derivatives as alpha 7 nAChR modulators |
| WO2019124577A1 (ko) * | 2017-12-20 | 2019-06-27 | 재단법인 경기도경제과학진흥원 | 트리아졸 유도체 및 이의 용도 |
| CN113045507B (zh) * | 2021-03-04 | 2022-10-25 | 中山大学南方学院 | 一种3,4-二羟基苯甲酸甲酯衍生物及其制备方法与应用 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1242216B (de) * | 1963-12-27 | 1967-06-15 | Union Carbide Corp | Verfahren zur Herstellung von Inaminsalzen |
| CA2469821C (en) * | 2001-12-18 | 2009-10-20 | Merck & Co., Inc. | Heteroaryl substituted triazole modulators of metabotropic glutamate receptor-5 |
| KR100755577B1 (ko) * | 2002-04-26 | 2007-09-12 | 일라이 릴리 앤드 캄파니 | 타키키닌 수용체 길항제로서의 트리아졸 유도체 |
| WO2005108347A2 (en) | 2004-05-06 | 2005-11-17 | The Regents Of The University Of California | Substituted enaminones, their derivatives and uses thereof |
| WO2006071184A1 (en) | 2004-12-28 | 2006-07-06 | Astrazeneca Ab | Aryl sulphonamide modulators |
| US20110060017A1 (en) | 2008-03-11 | 2011-03-10 | Neurosearch A/S | Novel 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors |
| WO2010015583A1 (en) | 2008-08-08 | 2010-02-11 | Neurosearch A/S | Novel diphenyl 1,2,3-triazole derivatives useful as modulators of nicotinic acetylcholine receptors |
-
2008
- 2008-08-06 EP EP08786915A patent/EP2185529A1/en not_active Withdrawn
- 2008-08-06 NZ NZ582520A patent/NZ582520A/en not_active IP Right Cessation
- 2008-08-06 CA CA2695812A patent/CA2695812A1/en not_active Abandoned
- 2008-08-06 CN CN200880102108A patent/CN101796034A/zh active Pending
- 2008-08-06 RU RU2010102994/04A patent/RU2010102994A/ru not_active Application Discontinuation
- 2008-08-06 AU AU2008285644A patent/AU2008285644A1/en not_active Abandoned
- 2008-08-06 MX MX2010001135A patent/MX2010001135A/es not_active Application Discontinuation
- 2008-08-06 KR KR1020107002808A patent/KR20100046179A/ko not_active Withdrawn
- 2008-08-06 JP JP2010519457A patent/JP2010535738A/ja not_active Abandoned
- 2008-08-06 WO PCT/EP2008/060307 patent/WO2009019278A1/en not_active Ceased
- 2008-08-06 US US12/672,252 patent/US8110588B2/en not_active Expired - Fee Related
-
2010
- 2010-01-07 ZA ZA2010/00127A patent/ZA201000127B/en unknown