JP2010533132A5 - - Google Patents

Download PDF

Info

Publication number
JP2010533132A5
JP2010533132A5 JP2010515363A JP2010515363A JP2010533132A5 JP 2010533132 A5 JP2010533132 A5 JP 2010533132A5 JP 2010515363 A JP2010515363 A JP 2010515363A JP 2010515363 A JP2010515363 A JP 2010515363A JP 2010533132 A5 JP2010533132 A5 JP 2010533132A5
Authority
JP
Japan
Prior art keywords
diseases
cancer
treatment
carcinoma
medicament
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2010515363A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010533132A (ja
JP5457343B2 (ja
Filing date
Publication date
Priority claimed from DE102007032739A external-priority patent/DE102007032739A1/de
Application filed filed Critical
Publication of JP2010533132A publication Critical patent/JP2010533132A/ja
Publication of JP2010533132A5 publication Critical patent/JP2010533132A5/ja
Application granted granted Critical
Publication of JP5457343B2 publication Critical patent/JP5457343B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2010515363A 2007-07-13 2008-06-16 キナゾリンアミド誘導体 Expired - Fee Related JP5457343B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102007032739.2 2007-07-13
DE102007032739A DE102007032739A1 (de) 2007-07-13 2007-07-13 Chinazolinamidderivate
PCT/EP2008/004846 WO2009010139A2 (de) 2007-07-13 2008-06-16 Chinazolinamidderivate

Publications (3)

Publication Number Publication Date
JP2010533132A JP2010533132A (ja) 2010-10-21
JP2010533132A5 true JP2010533132A5 (enExample) 2013-12-05
JP5457343B2 JP5457343B2 (ja) 2014-04-02

Family

ID=40121496

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010515363A Expired - Fee Related JP5457343B2 (ja) 2007-07-13 2008-06-16 キナゾリンアミド誘導体

Country Status (15)

Country Link
US (1) US8501754B2 (enExample)
EP (1) EP2164833B1 (enExample)
JP (1) JP5457343B2 (enExample)
KR (1) KR20100044846A (enExample)
CN (1) CN101743229B (enExample)
AR (1) AR067506A1 (enExample)
AU (1) AU2008278032B2 (enExample)
BR (1) BRPI0814236A2 (enExample)
CA (1) CA2694475C (enExample)
DE (1) DE102007032739A1 (enExample)
EA (1) EA017585B1 (enExample)
ES (1) ES2538218T3 (enExample)
IL (1) IL203206A (enExample)
WO (1) WO2009010139A2 (enExample)
ZA (1) ZA201001058B (enExample)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102008061214A1 (de) * 2008-12-09 2010-06-10 Merck Patent Gmbh Chinazolinamidderivate
AR077405A1 (es) 2009-07-10 2011-08-24 Sanofi Aventis Derivados del indol inhibidores de hsp90, composiciones que los contienen y utilizacion de los mismos para el tratamiento del cancer
FR2949467B1 (fr) 2009-09-03 2011-11-25 Sanofi Aventis Nouveaux derives de 5,6,7,8-tetrahydroindolizine inhibiteurs d'hsp90, compositions les contenant et utilisation
CN102711749A (zh) * 2009-11-05 2012-10-03 莱西肯医药有限公司 用于癌症治疗的色氨酸羟化酶抑制剂
DE102009054302A1 (de) * 2009-11-23 2011-05-26 Merck Patent Gmbh Chinazolinderivate
DE102010046837A1 (de) 2010-09-29 2012-03-29 Merck Patent Gmbh Phenylchinazolinderivate
LT2643313T (lt) 2010-11-24 2016-10-25 Merck Patent Gmbh Chinazolino karboksamido azetidinai
GB2486631A (en) * 2010-12-01 2012-06-27 Univ Sheffield Phenol/quinone boronic acids/esters and method of preparation thereof
TW201311149A (zh) * 2011-06-24 2013-03-16 Ishihara Sangyo Kaisha 有害生物防治劑
WO2014143960A1 (en) * 2013-03-15 2014-09-18 Rexahn Pharmaceuticals, Inc. Tetrahydroisoquinolin-2-yl-(quinazolin-4-yl) methanone compounds as cancer cell growth inhibitors
EP3253390B1 (en) 2015-02-06 2022-04-13 Merck Sharp & Dohme Corp. Aminoquinazoline compounds as a2a antagonist
EP3317278B1 (en) * 2015-07-01 2021-04-14 Crinetics Pharmaceuticals, Inc. Somatostatin modulators and uses thereof
JP6740354B2 (ja) 2015-10-05 2020-08-12 ザ トラスティーズ オブ コロンビア ユニバーシティー イン ザ シティー オブ ニューヨーク オートファジーの流れ及びホスホリパーゼd及びタウを含むタンパク質凝集体のクリアランスの活性化剤ならびにタンパク質症の治療方法
TWI734806B (zh) * 2016-07-19 2021-08-01 日商日本化藥股份有限公司 攝像元件用光電變換元件用材料及含有該材料之光電變換元件
AU2018290511B2 (en) * 2017-06-26 2022-01-27 Sunshine Lake Pharma Co., Ltd. Dihydropyrimidine compounds and uses thereof in medicine
CN107382976A (zh) * 2017-07-04 2017-11-24 孙秀芹 一种治疗盆腔炎的化合物及制备方法和应用
CN107488168A (zh) * 2017-07-18 2017-12-19 黄绍菊 一种治疗盆腔炎的化合物及制备方法和应用
EP3658560A4 (en) 2017-07-25 2021-01-06 Crinetics Pharmaceuticals, Inc. SOMATOSTAT IN MODULATORS AND USES THEREOF
TWI853814B (zh) 2018-05-31 2024-09-01 南韓商C&C新藥研究所 雜環衍生物及其用途
US20230250088A1 (en) * 2020-07-15 2023-08-10 Ifm Due, Inc. Compounds and compositions for treating conditions associated with sting activity
IL310724A (en) 2021-08-10 2024-04-01 Ifm Due Inc COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH STING ACTIVITY
WO2023244713A1 (en) * 2022-06-16 2023-12-21 Ensem Therapeutics, Inc. Quinazoline derivatives, compositions and methods thereof

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5968921A (en) 1997-10-24 1999-10-19 Orgegon Health Sciences University Compositions and methods for promoting nerve regeneration
AU3378599A (en) 1998-04-03 1999-10-25 University Of Pittsburgh Benzoquinoid ansamycins for the treatment of cardiac arrest and stroke
EP1161231A2 (en) 1999-03-12 2001-12-12 THE UNITED STATES OF AMERICA, represented by THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES NATIONAL INSTITUTES OF HEALTH Method of inhibiting a chaperone protein
CA2429196A1 (en) 2000-03-24 2001-10-04 Duke University Characterization of grp94-ligand interactions and purification, screening, and therapeutic methods relating thereto
AU2001271567A1 (en) 2000-06-29 2002-01-14 Trustees Of Boston University Use of geldanamycin and related compounds for prophylaxis or treatment of fibrogenic disorders
JP2004504356A (ja) 2000-07-20 2004-02-12 メルク エンド カムパニー インコーポレーテッド C型肝炎ウイルスのプロセシングおよび複製の抑制
ATE526019T1 (de) 2000-07-28 2011-10-15 Sloan Kettering Inst Cancer Verfahren zur behandlung von zellproliferationen störungen und virusinfektionen
CN1300116C (zh) 2001-04-16 2007-02-14 卫材株式会社 1h-吲唑化合物
EP1450784A4 (en) 2001-11-09 2005-02-09 Conforma Therapeutics Corp HSP90-INHIBITABLE ZEARALANOL COMPOUNDS AND METHOD FOR THEIR PREPARATION AND USE
WO2006010595A1 (en) 2004-07-27 2006-02-02 Novartis Ag Inhibitors of hsp90
US20070054916A1 (en) * 2004-10-01 2007-03-08 Amgen Inc. Aryl nitrogen-containing bicyclic compounds and methods of use
DE102005022977A1 (de) * 2005-05-19 2006-12-07 Merck Patent Gmbh Phenylchinazolinderivate

Similar Documents

Publication Publication Date Title
JP2010533132A5 (enExample)
JP2010516639A5 (enExample)
Kunnumakkara et al. Curcumin inhibits proliferation, invasion, angiogenesis and metastasis of different cancers through interaction with multiple cell signaling proteins
MX2019001302A (es) Conjugados de farmaco con enlazadores autoestabilizantes que tienen propiedades fisioquimicas mejoradas.
TW200640883A (en) Compounds for the treatment of proliferative disorders
CY1117440T1 (el) Συτηκτα παραγωγα ιμιδαζολης ως αναστολεις toy ido
AU2015231270B2 (en) Antifungal compound process
IL180979A (en) Isoindulin compounds and their use
BRPI0916356A2 (enExample)
EP3119754A1 (en) Antifungal compound process
WO2009066060A3 (en) 4-substituted-6-isopropyl-benzene-1,3-diol compounds and their use
JP2018527301A5 (ja) アジリジン含有dnaアルキル化剤
Huo et al. 2-Arylindoles: concise syntheses and a privileged scaffold for fungicide discovery
EA202090259A1 (ru) Новые гетероариламидные производные как селективные ингибиторы гистондеацетилаз 1 и/или 2 (hdac1-2)
TNSN07294A1 (en) Treatment of metastasized tumors
TW200745043A (en) Substituted pyrazoline compounds, their preparation and use as medicaments
MX2024002409A (es) Terapias contra el cancer.
Ozdemir et al. Synthesis, anticonvulsant and antimicrobial activities of some new [1-(2-naphthyl)-2-(pyrazol-1-yl) ethanone] oxime ethers
Ye et al. Actively targeted delivery of doxorubicin to bone metastases by a pH-sensitive conjugation
Movafagh et al. Histone deacetylase inhibitors in cancer prevention and therapy
JP2017511340A5 (enExample)
WO2007009721A3 (en) Indoline-substituted pyrazoline derivatives, their preparation and use as medicaments
EA201270347A1 (ru) Производные апогоссиполона в качестве противоопухолевых агентов
WO2015081867A1 (zh) 吉西他滨衍生物、含该衍生物的组合物及所述衍生物的制药用途
Hassan et al. Synthesis and pharmacological profiling of mono imine Schiff bases: Dual anti-inflammatory and antibacterial activity with computational insights