JP2010520306A - エストロゲン関連受容体−αモジュレーターとしての置換フェノキシチアゾリジンジオン - Google Patents
エストロゲン関連受容体−αモジュレーターとしての置換フェノキシチアゾリジンジオン Download PDFInfo
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- JP2010520306A JP2010520306A JP2009552881A JP2009552881A JP2010520306A JP 2010520306 A JP2010520306 A JP 2010520306A JP 2009552881 A JP2009552881 A JP 2009552881A JP 2009552881 A JP2009552881 A JP 2009552881A JP 2010520306 A JP2010520306 A JP 2010520306A
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/44—Two oxygen atoms
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US89345307P | 2007-03-07 | 2007-03-07 | |
| PCT/US2008/056004 WO2008109727A1 (en) | 2007-03-07 | 2008-03-06 | Substituted phenoxy thiazolidinediones as estrogen related receptor-alpha modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010520306A true JP2010520306A (ja) | 2010-06-10 |
| JP2010520306A5 JP2010520306A5 (OSRAM) | 2011-03-24 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2009552881A Pending JP2010520306A (ja) | 2007-03-07 | 2008-03-06 | エストロゲン関連受容体−αモジュレーターとしての置換フェノキシチアゾリジンジオン |
Country Status (21)
| Country | Link |
|---|---|
| US (2) | US7846953B2 (OSRAM) |
| EP (1) | EP2129668A1 (OSRAM) |
| JP (1) | JP2010520306A (OSRAM) |
| KR (1) | KR20090127410A (OSRAM) |
| CN (1) | CN101679322A (OSRAM) |
| AR (1) | AR065655A1 (OSRAM) |
| AU (1) | AU2008222745A1 (OSRAM) |
| BR (1) | BRPI0808445A2 (OSRAM) |
| CA (1) | CA2679944A1 (OSRAM) |
| CL (1) | CL2008000670A1 (OSRAM) |
| CO (1) | CO6231008A2 (OSRAM) |
| EA (1) | EA200970837A1 (OSRAM) |
| EC (1) | ECSP099614A (OSRAM) |
| IL (1) | IL200757A0 (OSRAM) |
| MX (1) | MX2009009517A (OSRAM) |
| NI (1) | NI200900163A (OSRAM) |
| NZ (1) | NZ579372A (OSRAM) |
| SV (1) | SV2009003367A (OSRAM) |
| TW (1) | TW200902508A (OSRAM) |
| UA (1) | UA98485C2 (OSRAM) |
| WO (1) | WO2008109727A1 (OSRAM) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013532682A (ja) * | 2010-07-28 | 2013-08-19 | オーキッド ケミカルズ アンド ファーマシューティカルズ リミテッド | 肝臓、肺の障害、糖尿病合併症および心血管疾患の処置のためのジフェニルエーテル化合物 |
| JP2023501081A (ja) * | 2019-10-18 | 2023-01-18 | リード ファーマ ホールディング ビー．ブイ． | エストロゲン関連受容体アルファ（ＥＲＲα）モジュレーター |
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| TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
| ATE516272T1 (de) | 2007-09-14 | 2011-07-15 | Ortho Mcneil Janssen Pharm | 1,3-disubstituierte 4-(aryl-x-phenyl)-1h-pyridin- 2-one |
| TWI475995B (zh) | 2007-09-14 | 2015-03-11 | Janssen Pharmaceuticals Inc | １’，３’－二取代－４－苯基－３，４，５，６－四氫－２ｈ，１’ｈ－〔１，４’〕聯吡啶基－２’－酮化物 |
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| AU2008222745A1 (en) * | 2007-03-07 | 2008-09-12 | Janssen Pharmaceutica N.V. | Substituted phenoxy thiazolidinediones as estrogen related receptor-alpha modulators |
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2008
- 2008-03-06 AU AU2008222745A patent/AU2008222745A1/en not_active Abandoned
- 2008-03-06 US US12/043,269 patent/US7846953B2/en not_active Expired - Fee Related
- 2008-03-06 CN CN200880015196A patent/CN101679322A/zh active Pending
- 2008-03-06 BR BRPI0808445-9A patent/BRPI0808445A2/pt not_active IP Right Cessation
- 2008-03-06 CL CL2008000670A patent/CL2008000670A1/es unknown
- 2008-03-06 EP EP08731504A patent/EP2129668A1/en not_active Ceased
- 2008-03-06 MX MX2009009517A patent/MX2009009517A/es active IP Right Grant
- 2008-03-06 CA CA002679944A patent/CA2679944A1/en not_active Abandoned
- 2008-03-06 UA UAA200910123A patent/UA98485C2/ru unknown
- 2008-03-06 NZ NZ579372A patent/NZ579372A/en not_active IP Right Cessation
- 2008-03-06 TW TW097107941A patent/TW200902508A/zh unknown
- 2008-03-06 WO PCT/US2008/056004 patent/WO2008109727A1/en not_active Ceased
- 2008-03-06 JP JP2009552881A patent/JP2010520306A/ja active Pending
- 2008-03-06 EA EA200970837A patent/EA200970837A1/ru unknown
- 2008-03-06 KR KR1020097020449A patent/KR20090127410A/ko not_active Withdrawn
- 2008-03-07 AR ARP080100962A patent/AR065655A1/es not_active Application Discontinuation
-
2009
- 2009-09-04 NI NI200900163A patent/NI200900163A/es unknown
- 2009-09-06 IL IL200757A patent/IL200757A0/en unknown
- 2009-09-07 SV SV2009003367A patent/SV2009003367A/es unknown
- 2009-09-07 EC EC2009009614A patent/ECSP099614A/es unknown
- 2009-09-11 CO CO09097934A patent/CO6231008A2/es not_active Application Discontinuation
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2010
- 2010-10-07 US US12/899,812 patent/US8344009B2/en not_active Expired - Fee Related
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| JPH09176162A (ja) * | 1995-12-22 | 1997-07-08 | Toubishi Yakuhin Kogyo Kk | チアゾリジンジオン誘導体及びその製造法並びにそれを含む医薬組成物 |
| WO2001025181A1 (en) * | 1999-10-01 | 2001-04-12 | Eisai Co., Ltd. | Carboxylic acid derivatives and drugs containing the same |
| WO2006019741A1 (en) * | 2004-07-14 | 2006-02-23 | Janssen Pharmaceutica N.V. | Arylidenes for the treatment of estrogen related receptor-alpha mediated diseases |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013532682A (ja) * | 2010-07-28 | 2013-08-19 | オーキッド ケミカルズ アンド ファーマシューティカルズ リミテッド | 肝臓、肺の障害、糖尿病合併症および心血管疾患の処置のためのジフェニルエーテル化合物 |
| JP2023501081A (ja) * | 2019-10-18 | 2023-01-18 | リード ファーマ ホールディング ビー．ブイ． | エストロゲン関連受容体アルファ（ＥＲＲα）モジュレーター |
| JP7629912B2 (ja) | 2019-10-18 | 2025-02-14 | リード ファーマ ホールディング ビー．ブイ． | エストロゲン関連受容体アルファ（ＥＲＲα）モジュレーター |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2129668A1 (en) | 2009-12-09 |
| BRPI0808445A2 (pt) | 2014-08-05 |
| WO2008109727A1 (en) | 2008-09-12 |
| ECSP099614A (es) | 2009-10-30 |
| AU2008222745A1 (en) | 2008-09-12 |
| TW200902508A (en) | 2009-01-16 |
| NZ579372A (en) | 2012-02-24 |
| CN101679322A (zh) | 2010-03-24 |
| US20110237625A1 (en) | 2011-09-29 |
| AR065655A1 (es) | 2009-06-24 |
| MX2009009517A (es) | 2009-09-16 |
| KR20090127410A (ko) | 2009-12-11 |
| EA200970837A1 (ru) | 2010-04-30 |
| IL200757A0 (en) | 2010-05-17 |
| WO2008109727A8 (en) | 2009-12-17 |
| CA2679944A1 (en) | 2008-09-12 |
| NI200900163A (es) | 2010-07-22 |
| SV2009003367A (es) | 2010-08-10 |
| US8344009B2 (en) | 2013-01-01 |
| US7846953B2 (en) | 2010-12-07 |
| CO6231008A2 (es) | 2010-12-20 |
| CL2008000670A1 (es) | 2008-11-03 |
| UA98485C2 (ru) | 2012-05-25 |
| US20090111855A1 (en) | 2009-04-30 |
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