JP2010501609A - コア層と１又は複数のバリヤー層を含む徐放性経口投与用配合剤 - Google Patents
コア層と１又は複数のバリヤー層を含む徐放性経口投与用配合剤 Download PDFInfo
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- OGWKCGZFUXNPDA-XQKSVPLYSA-N vincristine Chemical compound C([N@]1C[C@@H](C[C@]2(C(=O)OC)C=3C(=CC4=C([C@]56[C@H]([C@@]([C@H](OC(C)=O)[C@]7(CC)C=CCN([C@H]67)CC5)(O)C(=O)OC)N4C=O)C=3)OC)C[C@@](C1)(O)CC)CC1=C2NC2=CC=CC=C12 OGWKCGZFUXNPDA-XQKSVPLYSA-N 0.000 description 1
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- 229960004355 vindesine Drugs 0.000 description 1
- UGGWPQSBPIFKDZ-KOTLKJBCSA-N vindesine Chemical compound C([C@@H](C[C@]1(C(=O)OC)C=2C(=CC3=C([C@]45[C@H]([C@@]([C@H](O)[C@]6(CC)C=CCN([C@H]56)CC4)(O)C(N)=O)N3C)C=2)OC)C[C@@](C2)(O)CC)N2CCC2=C1N=C1[C]2C=CC=C1 UGGWPQSBPIFKDZ-KOTLKJBCSA-N 0.000 description 1
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- PJVWKTKQMONHTI-UHFFFAOYSA-N warfarin Chemical compound OC=1C2=CC=CC=C2OC(=O)C=1C(CC(=O)C)C1=CC=CC=C1 PJVWKTKQMONHTI-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4422—1,4-Dihydropyridines, e.g. nifedipine, nicardipine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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- A—HUMAN NECESSITIES
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
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- Medicinal Chemistry (AREA)
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- Engineering & Computer Science (AREA)
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- Physiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| JP2009525976A Pending JP2010501609A (ja) | 2006-08-30 | 2007-08-29 | コア層と１又は複数のバリヤー層を含む徐放性経口投与用配合剤 |
| JP2014031474A Active JP5788547B2 (ja) | 2006-08-30 | 2014-02-21 | コア層と１又は複数のバリヤー層を含む徐放性経口投与用配合剤 |
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| KR20200077542A (ko) * | 2017-10-25 | 2020-06-30 | 키에시 파르마슈티시 엣스. 피. 에이. | 지연 방출 데페리프론 정제 및 그의 사용 방법 |
| JP2022513906A (ja) * | 2018-12-14 | 2022-02-09 | ディピエッレ ファルマ ソシエタ ペル アチオニ | メサラジンまたはその誘導体を投与するための固体経口医薬組成物 |
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| WO2009012791A1 (en) * | 2007-07-23 | 2009-01-29 | Pharmathen S.A. | Pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof |
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- 2007-08-29 WO PCT/EP2007/007549 patent/WO2008025535A1/en not_active Ceased
- 2007-08-29 KR KR1020097006438A patent/KR101575679B1/ko active Active
- 2007-08-29 EP EP07801966A patent/EP2063871A1/en not_active Withdrawn
- 2007-08-29 CA CA002662122A patent/CA2662122A1/en not_active Abandoned
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- 2007-08-29 WO PCT/EP2007/007545 patent/WO2008025532A1/en not_active Ceased
- 2007-08-29 JP JP2009525973A patent/JP2010501607A/ja not_active Abandoned
- 2007-08-29 AU AU2007291509A patent/AU2007291509B2/en active Active
- 2007-08-29 AU AU2007291506A patent/AU2007291506A1/en not_active Abandoned
- 2007-08-29 JP JP2009525976A patent/JP2010501609A/ja active Pending
- 2007-08-29 KR KR1020097006435A patent/KR20090065519A/ko not_active Withdrawn
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- 2007-08-29 ES ES07801970T patent/ES2547226T5/es active Active
- 2007-08-29 EP EP07801970.0A patent/EP2063872B2/en active Active
- 2007-08-29 US US11/846,896 patent/US9101544B2/en active Active
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2009
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Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20200077542A (ko) * | 2017-10-25 | 2020-06-30 | 키에시 파르마슈티시 엣스. 피. 에이. | 지연 방출 데페리프론 정제 및 그의 사용 방법 |
| JP2021500377A (ja) * | 2017-10-25 | 2021-01-07 | キエージ・フアルマチエウテイチ・エツセ・ピ・ア | 遅延放出デフェリプロン錠剤及びその使用法 |
| JP7246384B2 (ja) | 2017-10-25 | 2023-03-27 | キエージ・フアルマチエウテイチ・エツセ・ピ・ア | 遅延放出デフェリプロン錠剤及びその使用法 |
| KR102624627B1 (ko) * | 2017-10-25 | 2024-01-16 | 키에시 파르마슈티시 엣스. 피. 에이. | 지연 방출 데페리프론 정제 및 그의 사용 방법 |
| JP2022513906A (ja) * | 2018-12-14 | 2022-02-09 | ディピエッレ ファルマ ソシエタ ペル アチオニ | メサラジンまたはその誘導体を投与するための固体経口医薬組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2063871A1 (en) | 2009-06-03 |
| MX2009002236A (es) | 2009-03-13 |
| ZA200901688B (en) | 2014-02-26 |
| US20080057123A1 (en) | 2008-03-06 |
| CA2662123A1 (en) | 2008-03-06 |
| AU2007291506A1 (en) | 2008-03-06 |
| KR101575679B1 (ko) | 2015-12-08 |
| CA2662122A1 (en) | 2008-03-06 |
| JP2010501607A (ja) | 2010-01-21 |
| KR20090065520A (ko) | 2009-06-22 |
| US20160008288A1 (en) | 2016-01-14 |
| EP2063872B1 (en) | 2015-05-06 |
| JP2014114323A (ja) | 2014-06-26 |
| KR20090065519A (ko) | 2009-06-22 |
| WO2008025532A1 (en) | 2008-03-06 |
| AU2007291509A1 (en) | 2008-03-06 |
| CA2662123C (en) | 2015-12-01 |
| EP2063872A1 (en) | 2009-06-03 |
| JP5788547B2 (ja) | 2015-09-30 |
| ES2547226T5 (es) | 2020-06-12 |
| US9101544B2 (en) | 2015-08-11 |
| US9622980B2 (en) | 2017-04-18 |
| AU2007291509B2 (en) | 2013-05-02 |
| US20080063711A1 (en) | 2008-03-13 |
| WO2008025535A1 (en) | 2008-03-06 |
| ES2547226T3 (es) | 2015-10-02 |
| MX2009002235A (es) | 2009-03-13 |
| EP2063872B2 (en) | 2019-12-04 |
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