JP2009536961A - インテグリンを阻害する新規複素環化合物及びその使用 - Google Patents

インテグリンを阻害する新規複素環化合物及びその使用 Download PDF

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JP2009536961A
JP2009536961A JP2009510340A JP2009510340A JP2009536961A JP 2009536961 A JP2009536961 A JP 2009536961A JP 2009510340 A JP2009510340 A JP 2009510340A JP 2009510340 A JP2009510340 A JP 2009510340A JP 2009536961 A JP2009536961 A JP 2009536961A
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ylamino
methyl
phenyl
acid compound
propanoic acid
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JP2009536961A5 (https=
Inventor
ツィシンスキー，グンター
シュトラギース，ロラント
オスターカンプ，フランク
シャルン，ディルク
フンメル，ゲルト
カルクホフ，ホルガー
ツァーン，グリット
フォッスマイアー，デルテ
クリストナー−アルブレヒト，クラウディア
ライネケ，ウルリッヒ
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Jerini AG
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Jerini AG
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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  • Ophthalmology & Optometry (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
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  • Pain & Pain Management (AREA)
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  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2009510340A 2006-05-12 2007-05-14 インテグリンを阻害する新規複素環化合物及びその使用 Pending JP2009536961A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06009872 2006-05-12
PCT/EP2007/004283 WO2007131764A2 (en) 2006-05-12 2007-05-14 New heterocyclic compounds for the inhibition of integrins and use thereof

Publications (2)

Publication Number Publication Date
JP2009536961A true JP2009536961A (ja) 2009-10-22
JP2009536961A5 JP2009536961A5 (https=) 2010-07-01

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Country Link
US (1) US8309735B2 (https=)
EP (1) EP2024357A2 (https=)
JP (1) JP2009536961A (https=)
KR (1) KR20090017512A (https=)
CN (1) CN101448818A (https=)
AR (1) AR060901A1 (https=)
AU (1) AU2007251756A1 (https=)
BR (1) BRPI0711659A2 (https=)
CA (1) CA2652101A1 (https=)
IL (1) IL194946A0 (https=)
MX (1) MX2008014345A (https=)
RU (1) RU2008148943A (https=)
TW (1) TW200811164A (https=)
WO (1) WO2007131764A2 (https=)
ZA (1) ZA200809074B (https=)

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AR059224A1 (es) 2006-01-31 2008-03-19 Jerini Ag Compuestos para la inhibicion de integrinas y uso de estas
TW200811164A (en) 2006-05-12 2008-03-01 Jerini Ag New heterocyclic compounds for the inhibition of integrins and use thereof
WO2008093064A1 (en) * 2007-01-29 2008-08-07 Astrazeneca Ab L-ALANINE DERIVATIVES AS α5 BETA 1 ANTAGONISTS
WO2010062829A1 (en) * 2008-11-28 2010-06-03 Lexicon Pharmaceuticals, Inc. Tryptophan hydroxylase inhibitors for treating osteoporosis
UA110924C2 (uk) * 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
AU2010315190A1 (en) * 2009-11-05 2012-05-10 Lexicon Pharmaceuticals, Inc. Tryptophan hydroxylase inhibitors for the treatment of cancer
WO2015048819A1 (en) 2013-09-30 2015-04-02 The Regents Of The University Of California Anti-alphavbeta1 integrin compounds and methods
CN103588770B (zh) * 2013-11-27 2016-08-17 武汉尚赛光电科技有限公司 1，2，4-噻二唑衍生物及其作为电致发光材料的应用
CA2981371A1 (en) * 2015-03-10 2016-09-15 The Regents Of The University Of California Anti-alphavbeta1 integrin inhibitors and methods of use
CN108794496B (zh) * 2018-04-28 2020-04-24 北京施安泰医药技术开发有限公司 一类cdk抑制剂、其药物组合物、制备方法及用途
EP3932912A4 (en) * 2019-02-28 2022-09-07 Osaka University PROTEIN AND/OR PEPTIDE MODIFICATION MOLECULE

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JP4250423B2 (ja) * 2001-03-19 2009-04-08 大日本住友製薬株式会社 アリール置換脂環式化合物及びそれを含有する医薬組成物
WO2003089410A1 (en) 2002-04-19 2003-10-30 Kyowa Hakko Kogyo Co., Ltd. Phenylalanine derivative
JP5032299B2 (ja) 2004-03-24 2012-09-26 シャイア・オーファン・セラピーズ・ゲーエムベーハー 血管形成を阻害する新規化合物及びその使用
EP1957476A1 (en) 2005-11-23 2008-08-20 AstraZeneca AB L-alanine derivatives
TW200811164A (en) 2006-05-12 2008-03-01 Jerini Ag New heterocyclic compounds for the inhibition of integrins and use thereof

Patent Citations (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH072851A (ja) * 1993-01-26 1995-01-06 Dr Karl Thomae Gmbh ５員複素環化合物、それらの調製方法及びこれらの化合物を含む医薬組成物
JP2000502708A (ja) * 1995-12-29 2000-03-07 スミスクライン・ビーチャム・コーポレイション ビトロネクチン受容体拮抗物質
JP2001517245A (ja) * 1997-05-29 2001-10-02 メルク エンド カンパニー インコーポレーテッド 細胞接着阻害薬としてのビアリールアルカン酸類
WO1999026923A1 (en) * 1997-11-20 1999-06-03 Merck & Co., Inc. Para-aminomethylaryl carboxamide derivatives
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ZA200809074B (en) 2009-08-26
CN101448818A (zh) 2009-06-03
US20090203745A1 (en) 2009-08-13
IL194946A0 (en) 2009-08-03
EP2024357A2 (en) 2009-02-18
BRPI0711659A2 (pt) 2012-01-17
WO2007131764A3 (en) 2008-01-10
WO2007131764A2 (en) 2007-11-22
RU2008148943A (ru) 2010-06-20
CA2652101A1 (en) 2007-11-22
MX2008014345A (es) 2008-11-27
TW200811164A (en) 2008-03-01
US8309735B2 (en) 2012-11-13

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