JP2009533472A - 癌治療法 - Google Patents
癌治療法 Download PDFInfo
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- JP2009533472A JP2009533472A JP2009505614A JP2009505614A JP2009533472A JP 2009533472 A JP2009533472 A JP 2009533472A JP 2009505614 A JP2009505614 A JP 2009505614A JP 2009505614 A JP2009505614 A JP 2009505614A JP 2009533472 A JP2009533472 A JP 2009533472A
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- inhibitor
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US79184106P | 2006-04-13 | 2006-04-13 | |
| PCT/US2007/066478 WO2007121279A2 (en) | 2006-04-13 | 2007-04-12 | Cancer treatment method |
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| JP2009533472A true JP2009533472A (ja) | 2009-09-17 |
| JP2009533472A5 JP2009533472A5 (enExample) | 2010-05-20 |
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| JP2009505614A Pending JP2009533472A (ja) | 2006-04-13 | 2007-04-12 | 癌治療法 |
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| EP (1) | EP2012587A2 (enExample) |
| JP (1) | JP2009533472A (enExample) |
| WO (1) | WO2007121279A2 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012026511A1 (ja) * | 2010-08-27 | 2012-03-01 | 協和発酵キリン株式会社 | 医薬組成物 |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI1015216A2 (pt) * | 2009-04-16 | 2016-04-12 | Merck Sharp & Dohme | método de tratar ou prevenir uma condição médica em um indivíduo. |
| US8623604B2 (en) * | 2009-09-09 | 2014-01-07 | Quintiles Transnational Corp. | Methods for predicting responsiveness of a cancer cell to an anti-IGFR1 antibody by analysis of mutations in PIK3CA |
| AU2011232219B2 (en) | 2010-03-23 | 2016-02-04 | Scinopharm Taiwan, Ltd. | Process and intermediates for preparing lapatinib |
| ITMI20110894A1 (it) * | 2011-05-20 | 2012-11-21 | Italiana Sint Spa | Impurezza del lapatinib e suoi sali |
| WO2014170910A1 (en) | 2013-04-04 | 2014-10-23 | Natco Pharma Limited | Process for the preparation of lapatinib |
| AU2020242287A1 (en) | 2019-03-21 | 2021-09-02 | INSERM (Institut National de la Santé et de la Recherche Médicale) | A Dbait molecule in combination with kinase inhibitor for the treatment of cancer |
| KR20220098759A (ko) | 2019-11-08 | 2022-07-12 | 인쎄름 (엥스띠뛰 나씨오날 드 라 쌍떼 에 드 라 흐쉐르슈 메디깔) | 키나제 억제제에 대해 내성을 획득한 암의 치료 방법 |
| WO2021148581A1 (en) | 2020-01-22 | 2021-07-29 | Onxeo | Novel dbait molecule and its use |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002500225A (ja) * | 1998-01-12 | 2002-01-08 | グラクソ グループ リミテッド | プロテインチロシンキナーゼ阻害剤としての二環式ヘテロ芳香族化合物 |
| JP2004533454A (ja) * | 2001-05-14 | 2004-11-04 | ノバルティス アクチエンゲゼルシャフト | ４−アミノ−５−フェニル−７−シクロブチル−ピロロ［２，３−ｄ］ピリミジン誘導体 |
| WO2005082415A2 (en) * | 2004-02-25 | 2005-09-09 | Dana Farber Cancer Institute, Inc. | Inhibitors of insulin-like growth factor receptor-1 for inhibiting tumor cell growth |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU7307101A (en) * | 2000-06-30 | 2002-01-14 | Glaxo Group Ltd | Quinazoline ditosylate salt compounds |
| EP1796711A2 (en) * | 2004-04-22 | 2007-06-20 | Oregon Health and Science University | Herstatin or intron 8-encoded domain thereof for modulating signaling mediated by igf-1 receptor and erbb receptors |
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2006
- 2006-04-13 US US12/296,972 patent/US20090203718A1/en not_active Abandoned
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2007
- 2007-04-12 WO PCT/US2007/066478 patent/WO2007121279A2/en not_active Ceased
- 2007-04-12 JP JP2009505614A patent/JP2009533472A/ja active Pending
- 2007-04-12 EP EP07781778A patent/EP2012587A2/en not_active Withdrawn
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002500225A (ja) * | 1998-01-12 | 2002-01-08 | グラクソ グループ リミテッド | プロテインチロシンキナーゼ阻害剤としての二環式ヘテロ芳香族化合物 |
| JP2004533454A (ja) * | 2001-05-14 | 2004-11-04 | ノバルティス アクチエンゲゼルシャフト | ４−アミノ−５−フェニル−７−シクロブチル−ピロロ［２，３−ｄ］ピリミジン誘導体 |
| WO2005082415A2 (en) * | 2004-02-25 | 2005-09-09 | Dana Farber Cancer Institute, Inc. | Inhibitors of insulin-like growth factor receptor-1 for inhibiting tumor cell growth |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012026511A1 (ja) * | 2010-08-27 | 2012-03-01 | 協和発酵キリン株式会社 | 医薬組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2012587A2 (en) | 2009-01-14 |
| US20090203718A1 (en) | 2009-08-13 |
| WO2007121279A3 (en) | 2008-01-03 |
| WO2007121279A2 (en) | 2007-10-25 |
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