JP2009526761A - ヘテロ二環式チオフェン化合物および使用の方法 - Google Patents
ヘテロ二環式チオフェン化合物および使用の方法 Download PDFInfo
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- JP2009526761A JP2009526761A JP2008552481A JP2008552481A JP2009526761A JP 2009526761 A JP2009526761 A JP 2009526761A JP 2008552481 A JP2008552481 A JP 2008552481A JP 2008552481 A JP2008552481 A JP 2008552481A JP 2009526761 A JP2009526761 A JP 2009526761A
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- alkyl
- aryl
- heteroaryl
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| PCT/US2007/002352 WO2008063202A2 (en) | 2006-01-30 | 2007-01-30 | Heterobicyclic thiophene compounds for the treatment of cancer |
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Cited By (9)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2010523568A (ja) * | 2007-04-05 | 2010-07-15 | アムジエン・インコーポレーテツド | オーロラキナーゼ調節物質及び使用方法 |
| WO2011162368A1 (ja) * | 2010-06-25 | 2011-12-29 | 興和株式会社 | 新規な縮合ピリジン又は縮合ピリミジン誘導体及びこれを含有する医薬 |
| JP2012525336A (ja) * | 2009-04-27 | 2012-10-22 | エラン ファーマシューティカルズ，インコーポレイテッド | α−４インテグリンのピリジノンアンタゴニスト |
| JP2013503903A (ja) * | 2009-09-03 | 2013-02-04 | アラーガン インコーポレイテッド | チロシンキナーゼモジュレーターとしての化合物 |
| WO2014038881A3 (ko) * | 2012-09-06 | 2014-05-08 | 씨제이제일제당 (주) | 피리돈 유도체를 포함하는 단백질 키나제 억제제 |
| JP2021500378A (ja) * | 2018-03-08 | 2021-01-07 | ウェルマーカー・バイオ・カンパニー・リミテッドＷｅｌｌｍａｒｋｅｒ Ｂｉｏ ＣＯ．， Ｌｔｄ． | チエノピリジン誘導体およびそれを含む医薬組成物 |
| JP2022535108A (ja) * | 2019-06-04 | 2022-08-04 | エグゼリクシス， インコーポレイテッド | キナーゼ依存性障害の処置のための化合物 |
| JP2023510296A (ja) * | 2020-01-07 | 2023-03-13 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP2023550380A (ja) * | 2020-11-24 | 2023-12-01 | チア タイ ティエンチン ファーマシューティカル グループ カンパニー リミテッド | 重水素修飾チエノピリドン化合物 |
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| BRPI0307077A2 (pt) * | 2002-01-22 | 2017-06-20 | Biomatera Inc | método para secar polímeros biodegradáveis |
| AU2006229343A1 (en) * | 2005-03-28 | 2006-10-05 | Kirin Pharma Kabushiki Kaisha | Thienopyridine derivative, or quinoline derivative, or quinazoline derivative, having c-Met autophosphorylation inhibiting potency |
| WO2008041053A2 (en) | 2005-05-20 | 2008-04-10 | Methylgene, Inc. | Inhibitors of vegf receptor and hgf receptor signaling |
| MX2007014617A (es) | 2005-05-20 | 2008-02-11 | Methylgene Inc | Inhibidores de senalizacion de receptor de factor de crecimiento endotelial bascular y receptor de factor de crecimiento de hepatocitos. |
| EP2038289A2 (en) * | 2006-04-21 | 2009-03-25 | Amgen Inc. | Thieno-[2,3-d]pyrimidine and thieno-pyridazine compounds and methods of use |
| US20110053931A1 (en) * | 2006-06-08 | 2011-03-03 | John Gaudino | Quinoline compounds and methods of use |
| ES2431466T3 (es) | 2006-06-30 | 2013-11-26 | Sunesis Pharmaceuticals, Inc. | Inhibidores de piridinonil pdk1 |
| EP2183254B1 (en) | 2007-08-29 | 2017-06-21 | MethylGene Inc. | Inhibitors of protein tyrosine kinase activity |
| WO2009026720A1 (en) | 2007-08-29 | 2009-03-05 | Methylgene Inc. | Processes and intermediates for preparing fused heterocyclic kinase inhibitors |
| ES2531396T3 (es) | 2008-01-23 | 2015-03-13 | Bristol Myers Squibb Co | Proceso para preparar compuestos de piridinona |
| PE20091624A1 (es) | 2008-03-03 | 2009-11-19 | Takeda Pharmaceutical | Farmaco combinado a base de un inhibidor de her2 derivado de pirrolopirimidina o pirazolopirimidina |
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| JP2013503903A (ja) * | 2009-09-03 | 2013-02-04 | アラーガン インコーポレイテッド | チロシンキナーゼモジュレーターとしての化合物 |
| JP5889788B2 (ja) * | 2010-06-25 | 2016-03-22 | 興和株式会社 | 新規な縮合ピリジン又は縮合ピリミジン誘導体及びこれを含有する医薬 |
| US8765771B2 (en) | 2010-06-25 | 2014-07-01 | Kowa Co., Ltd. | Condensed pyridine or condensed pyrimidine derivative, and medicinal agent comprising same |
| WO2011162368A1 (ja) * | 2010-06-25 | 2011-12-29 | 興和株式会社 | 新規な縮合ピリジン又は縮合ピリミジン誘導体及びこれを含有する医薬 |
| WO2014038881A3 (ko) * | 2012-09-06 | 2014-05-08 | 씨제이제일제당 (주) | 피리돈 유도체를 포함하는 단백질 키나제 억제제 |
| JP2021500378A (ja) * | 2018-03-08 | 2021-01-07 | ウェルマーカー・バイオ・カンパニー・リミテッドＷｅｌｌｍａｒｋｅｒ Ｂｉｏ ＣＯ．， Ｌｔｄ． | チエノピリジン誘導体およびそれを含む医薬組成物 |
| JP2022535108A (ja) * | 2019-06-04 | 2022-08-04 | エグゼリクシス， インコーポレイテッド | キナーゼ依存性障害の処置のための化合物 |
| JP7820152B2 (ja) | 2019-06-04 | 2026-02-25 | エグゼリクシス， インコーポレイテッド | キナーゼ依存性障害の処置のための化合物 |
| JP2023510296A (ja) * | 2020-01-07 | 2023-03-13 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP7434575B2 (ja) | 2020-01-07 | 2024-02-20 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP2023550380A (ja) * | 2020-11-24 | 2023-12-01 | チア タイ ティエンチン ファーマシューティカル グループ カンパニー リミテッド | 重水素修飾チエノピリドン化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2008063202A3 (en) | 2009-01-22 |
| US20070197537A1 (en) | 2007-08-23 |
| US8003662B2 (en) | 2011-08-23 |
| WO2008063202A2 (en) | 2008-05-29 |
| AR059246A1 (es) | 2008-03-19 |
| CN101522687A (zh) | 2009-09-02 |
| EP1989211A2 (en) | 2008-11-12 |
| CA2636242A1 (en) | 2008-05-29 |
| TW200806675A (en) | 2008-02-01 |
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