JP2009526761A - ヘテロ二環式チオフェン化合物および使用の方法 - Google Patents
ヘテロ二環式チオフェン化合物および使用の方法 Download PDFInfo
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- JP2009526761A JP2009526761A JP2008552481A JP2008552481A JP2009526761A JP 2009526761 A JP2009526761 A JP 2009526761A JP 2008552481 A JP2008552481 A JP 2008552481A JP 2008552481 A JP2008552481 A JP 2008552481A JP 2009526761 A JP2009526761 A JP 2009526761A
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- alkyl
- aryl
- heteroaryl
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| PCT/US2007/002352 WO2008063202A2 (en) | 2006-01-30 | 2007-01-30 | Heterobicyclic thiophene compounds for the treatment of cancer |
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| JP2009526761A true JP2009526761A (ja) | 2009-07-23 |
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| JP2010523568A (ja) * | 2007-04-05 | 2010-07-15 | アムジエン・インコーポレーテツド | オーロラキナーゼ調節物質及び使用方法 |
| WO2011162368A1 (ja) * | 2010-06-25 | 2011-12-29 | 興和株式会社 | 新規な縮合ピリジン又は縮合ピリミジン誘導体及びこれを含有する医薬 |
| JP2012525336A (ja) * | 2009-04-27 | 2012-10-22 | エラン ファーマシューティカルズ，インコーポレイテッド | α−４インテグリンのピリジノンアンタゴニスト |
| JP2013503903A (ja) * | 2009-09-03 | 2013-02-04 | アラーガン インコーポレイテッド | チロシンキナーゼモジュレーターとしての化合物 |
| WO2014038881A3 (ko) * | 2012-09-06 | 2014-05-08 | 씨제이제일제당 (주) | 피리돈 유도체를 포함하는 단백질 키나제 억제제 |
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| JP2022535108A (ja) * | 2019-06-04 | 2022-08-04 | エグゼリクシス， インコーポレイテッド | キナーゼ依存性障害の処置のための化合物 |
| JP2023510296A (ja) * | 2020-01-07 | 2023-03-13 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP2023550380A (ja) * | 2020-11-24 | 2023-12-01 | チア タイ ティエンチン ファーマシューティカル グループ カンパニー リミテッド | 重水素修飾チエノピリドン化合物 |
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| CA2473521C (en) * | 2002-01-22 | 2014-04-15 | Biomatera Inc. | Method of drying biodegradable polymers |
| AU2006229343A1 (en) * | 2005-03-28 | 2006-10-05 | Kirin Pharma Kabushiki Kaisha | Thienopyridine derivative, or quinoline derivative, or quinazoline derivative, having c-Met autophosphorylation inhibiting potency |
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| CA2608726C (en) | 2005-05-20 | 2013-07-09 | Methylgene Inc. | Inhibitors of vegf receptor and hgf receptor signaling |
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| US20110053931A1 (en) * | 2006-06-08 | 2011-03-03 | John Gaudino | Quinoline compounds and methods of use |
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| WO2009026720A1 (en) * | 2007-08-29 | 2009-03-05 | Methylgene Inc. | Processes and intermediates for preparing fused heterocyclic kinase inhibitors |
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| JP5889788B2 (ja) * | 2010-06-25 | 2016-03-22 | 興和株式会社 | 新規な縮合ピリジン又は縮合ピリミジン誘導体及びこれを含有する医薬 |
| WO2014038881A3 (ko) * | 2012-09-06 | 2014-05-08 | 씨제이제일제당 (주) | 피리돈 유도체를 포함하는 단백질 키나제 억제제 |
| JP2021500378A (ja) * | 2018-03-08 | 2021-01-07 | ウェルマーカー・バイオ・カンパニー・リミテッドＷｅｌｌｍａｒｋｅｒ Ｂｉｏ ＣＯ．， Ｌｔｄ． | チエノピリジン誘導体およびそれを含む医薬組成物 |
| JP2022535108A (ja) * | 2019-06-04 | 2022-08-04 | エグゼリクシス， インコーポレイテッド | キナーゼ依存性障害の処置のための化合物 |
| JP2023510296A (ja) * | 2020-01-07 | 2023-03-13 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP7434575B2 (ja) | 2020-01-07 | 2024-02-20 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP2023550380A (ja) * | 2020-11-24 | 2023-12-01 | チア タイ ティエンチン ファーマシューティカル グループ カンパニー リミテッド | 重水素修飾チエノピリドン化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| TW200806675A (en) | 2008-02-01 |
| WO2008063202A2 (en) | 2008-05-29 |
| AR059246A1 (es) | 2008-03-19 |
| US8003662B2 (en) | 2011-08-23 |
| EP1989211A2 (en) | 2008-11-12 |
| CN101522687A (zh) | 2009-09-02 |
| CA2636242A1 (en) | 2008-05-29 |
| US20070197537A1 (en) | 2007-08-23 |
| WO2008063202A3 (en) | 2009-01-22 |
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