JP2009520038A5 - - Google Patents

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Publication number
JP2009520038A5
JP2009520038A5 JP2008547699A JP2008547699A JP2009520038A5 JP 2009520038 A5 JP2009520038 A5 JP 2009520038A5 JP 2008547699 A JP2008547699 A JP 2008547699A JP 2008547699 A JP2008547699 A JP 2008547699A JP 2009520038 A5 JP2009520038 A5 JP 2009520038A5
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JP
Japan
Prior art keywords
alkyl
carbocycle
heterocycle
hydroxyl
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2008547699A
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English (en)
Japanese (ja)
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JP2009520038A (ja
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Publication date
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Priority claimed from PCT/US2006/062181 external-priority patent/WO2007120339A1/en
Publication of JP2009520038A publication Critical patent/JP2009520038A/ja
Publication of JP2009520038A5 publication Critical patent/JP2009520038A5/ja
Pending legal-status Critical Current

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JP2008547699A 2005-12-19 2006-12-15 ピリミジンキナーゼインヒビター Pending JP2009520038A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75201305P 2005-12-19 2005-12-19
PCT/US2006/062181 WO2007120339A1 (en) 2005-12-19 2006-12-15 Pyrimidine kinase inhibitors

Publications (2)

Publication Number Publication Date
JP2009520038A JP2009520038A (ja) 2009-05-21
JP2009520038A5 true JP2009520038A5 (https=) 2010-02-04

Family

ID=38609816

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008547699A Pending JP2009520038A (ja) 2005-12-19 2006-12-15 ピリミジンキナーゼインヒビター

Country Status (4)

Country Link
US (1) US20080318989A1 (https=)
EP (1) EP1968950A4 (https=)
JP (1) JP2009520038A (https=)
WO (1) WO2007120339A1 (https=)

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US9273077B2 (en) 2008-05-21 2016-03-01 Ariad Pharmaceuticals, Inc. Phosphorus derivatives as kinase inhibitors
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US8338439B2 (en) 2008-06-27 2012-12-25 Celgene Avilomics Research, Inc. 2,4-disubstituted pyrimidines useful as kinase inhibitors
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BR112014022790B1 (pt) 2012-03-15 2022-04-19 Celgene Car Llc Sais de um inibidor de quinase de receptor de fator do crescimento epidermal, composição farmacêutica e usos do mesmo
WO2013169401A1 (en) 2012-05-05 2013-11-14 Ariad Pharmaceuticals, Inc. Compounds for inhibiting cell proliferation in egfr-driven cancers
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US9266892B2 (en) 2012-12-19 2016-02-23 Incyte Holdings Corporation Fused pyrazoles as FGFR inhibitors
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