JP2009520038A5 - - Google Patents

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Publication number
JP2009520038A5
JP2009520038A5 JP2008547699A JP2008547699A JP2009520038A5 JP 2009520038 A5 JP2009520038 A5 JP 2009520038A5 JP 2008547699 A JP2008547699 A JP 2008547699A JP 2008547699 A JP2008547699 A JP 2008547699A JP 2009520038 A5 JP2009520038 A5 JP 2009520038A5
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JP
Japan
Prior art keywords
alkyl
carbocycle
heterocycle
hydroxyl
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2008547699A
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English (en)
Japanese (ja)
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JP2009520038A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2006/062181 external-priority patent/WO2007120339A1/en
Publication of JP2009520038A publication Critical patent/JP2009520038A/ja
Publication of JP2009520038A5 publication Critical patent/JP2009520038A5/ja
Pending legal-status Critical Current

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JP2008547699A 2005-12-19 2006-12-15 ピリミジンキナーゼインヒビター Pending JP2009520038A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75201305P 2005-12-19 2005-12-19
PCT/US2006/062181 WO2007120339A1 (en) 2005-12-19 2006-12-15 Pyrimidine kinase inhibitors

Publications (2)

Publication Number Publication Date
JP2009520038A JP2009520038A (ja) 2009-05-21
JP2009520038A5 true JP2009520038A5 (enExample) 2010-02-04

Family

ID=38609816

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008547699A Pending JP2009520038A (ja) 2005-12-19 2006-12-15 ピリミジンキナーゼインヒビター

Country Status (4)

Country Link
US (1) US20080318989A1 (enExample)
EP (1) EP1968950A4 (enExample)
JP (1) JP2009520038A (enExample)
WO (1) WO2007120339A1 (enExample)

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ES2880109T3 (es) 2012-03-15 2021-11-23 Celgene Car Llc Formas sólidas de un inhibidor de la cinasa del receptor del factor de crecimiento epidérmico
ES2698298T3 (es) 2012-03-15 2019-02-04 Celgene Car Llc Sales de un inhibidor de quinasa receptor de factor de crecimiento epidérmico
JP6469567B2 (ja) 2012-05-05 2019-02-13 アリアド・ファーマシューティカルズ・インコーポレイテッド Ｅｇｆｒ発動性がんの細胞増殖阻害用化合物
UA112897C2 (uk) 2012-05-09 2016-11-10 Байєр Фарма Акцієнгезелльшафт Біциклічно заміщені урацили та їх застосування для лікування і/або профілактики захворювань
UA125503C2 (uk) 2012-06-13 2022-04-13 Інсайт Холдинґс Корпорейшн Заміщені трициклічні сполуки як інгібітори fgfr
US9388185B2 (en) 2012-08-10 2016-07-12 Incyte Holdings Corporation Substituted pyrrolo[2,3-b]pyrazines as FGFR inhibitors
CN102827085A (zh) * 2012-09-17 2012-12-19 符爱清 2,4,5-三氯嘧啶化合物的制备方法
US9266892B2 (en) 2012-12-19 2016-02-23 Incyte Holdings Corporation Fused pyrazoles as FGFR inhibitors
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US10851105B2 (en) 2014-10-22 2020-12-01 Incyte Corporation Bicyclic heterocycles as FGFR4 inhibitors
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MA41551A (fr) 2015-02-20 2017-12-26 Incyte Corp Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4
WO2017162661A1 (en) 2016-03-22 2017-09-28 Bayer Pharma Aktiengesellschaft 1h-benzo[de]isoquinoline-1,3(2h)-diones
AR111960A1 (es) 2017-05-26 2019-09-04 Incyte Corp Formas cristalinas de un inhibidor de fgfr y procesos para su preparación
MA50250A (fr) 2017-09-15 2020-07-22 Forma Therapeutics Inc Compositions de tétrahydroimidazo quinoléine utilisées en tant qu'inhibiteurs de cbp/p300
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TW202304459A (zh) 2021-04-12 2023-02-01 美商英塞特公司 包含ｆｇｆｒ抑制劑及ｎｅｃｔｉｎ－４靶向劑之組合療法
CA3220155A1 (en) 2021-06-09 2022-12-15 Incyte Corporation Tricyclic heterocycles as fgfr inhibitors
TW202313611A (zh) 2021-06-09 2023-04-01 美商英塞特公司 作為ｆｇｆｒ抑制劑之三環雜環
CN115677595B (zh) * 2022-10-26 2024-06-14 江苏睿实生物科技有限公司 一种2,4,5-三氯嘧啶的制备方法

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MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
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