JP2009513718A5 - - Google Patents

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JP2009513718A5
JP2009513718A5 JP2008539013A JP2008539013A JP2009513718A5 JP 2009513718 A5 JP2009513718 A5 JP 2009513718A5 JP 2008539013 A JP2008539013 A JP 2008539013A JP 2008539013 A JP2008539013 A JP 2008539013A JP 2009513718 A5 JP2009513718 A5 JP 2009513718A5
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alkyl
aryl
group
compound according
trisubstituted
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JP2008539013A
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JP5241501B2 (ja
JP2009513718A (ja
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Priority claimed from PCT/US2006/042753 external-priority patent/WO2007053725A2/en
Publication of JP2009513718A publication Critical patent/JP2009513718A/ja
Publication of JP2009513718A5 publication Critical patent/JP2009513718A5/ja
Application granted granted Critical
Publication of JP5241501B2 publication Critical patent/JP5241501B2/ja
Expired - Fee Related legal-status Critical Current
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JP2008539013A 2005-11-01 2006-11-01 治療特性を有する新規の１，４−ベンゾジアゼピン−２，５−ジオン Expired - Fee Related JP5241501B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US73204505P 2005-11-01 2005-11-01
US60/732,045 2005-11-01
PCT/US2006/042753 WO2007053725A2 (en) 2005-11-01 2006-11-01 Novel 1,4-benzodiazepine-2,5-diones with therapeutic properties

Publications (3)

Publication Number Publication Date
JP2009513718A JP2009513718A (ja) 2009-04-02
JP2009513718A5 true JP2009513718A5 (OSRAM) 2011-01-06
JP5241501B2 JP5241501B2 (ja) 2013-07-17

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ID=38006506

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008539013A Expired - Fee Related JP5241501B2 (ja) 2005-11-01 2006-11-01 治療特性を有する新規の１，４−ベンゾジアゼピン−２，５−ジオン

Country Status (8)

Country Link
US (3) US8088759B2 (OSRAM)
EP (2) EP1948191B1 (OSRAM)
JP (1) JP5241501B2 (OSRAM)
AU (2) AU2006308655B2 (OSRAM)
CA (2) CA2779041A1 (OSRAM)
IL (1) IL191175A (OSRAM)
NZ (1) NZ568254A (OSRAM)
WO (1) WO2007053725A2 (OSRAM)

Families Citing this family (19)

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CA2372150C (en) 1999-04-30 2011-08-30 The Regents Of The University Of Michigan Therapeutic applications of pro-apoptotic benzodiazepines
AU2006203946B2 (en) 2005-01-03 2009-07-23 The Regents Of The University Of Michigan Compositions and methods relating to novel compounds and targets thereof
JP2008545757A (ja) 2005-06-01 2008-12-18 ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン 溶媒和されていないベンゾジアゼピン組成物および方法
EP1948191B1 (en) 2005-11-01 2013-01-16 The Regents of the University of Michigan Novel 1,4-benzodiazepine-2,5-diones with therapeutic properties
US7759338B2 (en) * 2006-04-27 2010-07-20 The Regents Of The University Of Michigan Soluble 1,4 benzodiazepine compounds and stable salts thereof
EP2418206A3 (en) 2006-06-09 2012-06-27 The Regents of the University of Michigan Benzodiazepine derivatives useful in the treatment of autoimmune disorders
JP5383513B2 (ja) 2007-03-09 2014-01-08 ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン 化合物およびその標的に関連する組成物ならびに方法
WO2009036175A2 (en) 2007-09-14 2009-03-19 The Regents Of The University Of Michigan F1f0-atpase inhibitors and related methods
AU2008323945B2 (en) 2007-11-06 2013-11-28 The Regents Of The University Of Michigan Benzodiazepinone compounds useful in the treatment of skin conditions
US8497307B2 (en) 2008-09-11 2013-07-30 The Regents Of The University Of Michigan Aryl guanidine F1F0-ATPase inhibitors and related methods
US8604023B2 (en) 2009-04-17 2013-12-10 The Regents Of The University Of Michigan 1,4-benzodiazepinone compounds and their use in treating cancer
CN102712643B (zh) 2009-05-22 2015-12-16 Abbvie公司 5-ht受体的调节剂及其使用方法
JP2013505258A (ja) 2009-09-18 2013-02-14 ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン ベンゾジアゼピノン化合物およびそれを使用する治療方法
CN102753544A (zh) * 2009-11-17 2012-10-24 密执安大学评议会 具有治疗性能的1，4-苯并二氮杂*-2，5-二酮和相关化合物
JP5856063B2 (ja) * 2009-11-17 2016-02-09 ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン 治療特性を有する１，４−ベンゾジアゼピン−２，５−ジオンおよび関連化合物
KR101770979B1 (ko) 2010-05-21 2017-08-24 애브비 인코포레이티드 5­ｈｔ 수용체의 조절제 및 이의 사용방법
CN111529534A (zh) 2012-09-27 2020-08-14 儿童医学中心公司 用于治疗肥胖症的化合物和其使用方法
CN103435562B (zh) * 2013-08-26 2016-02-24 华东理工大学 6-取代苯并二氮卓-2,4-二酮类化合物及其用途
CN105693634B (zh) * 2016-03-17 2018-12-11 清华大学 化合物及其用途

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