JP2009507073A - 子宮内膜症の治療のためのｉｋｋ阻害剤 - Google Patents
子宮内膜症の治療のためのｉｋｋ阻害剤 Download PDFInfo
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- JP2009507073A JP2009507073A JP2008530093A JP2008530093A JP2009507073A JP 2009507073 A JP2009507073 A JP 2009507073A JP 2008530093 A JP2008530093 A JP 2008530093A JP 2008530093 A JP2008530093 A JP 2008530093A JP 2009507073 A JP2009507073 A JP 2009507073A
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Landscapes
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| EP2303841A1 (en) | 2008-07-14 | 2011-04-06 | Gilead Sciences, Inc. | Oxindolyl inhibitor compounds |
| EP2303881A2 (en) | 2008-07-14 | 2011-04-06 | Gilead Sciences, Inc. | Fused heterocyclyc inhibitors of histone deacetylase and/or cyclin-dependent kinases |
| JP5640005B2 (ja) | 2008-07-14 | 2014-12-10 | ギリアード サイエンシーズ， インコーポレイテッド | Ｈｄａｃおよび／またはｃｄｋ阻害剤としてのイミダゾシルピリジン化合物 |
| KR20110038159A (ko) | 2008-07-28 | 2011-04-13 | 길리애드 사이언시즈, 인코포레이티드 | 사이클로알킬리덴 및 헤테로사이클로알킬리덴 히스톤 데아세틸라아제 억제제 화합물 |
| CN101503402B (zh) * | 2009-03-10 | 2014-06-25 | 沈阳药科大学 | 2-苯胺嘧啶衍生物及其制备和用途 |
| CA2763786C (en) | 2009-06-08 | 2014-09-30 | Gilead Sciences, Inc. | Alkanoylamino benzamide aniline hdac inihibitor compounds |
| ES2463826T3 (es) | 2009-06-08 | 2014-05-29 | Gilead Sciences, Inc. | Compuestos inhibidores de HDAC de cicloalquilcarbamato benzamida anilina |
| CN105132529A (zh) | 2009-07-24 | 2015-12-09 | 吉第克生物技术有限公司 | 子宫内膜癌的标记物 |
| AU2011260323A1 (en) | 2010-06-04 | 2012-11-15 | F. Hoffmann-La Roche Ag | Aminopyrimidine derivatives as LRRK2 modulators |
| KR101566091B1 (ko) | 2010-11-10 | 2015-11-04 | 에프. 호프만-라 로슈 아게 | Lrrk2 조절제로서 피라졸 아미노피리미딘 유도체 |
| WO2019169113A1 (en) * | 2018-03-02 | 2019-09-06 | Ponce Medical School Foundation, Inc. | Compositions and methods for the treatment of endometriosis |
| US11066404B2 (en) | 2018-10-11 | 2021-07-20 | Incyte Corporation | Dihydropyrido[2,3-d]pyrimidinone compounds as CDK2 inhibitors |
| WO2020168197A1 (en) | 2019-02-15 | 2020-08-20 | Incyte Corporation | Pyrrolo[2,3-d]pyrimidinone compounds as cdk2 inhibitors |
| TW202100520A (zh) | 2019-03-05 | 2021-01-01 | 美商英塞特公司 | 作為cdk2 抑制劑之吡唑基嘧啶基胺化合物 |
| US11919904B2 (en) | 2019-03-29 | 2024-03-05 | Incyte Corporation | Sulfonylamide compounds as CDK2 inhibitors |
| WO2020223558A1 (en) | 2019-05-01 | 2020-11-05 | Incyte Corporation | Tricyclic amine compounds as cdk2 inhibitors |
| WO2020223469A1 (en) | 2019-05-01 | 2020-11-05 | Incyte Corporation | N-(1-(methylsulfonyl)piperidin-4-yl)-4,5-di hydro-1h-imidazo[4,5-h]quinazolin-8-amine derivatives and related compounds as cyclin-dependent kinase 2 (cdk2) inhibitors for treating cancer |
| WO2021030537A1 (en) | 2019-08-14 | 2021-02-18 | Incyte Corporation | Imidazolyl pyrimidinylamine compounds as cdk2 inhibitors |
| CR20220170A (es) | 2019-10-11 | 2022-10-10 | Incyte Corp | Aminas bicíclicas como inhibidoras de la cdk2 |
| US11981671B2 (en) | 2021-06-21 | 2024-05-14 | Incyte Corporation | Bicyclic pyrazolyl amines as CDK2 inhibitors |
| US11976073B2 (en) | 2021-12-10 | 2024-05-07 | Incyte Corporation | Bicyclic amines as CDK2 inhibitors |
| CN119769990B (zh) * | 2024-12-26 | 2025-09-09 | 大连医科大学附属第二医院 | 子宫内膜异位症的检测系统和治疗剂 |
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| JP2004523497A (ja) * | 2000-12-06 | 2004-08-05 | シグナル ファーマシューティカルズ， インコーポレイテッド | Ｉｋｋ阻害剤としてのアニリノピリミジン誘導体ならびにそれに関する組成物および方法 |
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| US4923805A (en) | 1983-11-02 | 1990-05-08 | Integrated Genetics, Inc. | Fsh |
| DE10199028I2 (de) | 1983-11-02 | 2004-07-01 | Applied Research Systems | Produkte und Methoden für die Herstellung einer heterodimerer menschlicher LH mit einem Met42 Val55 alpha Untereinheit. |
| IT1206302B (it) | 1987-06-26 | 1989-04-14 | Serono Cesare Ist Ricerca | Ormone follicolo-stimolante urinario |
| JP2002193938A (ja) * | 2000-12-01 | 2002-07-10 | Bayer Ag | ４−アリールピリジン誘導体 |
| US20030134836A1 (en) * | 2001-01-12 | 2003-07-17 | Amgen Inc. | Substituted arylamine derivatives and methods of use |
| CZ20032287A3 (cs) * | 2001-02-01 | 2004-02-18 | Bristol-Myers Squibb Company | Způsoby léčení zánětlivých a imunitních nemocí za použití inhibitorů IkB kinázy (IKK) |
| SE0102616D0 (sv) * | 2001-07-25 | 2001-07-25 | Astrazeneca Ab | Novel compounds |
| WO2003015820A1 (en) * | 2001-08-10 | 2003-02-27 | Takeda Chemical Industries, Ltd. | GnRH AGONIST COMBINATION DRUGS |
| DE10237722A1 (de) | 2002-08-17 | 2004-08-19 | Aventis Pharma Deutschland Gmbh | Indol- oder Benzimidazolderivate zur Modulation der IKappaB-Kinase |
| WO2004048343A1 (en) * | 2002-11-28 | 2004-06-10 | Schering Aktiengesellschaft | Chk-, pdk- and akt-inhibitory pyrimidines, their production and use as pharmaceutical agents |
| EP1670908A2 (en) * | 2003-10-02 | 2006-06-21 | Xantos Biomedicine AG | Medical use of tbk-1 or of inhibitors thereof |
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- 2006-08-28 EA EA200800755A patent/EA200800755A1/ru unknown
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- 2006-08-28 CA CA002621057A patent/CA2621057A1/en not_active Abandoned
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- 2006-08-28 EP EP10184024A patent/EP2266561A3/en not_active Withdrawn
- 2006-08-28 JP JP2008530093A patent/JP2009507073A/ja active Pending
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Patent Citations (1)
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| JP2004523497A (ja) * | 2000-12-06 | 2004-08-05 | シグナル ファーマシューティカルズ， インコーポレイテッド | Ｉｋｋ阻害剤としてのアニリノピリミジン誘導体ならびにそれに関する組成物および方法 |
Also Published As
| Publication number | Publication date |
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| US20100069387A1 (en) | 2010-03-18 |
| EP2266561A3 (en) | 2011-05-18 |
| EA200800755A1 (ru) | 2008-10-30 |
| KR20080052650A (ko) | 2008-06-11 |
| AU2006287767A1 (en) | 2007-03-15 |
| EP1931322A1 (en) | 2008-06-18 |
| EP1931322B1 (en) | 2012-08-15 |
| IL189659A0 (en) | 2008-08-07 |
| WO2007030362A1 (en) | 2007-03-15 |
| AU2006287767B2 (en) | 2010-05-13 |
| CN101304736A (zh) | 2008-11-12 |
| EP2266561A2 (en) | 2010-12-29 |
| CA2621057A1 (en) | 2007-03-15 |
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