JP2008545782A5 - - Google Patents

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Publication number
JP2008545782A5
JP2008545782A5 JP2008515848A JP2008515848A JP2008545782A5 JP 2008545782 A5 JP2008545782 A5 JP 2008545782A5 JP 2008515848 A JP2008515848 A JP 2008515848A JP 2008515848 A JP2008515848 A JP 2008515848A JP 2008545782 A5 JP2008545782 A5 JP 2008545782A5
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JP
Japan
Prior art keywords
methyl
process according
imidazole
trifluoromethyl
nitro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2008515848A
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English (en)
Japanese (ja)
Other versions
JP5139273B2 (ja
JP2008545782A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2006/022026 external-priority patent/WO2006135619A1/en
Publication of JP2008545782A publication Critical patent/JP2008545782A/ja
Publication of JP2008545782A5 publication Critical patent/JP2008545782A5/ja
Application granted granted Critical
Publication of JP5139273B2 publication Critical patent/JP5139273B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2008515848A 2005-06-09 2006-06-07 5−(4−メチル−1h−イミダゾール−1−イル)−3−(トリフルオロメチル)−ベンゼンアミンの合成法 Expired - Fee Related JP5139273B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US68892005P 2005-06-09 2005-06-09
US60/688,920 2005-06-09
PCT/US2006/022026 WO2006135619A1 (en) 2005-06-09 2006-06-07 Process for the synthesis of 5- (methyl- 1h-imidazol-1-yl) -3- (trifluoromethyl) -benzeneamine

Publications (3)

Publication Number Publication Date
JP2008545782A JP2008545782A (ja) 2008-12-18
JP2008545782A5 true JP2008545782A5 (https=) 2009-07-23
JP5139273B2 JP5139273B2 (ja) 2013-02-06

Family

ID=37085334

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008515848A Expired - Fee Related JP5139273B2 (ja) 2005-06-09 2006-06-07 5−(4−メチル−1h−イミダゾール−1−イル)−3−(トリフルオロメチル)−ベンゼンアミンの合成法

Country Status (20)

Country Link
US (1) US7709657B2 (https=)
EP (1) EP1896425B1 (https=)
JP (1) JP5139273B2 (https=)
KR (1) KR101319071B1 (https=)
CN (1) CN101193866B (https=)
AR (1) AR057351A1 (https=)
AT (1) ATE483690T1 (https=)
AU (1) AU2006258116B2 (https=)
BR (1) BRPI0611924A2 (https=)
CA (1) CA2610402C (https=)
DE (1) DE602006017369D1 (https=)
ES (1) ES2354115T3 (https=)
GT (1) GT200600207A (https=)
MX (1) MX2007015420A (https=)
PE (1) PE20070084A1 (https=)
PL (1) PL1896425T3 (https=)
PT (1) PT1896425E (https=)
RU (1) RU2404167C2 (https=)
TW (1) TW200710084A (https=)
WO (1) WO2006135619A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY146795A (en) * 2005-06-09 2012-09-28 Novartis Ag Process for the synthesis of organic compounds
GB0618832D0 (en) * 2006-09-25 2006-11-01 Phoenix Chemicals Ltd Chemical process
US20110053968A1 (en) * 2009-06-09 2011-03-03 Auspex Pharmaceuticals, Inc. Aminopyrimidine inhibitors of tyrosine kinase
EP3144194B1 (en) 2014-05-16 2018-05-09 Robert Bosch GmbH Abs hydraulic unit
KR102335216B1 (ko) 2017-04-26 2021-12-03 삼성전자 주식회사 발광소자 패키지
CN107235910B (zh) * 2017-07-31 2020-04-24 安礼特(上海)医药科技有限公司 一种尼洛胺的合成方法
CN108530364B (zh) 2018-04-10 2020-01-21 江苏创诺制药有限公司 一种3-(4-甲基-1h-咪唑-1-基)-5-三氟甲基苯胺单盐酸盐的晶型及其应用
TWI831259B (zh) 2018-06-15 2024-02-01 漢達生技醫藥股份有限公司 包含達沙替尼十二烷基硫酸鹽組合物的膠囊
EP3904342A1 (en) 2020-04-28 2021-11-03 Grindeks, A Joint Stock Company Process for the preparation of 3-(trifluoromethyl)-5-(4-methyl-1h-imidazole-1-yl)-benzeneamine hydrochloride

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8413685D0 (en) * 1984-05-29 1984-07-04 Pfizer Ltd Quinolone inotropic agents
US5516775A (en) * 1992-08-31 1996-05-14 Ciba-Geigy Corporation Further use of pyrimidine derivatives
PT672041E (pt) * 1993-10-01 2002-04-29 Novartis Ag Derivados da piridina farmacologicamente activos e processos para a sua preparacao
US6323366B1 (en) 1997-07-29 2001-11-27 Massachusetts Institute Of Technology Arylamine synthesis
US6395916B1 (en) 1998-07-10 2002-05-28 Massachusetts Institute Of Technology Ligands for metals and improved metal-catalyzed processes based thereon
HN2001000008A (es) * 2000-01-21 2003-12-11 Inc Agouron Pharmaceuticals Compuesto de amida y composiciones farmaceuticas para inhibir proteinquinasas, y su modo de empleo
PE20040522A1 (es) * 2002-05-29 2004-09-28 Novartis Ag Derivados de diarilurea dependientes de la cinasa de proteina
US7202367B2 (en) 2002-05-31 2007-04-10 Rhodia Chimie Process for arylating or vinylating or alkynating a nucleophilic compound
GB0215676D0 (en) 2002-07-05 2002-08-14 Novartis Ag Organic compounds

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