JP2008525477A5 - - Google Patents

Download PDF

Info

Publication number
JP2008525477A5
JP2008525477A5 JP2007548473A JP2007548473A JP2008525477A5 JP 2008525477 A5 JP2008525477 A5 JP 2008525477A5 JP 2007548473 A JP2007548473 A JP 2007548473A JP 2007548473 A JP2007548473 A JP 2007548473A JP 2008525477 A5 JP2008525477 A5 JP 2008525477A5
Authority
JP
Japan
Prior art keywords
glp
seq
polypeptide
formulation
deleted mimetibody
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2007548473A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008525477A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/046602 external-priority patent/WO2007046834A2/en
Publication of JP2008525477A publication Critical patent/JP2008525477A/ja
Publication of JP2008525477A5 publication Critical patent/JP2008525477A5/ja
Pending legal-status Critical Current

Links

JP2007548473A 2004-12-22 2005-12-22 Glp−1アゴニスト、組成物、方法および使用 Pending JP2008525477A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63831304P 2004-12-22 2004-12-22
PCT/US2005/046602 WO2007046834A2 (en) 2004-12-22 2005-12-22 Glp-1 agonists, compositions, methods and uses

Publications (2)

Publication Number Publication Date
JP2008525477A JP2008525477A (ja) 2008-07-17
JP2008525477A5 true JP2008525477A5 (https=) 2009-02-12

Family

ID=37962937

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007548473A Pending JP2008525477A (ja) 2004-12-22 2005-12-22 Glp−1アゴニスト、組成物、方法および使用

Country Status (17)

Country Link
US (1) US20070128193A1 (https=)
EP (1) EP1843788A4 (https=)
JP (1) JP2008525477A (https=)
KR (1) KR20070090036A (https=)
CN (1) CN101415439A (https=)
AU (1) AU2005337493A1 (https=)
BR (1) BRPI0519241A2 (https=)
CA (1) CA2592065A1 (https=)
CR (1) CR9266A (https=)
EA (1) EA200701362A1 (https=)
IL (1) IL183940A0 (https=)
MX (1) MX2007007602A (https=)
NI (1) NI200700158A (https=)
NO (1) NO20073814L (https=)
SG (1) SG158158A1 (https=)
WO (1) WO2007046834A2 (https=)
ZA (1) ZA200706030B (https=)

Families Citing this family (56)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9006175B2 (en) 1999-06-29 2015-04-14 Mannkind Corporation Potentiation of glucose elimination
WO2003080149A2 (en) 2002-03-20 2003-10-02 Mannkind Corporation Inhalation apparatus
PL1786784T3 (pl) 2004-08-20 2011-04-29 Mannkind Corp Kataliza syntezy diketopiperazyn
KR101644250B1 (ko) 2004-08-23 2016-07-29 맨카인드 코포레이션 약물 전달용 디케토피페라진염, 디케토모르포린염 또는 디케토디옥산염
US20090305964A1 (en) * 2005-04-21 2009-12-10 Gastrotech Pharma A/S Pharmaceutical preparations of a glp-1 molecule and an anti-emetic drug
CN104324362B (zh) 2005-09-14 2018-04-24 曼金德公司 以提高活性试剂对结晶微粒表面的亲和力为基础的药物配制方法
US20070148140A1 (en) * 2005-12-28 2007-06-28 Zoltan Laboratories Llc Compositions and methods to enhance viability and function of islet cells
IN2015DN00888A (https=) 2006-02-22 2015-07-10 Mannkind Corp
AR064623A1 (es) * 2006-12-21 2009-04-15 Centocor Inc Uso de agonistas del receptor de glp -1 de accion prolongada para mejorar la sensibilidad a la insulina y los perfiles lipidicos
WO2008092209A1 (en) * 2007-02-01 2008-08-07 Arana Therapeutics Limited Protein construct with improved properties
US8485180B2 (en) 2008-06-13 2013-07-16 Mannkind Corporation Dry powder drug delivery system
ES2929343T3 (es) 2008-06-13 2022-11-28 Mannkind Corp Inhalador de polvo seco accionado por aspiración para la administración de fármacos
KR101628410B1 (ko) 2008-06-20 2016-06-08 맨카인드 코포레이션 흡입 활동에 관한 실시간 프로파일링을 위한 대화형 장치 및 방법
TWI614024B (zh) 2008-08-11 2018-02-11 曼凱公司 超快起作用胰島素之用途
MX2011003277A (es) * 2008-10-14 2012-09-21 Salubrious Pharmaceuticals LLC Proceso para el tratamiento de la artritis reumatoide, temblores/enfermedad de parkinson, esclerosis multiple y cancer de tipo no viral.
RS59913B1 (sr) 2008-10-17 2020-03-31 Sanofi Aventis Deutschland Kombinacija insulina i glp-1-agonista
PT2373681T (pt) 2008-12-10 2017-04-11 Glaxosmithkline Llc Composições farmacêuticas de albiglutida
US8314106B2 (en) 2008-12-29 2012-11-20 Mannkind Corporation Substituted diketopiperazine analogs for use as drug delivery agents
DK2405963T3 (da) 2009-03-11 2013-12-16 Mannkind Corp Apparat, system og fremgangsmåde til at måle modstand i en inhalator
CN104721825B (zh) 2009-06-12 2019-04-12 曼金德公司 具有确定比表面积的二酮哌嗪颗粒
CN102596175A (zh) 2009-07-06 2012-07-18 赛诺菲-安万特德国有限公司 含有甲硫氨酸的水性胰岛素制备物
WO2011056889A1 (en) 2009-11-03 2011-05-12 Mannkind Corporation An apparatus and method for simulating inhalation efforts
MY180661A (en) 2009-11-13 2020-12-04 Sanofi Aventis Deutschland Pharmaceutical composition comprising a glp-1 agonist, an insulin and methionine
PT3345593T (pt) 2009-11-13 2023-11-27 Sanofi Aventis Deutschland Composição farmacêutica compreendendo despro36exendina- 4(1-39)-lys6-nh2 e metionina
US8691763B2 (en) 2010-05-04 2014-04-08 Glaxosmithkline Llc Methods for treating or preventing cardiovascular disorders and providing cardiovascular protection
MX2012013001A (es) 2010-05-13 2013-02-26 Univ Indiana Res & Tech Corp Peptidos de la superfamilia de glucagon que presentan actividad del receptor nuclear de hormonas.
AU2011202239C1 (en) 2010-05-19 2017-03-16 Sanofi Long-acting formulations of insulins
IL223742A (en) 2010-06-21 2016-06-30 Mannkind Corp A dry powder inhaler and preparation for it
EP2588126A4 (en) 2010-06-24 2015-07-08 Univ Indiana Res & Tech Corp AMID-BASED GLUCAGON SUPERFAMILY PEPTIDE PRODRUGS
PL2611458T3 (pl) 2010-08-30 2017-02-28 Sanofi-Aventis Deutschland Gmbh Zastosowanie AVE0010 do produkcji leku do leczenia cukrzycy typu 2
WO2012098187A1 (en) * 2011-01-19 2012-07-26 Novo Nordisk A/S Glp-1 compositions
AU2012236150B2 (en) 2011-04-01 2016-03-31 Mannkind Corporation Blister package for pharmaceutical cartridges
US9821032B2 (en) 2011-05-13 2017-11-21 Sanofi-Aventis Deutschland Gmbh Pharmaceutical combination for improving glycemic control as add-on therapy to basal insulin
WO2012174472A1 (en) 2011-06-17 2012-12-20 Mannkind Corporation High capacity diketopiperazine microparticles
US9950038B2 (en) 2011-08-05 2018-04-24 The Trustees Of The Universiy Of Pennsylvania Methods and compositions for inhibiting delayed graft function
AR087693A1 (es) 2011-08-29 2014-04-09 Sanofi Aventis Deutschland Combinacion farmaceutica para uso en el control glucemico en pacientes con diabetes de tipo 2
TWI559929B (en) 2011-09-01 2016-12-01 Sanofi Aventis Deutschland Pharmaceutical composition for use in the treatment of a neurodegenerative disease
BR112014009686A2 (pt) 2011-10-24 2018-08-07 Mannkind Corp composição analgésica inalável, pó seco e método para tratar dor
JP6324315B2 (ja) 2011-11-17 2018-05-16 インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションIndiana University Research And Technology Corporation グルココルチコイド受容体の活性を示すグルカゴンスーパーファミリーのペプチド
WO2013128450A1 (en) * 2012-03-01 2013-09-06 Yeda Research And Development Co. Ltd. Hsp60 derived peptides and peptide analogs for suppression and treatment of non-autoimmune diabetes
CN104619369B (zh) 2012-07-12 2018-01-30 曼金德公司 干粉药物输送系统和方法
US10159644B2 (en) 2012-10-26 2018-12-25 Mannkind Corporation Inhalable vaccine compositions and methods
AU2014228415B2 (en) 2013-03-15 2018-08-09 Mannkind Corporation Microcrystalline diketopiperazine compositions and methods
UA117480C2 (uk) 2013-04-03 2018-08-10 Санофі Лікування цукрового діабету за допомогою складу інсуліну тривалої дії
MX375448B (es) 2013-07-18 2025-03-06 Mannkind Corp Composiciones farmacéuticas en polvo seco estables al calor y métodos.
US11446127B2 (en) 2013-08-05 2022-09-20 Mannkind Corporation Insufflation apparatus and methods
US10307464B2 (en) 2014-03-28 2019-06-04 Mannkind Corporation Use of ultrarapid acting insulin
US10561806B2 (en) 2014-10-02 2020-02-18 Mannkind Corporation Mouthpiece cover for an inhaler
EP3229828B1 (en) 2014-12-12 2023-04-05 Sanofi-Aventis Deutschland GmbH Insulin glargine/lixisenatide fixed ratio formulation
TWI748945B (zh) 2015-03-13 2021-12-11 德商賽諾菲阿凡提斯德意志有限公司 第2型糖尿病病患治療
TW201705975A (zh) 2015-03-18 2017-02-16 賽諾菲阿凡提斯德意志有限公司 第2型糖尿病病患之治療
WO2016174130A1 (en) * 2015-04-28 2016-11-03 Université De Strasbourg Clinical gene signature-based human cell culture model and uses thereof
CN105504026B (zh) * 2015-12-24 2018-12-07 广东医科大学 一种pac1-r和glp-1r的双向激动剂ot23及应用
EP3470424B1 (en) * 2016-06-08 2025-04-23 Shanghai Jiao Tong University School of Medicine Sequence of antibody heavy chain constant region for enhancing agonist antibody activity
TWI829687B (zh) 2018-05-07 2024-01-21 丹麥商諾佛 儂迪克股份有限公司 包含glp-1促效劑與n-(8-(2-羥基苯甲醯基)胺基)辛酸之鹽的固體組成物
AU2021285138A1 (en) 2020-06-03 2023-02-02 Københavns Universitet GLP1R agonist NMDAR antagonist conjugates

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5614492A (en) * 1986-05-05 1997-03-25 The General Hospital Corporation Insulinotropic hormone GLP-1 (7-36) and uses thereof
IL155812A0 (en) * 2000-12-07 2003-12-23 Lilly Co Eli Glp-1 fusion proteins
US20020187926A1 (en) * 2001-03-07 2002-12-12 Knudsen Liselotte Bjerre Combined use of derivatives of GLP-1 analogs and PPAR ligands
US7241733B2 (en) * 2002-06-28 2007-07-10 Centocor, Inc. Mammalian EPO mimetic CH1 deleted mimetibodies, compositions, methods and uses
US20070135338A1 (en) * 2004-03-31 2007-06-14 Karyn O'neil Human GLP-1 mimetibodies, compositions, methods and uses

Similar Documents

Publication Publication Date Title
JP2008525477A5 (https=)
ES2875748T3 (es) Nuevos derivados de oxintomodulina y composición farmacéutica para el tratamiento de la obesidad que los comprende
ES2646545T3 (es) Métodos y composiciones basadas en conjugados de toxina diftérica-interleucina-3
JP6200025B2 (ja) 心臓病の処置
US10786551B2 (en) Use of interleukin-22 in the treatment of fatty liver disease
ES2897732T3 (es) Composición para tratar la diabetes mellitus que comprende insulina y un agonista doble de glp-1/glucagón
ES2732291T3 (es) Péptidos terapéuticos
JP2006515351A5 (https=)
JP2007508011A5 (https=)
US20180280480A1 (en) Compositions and peptides having dual glp-1r and glp-2r agonist activity
MX2014013319A (es) Análogos de péptido-2 tipo glucagón (glp-2).
JPWO2015147240A1 (ja) 敗血症の予防治療剤
TW201934571A (zh) Fgf21變體、融合蛋白及其應用
RU2013139651A (ru) Новые соединения, влияющие на пищевое поведение
TW200843794A (en) Use of long-acting GLP-1 receptor agonists to improve insulin sensitivity and lipid profiles
ES2970116T3 (es) Composición farmacéutica para tratar la sarcopenia agonista del receptor del péptido de tipo 1 similar al glucagón
CN101466399B (zh) 稳定的胰岛素样生长因子多肽
JP2020533302A (ja) 肥満の治療において使用するためのmic−1およびglp−1
CN108697768A (zh) 长效glp-1r激动剂作为神经系统病状和神经退行性病状的治疗方法
CN1655675A (zh) 利用三叶肽的联合治疗
JP2009526750A5 (https=)
JP2011517548A5 (https=)
TWI496579B (zh) 類鋅手指胜肽、其表現質體、及包含其之醫藥組成物之用途
JP2021505656A (ja) グルカゴン様ペプチド
US20170071912A1 (en) Polyamide Compound and Pharmaceutical Composition for Treating Mitochondrial Genetic Diseases