JP2008523091A5 - - Google Patents

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Publication number
JP2008523091A5
JP2008523091A5 JP2007545664A JP2007545664A JP2008523091A5 JP 2008523091 A5 JP2008523091 A5 JP 2008523091A5 JP 2007545664 A JP2007545664 A JP 2007545664A JP 2007545664 A JP2007545664 A JP 2007545664A JP 2008523091 A5 JP2008523091 A5 JP 2008523091A5
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JP
Japan
Prior art keywords
alkyl
aryl
group
heteroaryl
haloalkyl
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JP2007545664A
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English (en)
Japanese (ja)
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JP2008523091A (ja
JP4960254B2 (ja
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Priority claimed from PCT/US2005/044613 external-priority patent/WO2006065646A1/en
Publication of JP2008523091A publication Critical patent/JP2008523091A/ja
Publication of JP2008523091A5 publication Critical patent/JP2008523091A5/ja
Application granted granted Critical
Publication of JP4960254B2 publication Critical patent/JP4960254B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2007545664A 2004-12-13 2005-12-07 バニロイド受容体サブタイプ1(vr1)に対するアンタゴニストとして作用するベンズイソチアゾール−1,1−ジオキシドおよびこれらの使用 Expired - Fee Related JP4960254B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US63549104P 2004-12-13 2004-12-13
US60/635,491 2004-12-13
PCT/US2005/044613 WO2006065646A1 (en) 2004-12-13 2005-12-07 Benzisothiazole-1, 1-dioxide acting as antagonists to the vanilloid receptor subtype 1 (vr1) and uses thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012001109A Division JP2012121887A (ja) 2004-12-13 2012-01-06 バニロイド受容体サブタイプ1(vr1)に対するアンタゴニストとして作用するベンズイソチアゾール−1,1−ジオキシドおよびこれらの使用

Publications (3)

Publication Number Publication Date
JP2008523091A JP2008523091A (ja) 2008-07-03
JP2008523091A5 true JP2008523091A5 (enExample) 2011-10-06
JP4960254B2 JP4960254B2 (ja) 2012-06-27

Family

ID=36129676

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2007545664A Expired - Fee Related JP4960254B2 (ja) 2004-12-13 2005-12-07 バニロイド受容体サブタイプ1(vr1)に対するアンタゴニストとして作用するベンズイソチアゾール−1,1−ジオキシドおよびこれらの使用
JP2012001109A Pending JP2012121887A (ja) 2004-12-13 2012-01-06 バニロイド受容体サブタイプ1(vr1)に対するアンタゴニストとして作用するベンズイソチアゾール−1,1−ジオキシドおよびこれらの使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2012001109A Pending JP2012121887A (ja) 2004-12-13 2012-01-06 バニロイド受容体サブタイプ1(vr1)に対するアンタゴニストとして作用するベンズイソチアゾール−1,1−ジオキシドおよびこれらの使用

Country Status (6)

Country Link
US (1) US7615570B2 (enExample)
EP (1) EP1836200B1 (enExample)
JP (2) JP4960254B2 (enExample)
CA (1) CA2591069A1 (enExample)
MX (1) MX2007007100A (enExample)
WO (1) WO2006065646A1 (enExample)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7615570B2 (en) * 2004-12-13 2009-11-10 Abbott Laboratories Antagonists to the vanilloid receptor subtype 1 (VR1) and uses thereof
JP2009506988A (ja) * 2005-08-19 2009-02-19 エラン ファーマシューティカルズ,インコーポレイテッド ガンマセクレターゼの架橋n−環状スルホンアミド阻害剤
BRPI0710507A2 (pt) * 2006-04-18 2011-08-16 Abbott Lab Antagonistas do receptor vanilóide de subtipo 1 (vr1) e usos destes
ATE549325T1 (de) * 2007-01-26 2012-03-15 Basf Se 3-amino-1,2-benzisothiazol-verbindungen zur bekämpfung von tierpest ii
SI2349263T1 (sl) 2008-10-23 2014-09-30 Vertex Pharmaceuticals Incorporated Modulatorji cistiäśno-fibroznega transmembranskega regulatorja prevodnosti
US8349852B2 (en) 2009-01-13 2013-01-08 Novartis Ag Quinazolinone derivatives useful as vanilloid antagonists
CN102762572A (zh) 2010-02-01 2012-10-31 诺瓦提斯公司 作为CRF-1受体拮抗剂的吡唑并[5,1b]*唑衍生物
WO2011092293A2 (en) 2010-02-01 2011-08-04 Novartis Ag Cyclohexyl amide derivatives as crf receptor antagonists
US8835444B2 (en) 2010-02-02 2014-09-16 Novartis Ag Cyclohexyl amide derivatives as CRF receptor antagonists
CN102718701B (zh) 2011-03-30 2014-05-07 中国中化股份有限公司 芳氧基二卤丙烯醚类化合物与应用
KR20160005356A (ko) * 2013-05-07 2016-01-14 더 리젠츠 오브 더 유니버시티 오브 캘리포니아 방사선완화 약제학적 제형
CN105707076B (zh) * 2014-12-05 2018-12-14 沈阳中化农药化工研发有限公司 除草组合物及应用
WO2019185413A1 (en) 2018-03-27 2019-10-03 Basf Se Pesticidal substituted cyclopropyl derivatives
CN113264900B (zh) * 2021-06-07 2023-05-26 南京中医药大学 一种苯并异噻唑和苯并噻吩的制备方法及其医药用途

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US473692A (en) * 1892-04-26 Rington
US4147698A (en) * 1978-07-13 1979-04-03 E. R. Squibb & Sons, Inc. 3-(Heterocyclicalkylamino)benzisothiazole-1,1-dioxides
US4166910A (en) * 1978-07-13 1979-09-04 E. R. Squibb & Sons, Inc. 3-(Nitrogen containing heterocyclic)amino) benzisothiazole-1,1-dioxide
US4743692A (en) * 1986-09-30 1988-05-10 American Home Products Corporation N-(pyridinylalkyl)-thieno-or benzo-isothiazol-3-amine derivatives
JP2006526660A (ja) 2003-06-05 2006-11-24 バーテックス ファーマシューティカルズ インコーポレイテッド Vr1レセプターのモジュレーター
CA2531515A1 (en) 2003-07-10 2005-02-03 Neurogen Corporation Aryl-substituted benzo[d]isothiazol-3-ylamine analogues as capsaicin receptor modulators
US7615570B2 (en) * 2004-12-13 2009-11-10 Abbott Laboratories Antagonists to the vanilloid receptor subtype 1 (VR1) and uses thereof

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