JP2004131511A5 - - Google Patents
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- Publication number
- JP2004131511A5 JP2004131511A5 JP2004017703A JP2004017703A JP2004131511A5 JP 2004131511 A5 JP2004131511 A5 JP 2004131511A5 JP 2004017703 A JP2004017703 A JP 2004017703A JP 2004017703 A JP2004017703 A JP 2004017703A JP 2004131511 A5 JP2004131511 A5 JP 2004131511A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- following structure
- compound according
- alkyl
- halide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41051895A | 1995-03-24 | 1995-03-24 | |
| US54900695A | 1995-10-27 | 1995-10-27 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000079170A Division JP2000319295A (ja) | 1995-03-24 | 2000-03-21 | βシート模倣物およびプロテアーゼインヒビターとしてのその使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2004131511A JP2004131511A (ja) | 2004-04-30 |
| JP2004131511A5 true JP2004131511A5 (enExample) | 2007-01-18 |
| JP4152900B2 JP4152900B2 (ja) | 2008-09-17 |
Family
ID=27021026
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP8529567A Pending JPH10508034A (ja) | 1995-03-24 | 1996-03-25 | βシート模倣物および生物学的に活性なペプチドまたはタンパク質のインヒビターとしてのその使用 |
| JP8529594A Withdrawn JPH10508035A (ja) | 1995-03-24 | 1996-03-25 | βシート模倣物およびプロテアーゼインヒビターとしてのその使用 |
| JP2000079170A Withdrawn JP2000319295A (ja) | 1995-03-24 | 2000-03-21 | βシート模倣物およびプロテアーゼインヒビターとしてのその使用 |
| JP2004017703A Expired - Lifetime JP4152900B2 (ja) | 1995-03-24 | 2004-01-26 | βシート模倣物およびプロテアーゼインヒビターとしてのその使用 |
Family Applications Before (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP8529567A Pending JPH10508034A (ja) | 1995-03-24 | 1996-03-25 | βシート模倣物および生物学的に活性なペプチドまたはタンパク質のインヒビターとしてのその使用 |
| JP8529594A Withdrawn JPH10508035A (ja) | 1995-03-24 | 1996-03-25 | βシート模倣物およびプロテアーゼインヒビターとしてのその使用 |
| JP2000079170A Withdrawn JP2000319295A (ja) | 1995-03-24 | 2000-03-21 | βシート模倣物およびプロテアーゼインヒビターとしてのその使用 |
Country Status (8)
| Country | Link |
|---|---|
| EP (2) | EP0817642A1 (enExample) |
| JP (4) | JPH10508034A (enExample) |
| AT (1) | ATE206433T1 (enExample) |
| AU (2) | AU712581B2 (enExample) |
| CA (2) | CA2215720A1 (enExample) |
| DE (1) | DE69615671T2 (enExample) |
| ES (1) | ES2161354T3 (enExample) |
| WO (1) | WO1996030035A1 (enExample) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5840835A (en) * | 1995-10-30 | 1998-11-24 | Merck & Co., Inc. | Inhibitors of peptide binding to MHC class II proteins |
| US5719296A (en) * | 1995-10-30 | 1998-02-17 | Merck & Co., Inc. | Pseudopeptide lactam inhibitors of peptide binding to MHC class II proteins |
| AU7604196A (en) * | 1995-10-30 | 1997-05-22 | Merck & Co., Inc. | Novel inhibitors of peptide binding to mhc class ii proteins |
| US5817757A (en) * | 1995-10-30 | 1998-10-06 | Merck & Co., Inc. | Inhibitors of peptide binding to MHO class II proteins |
| GB9702377D0 (en) * | 1996-02-23 | 1997-03-26 | Zeneca Ltd | Peptide derivatives |
| WO1997046578A1 (en) | 1996-06-07 | 1997-12-11 | Zeneca Limited | Peptide derivatives |
| AU733562B2 (en) * | 1996-06-18 | 2001-05-17 | Warner-Lambert Company | Process for the preparation of chiral keto-heterocycles of basic amino acids |
| NZ334227A (en) * | 1996-08-05 | 2000-10-27 | Molecumetics Ltd | Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors |
| EP1661566A3 (en) * | 1996-08-05 | 2008-04-16 | Myriad Genetics, Inc. | Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors |
| GB9621836D0 (en) | 1996-10-19 | 1996-12-11 | Zeneca Ltd | Peptide compounds |
| GB9624562D0 (en) | 1996-11-27 | 1997-01-15 | Zeneca Ltd | Peptide derivatives |
| GB9625865D0 (en) * | 1996-12-12 | 1997-01-29 | Zeneca Ltd | Peptides |
| CA2319766A1 (en) * | 1998-02-12 | 1999-08-19 | Molecumetics Ltd. | .beta.-sheet mimetics and methods relating to the use thereof |
| US6323219B1 (en) | 1998-04-02 | 2001-11-27 | Ortho-Mcneil Pharmaceutical, Inc. | Methods for treating immunomediated inflammatory disorders |
| US8093293B2 (en) | 1998-07-06 | 2012-01-10 | Johnson & Johnson Consumer Companies, Inc. | Methods for treating skin conditions |
| US8106094B2 (en) | 1998-07-06 | 2012-01-31 | Johnson & Johnson Consumer Companies, Inc. | Compositions and methods for treating skin conditions |
| AU3208500A (en) | 1999-01-27 | 2000-08-18 | Ortho-Mcneil Pharmaceutical, Inc. | Peptidyl heterocyclic ketones useful as tryptase inhibitors |
| US7309688B2 (en) | 2000-10-27 | 2007-12-18 | Johnson & Johnson Consumer Companies | Topical anti-cancer compositions and methods of use thereof |
| EP1261611A2 (en) * | 2000-02-29 | 2002-12-04 | Bristol-Myers Squibb Pharma Company | Inhibitors of hepatitis c virus ns3 protease |
| US8431550B2 (en) | 2000-10-27 | 2013-04-30 | Johnson & Johnson Consumer Companies, Inc. | Topical anti-cancer compositions and methods of use thereof |
| US7192615B2 (en) | 2001-02-28 | 2007-03-20 | J&J Consumer Companies, Inc. | Compositions containing legume products |
| JPWO2011096440A1 (ja) | 2010-02-03 | 2013-06-10 | 株式会社 ＰＲＩＳＭ ＢｉｏＬａｂ | 天然変性タンパク質に結合する化合物およびそのスクリーニング方法 |
| SG11201702797RA (en) | 2014-10-06 | 2017-05-30 | Cortexyme Inc | Inhibitors of lysine gingipain |
| CA3004095A1 (en) | 2015-11-09 | 2017-05-18 | Cortexyme, Inc. | Inhibitors of arginine gingipain |
| MX2019003087A (es) | 2016-09-16 | 2019-08-12 | Cortexyme Inc | Inhibidores cetónicos de gingipain de lisina. |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA896851B (en) * | 1988-09-14 | 1990-06-27 | Hoffmann La Roche | Use of ace-inhibitors |
-
1996
- 1996-03-25 EP EP96910547A patent/EP0817642A1/en not_active Withdrawn
- 1996-03-25 DE DE69615671T patent/DE69615671T2/de not_active Expired - Fee Related
- 1996-03-25 ES ES96910566T patent/ES2161354T3/es not_active Expired - Lifetime
- 1996-03-25 CA CA002215720A patent/CA2215720A1/en not_active Abandoned
- 1996-03-25 AU AU53714/96A patent/AU712581B2/en not_active Ceased
- 1996-03-25 WO PCT/US1996/004044 patent/WO1996030035A1/en not_active Ceased
- 1996-03-25 EP EP96910566A patent/EP0815123B1/en not_active Expired - Lifetime
- 1996-03-25 AT AT96910566T patent/ATE206433T1/de not_active IP Right Cessation
- 1996-03-25 CA CA002215695A patent/CA2215695C/en not_active Expired - Fee Related
- 1996-03-25 AU AU53729/96A patent/AU713530B2/en not_active Ceased
- 1996-03-25 JP JP8529567A patent/JPH10508034A/ja active Pending
- 1996-03-25 JP JP8529594A patent/JPH10508035A/ja not_active Withdrawn
-
2000
- 2000-03-21 JP JP2000079170A patent/JP2000319295A/ja not_active Withdrawn
-
2004
- 2004-01-26 JP JP2004017703A patent/JP4152900B2/ja not_active Expired - Lifetime
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