JP2008515905A - 有機化合物の組合せ剤 - Google Patents
有機化合物の組合せ剤 Download PDFInfo
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- JP2008515905A JP2008515905A JP2007535797A JP2007535797A JP2008515905A JP 2008515905 A JP2008515905 A JP 2008515905A JP 2007535797 A JP2007535797 A JP 2007535797A JP 2007535797 A JP2007535797 A JP 2007535797A JP 2008515905 A JP2008515905 A JP 2008515905A
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- methyl
- pharmaceutically acceptable
- phenyl
- combination
- ylamino
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| DE102004054054A1 (de) | 2004-11-05 | 2006-05-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine |
| PE20080251A1 (es) | 2006-05-04 | 2008-04-25 | Boehringer Ingelheim Int | Usos de inhibidores de dpp iv |
| CN102838599A (zh) | 2006-05-04 | 2012-12-26 | 贝林格尔.英格海姆国际有限公司 | 多晶型 |
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| JP5523107B2 (ja) | 2006-11-30 | 2014-06-18 | プロビオドルグ エージー | グルタミニルシクラーゼの新規阻害剤 |
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| PE20091730A1 (es) | 2008-04-03 | 2009-12-10 | Boehringer Ingelheim Int | Formulaciones que comprenden un inhibidor de dpp4 |
| TW201006823A (en) * | 2008-07-14 | 2010-02-16 | Novartis Ag | Use of pyrimidylaminobenzamide derivatives for the treatment of fibrosis |
| KR20200118243A (ko) | 2008-08-06 | 2020-10-14 | 베링거 인겔하임 인터내셔날 게엠베하 | 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료 |
| UY32030A (es) | 2008-08-06 | 2010-03-26 | Boehringer Ingelheim Int | "tratamiento para diabetes en pacientes inapropiados para terapia con metformina" |
| MX370599B (es) | 2008-08-15 | 2019-12-18 | Boehringer Ingelheim Int | Derivados de purina para su uso en el tratamiento de enfermedades relacionadas con fab. |
| US20200155558A1 (en) | 2018-11-20 | 2020-05-21 | Boehringer Ingelheim International Gmbh | Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug |
| EA022310B1 (ru) | 2008-12-23 | 2015-12-30 | Бёрингер Ингельхайм Интернациональ Гмбх | Солевые формы органического соединения |
| AR074990A1 (es) | 2009-01-07 | 2011-03-02 | Boehringer Ingelheim Int | Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina |
| TWI466672B (zh) | 2009-01-29 | 2015-01-01 | Boehringer Ingelheim Int | 小兒科病人糖尿病之治療 |
| NZ619520A (en) | 2009-02-13 | 2015-06-26 | Boehringer Ingelheim Int | Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics |
| SG174504A1 (en) * | 2009-03-27 | 2011-10-28 | Bristol Myers Squibb Co | Methods for preventing major adverse cardiovascular events with dpp-iv inhibitors |
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| EA030999B1 (ru) | 2009-10-02 | 2018-10-31 | Бёрингер Ингельхайм Интернациональ Гмбх | Применение фармацевтической композиции, включающей ингибитор дпп-4 и гидрохлорид метформина |
| NZ599298A (en) | 2009-11-27 | 2014-11-28 | Boehringer Ingelheim Int | Treatment of genotyped diabetic patients with dpp-iv inhibitors such as linagliptin |
| JP6026284B2 (ja) | 2010-03-03 | 2016-11-16 | プロビオドルグ エージー | グルタミニルシクラーゼの阻害剤 |
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| WO2011138421A1 (en) | 2010-05-05 | 2011-11-10 | Boehringer Ingelheim International Gmbh | Combination therapy |
| NZ603319A (en) | 2010-06-24 | 2015-04-24 | Boehringer Ingelheim Int | Diabetes therapy |
| AR083878A1 (es) | 2010-11-15 | 2013-03-27 | Boehringer Ingelheim Int | Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento |
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| CA2841552C (en) | 2011-07-15 | 2020-06-23 | Boehringer Ingelheim International Gmbh | Substituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions |
| US8722716B2 (en) | 2011-11-23 | 2014-05-13 | The Board Of Regents Of The University Of Texas System | Isoxazole treatments for diabetes |
| US20130172244A1 (en) | 2011-12-29 | 2013-07-04 | Thomas Klein | Subcutaneous therapeutic use of dpp-4 inhibitor |
| US9555001B2 (en) | 2012-03-07 | 2017-01-31 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition and uses thereof |
| US20130303554A1 (en) | 2012-05-14 | 2013-11-14 | Boehringer Ingelheim International Gmbh | Use of a dpp-4 inhibitor in sirs and/or sepsis |
| EP3685839A1 (en) | 2012-05-14 | 2020-07-29 | Boehringer Ingelheim International GmbH | Linagliptin for use in the treatment of albuminuria and kidney related diseases |
| WO2013174767A1 (en) | 2012-05-24 | 2013-11-28 | Boehringer Ingelheim International Gmbh | A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference |
| JP6374862B2 (ja) | 2012-05-24 | 2018-08-15 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 自己免疫性糖尿病、特に、ｌａｄａの治療に使用するためのｄｐｐ−４阻害剤としてのキサンチン誘導体 |
| KR101386697B1 (ko) * | 2012-06-18 | 2014-04-18 | 아주대학교산학협력단 | 이매티닙 또는 이의 약학적으로 허용되는 염을 유효성분으로 포함하는 혈관 투과성 관련 질환의 치료 또는 예방용 조성물 |
| WO2014124860A1 (en) | 2013-02-14 | 2014-08-21 | Boehringer Ingelheim International Gmbh | Specific pde4b-inhibitors for the treatment of diabetes mellitus |
| KR20210099201A (ko) | 2013-03-15 | 2021-08-11 | 베링거 인겔하임 인터내셔날 게엠베하 | 심장보호 및 신장보호 항당뇨병 치료요법에서의 리나글립틴의 사용 |
| WO2014198906A1 (en) * | 2013-06-14 | 2014-12-18 | Boehringer Ingelheim International Gmbh | Dpp-4 inhibitors for treating diabetes and its complications |
| ES2950384T3 (es) | 2014-02-28 | 2023-10-09 | Boehringer Ingelheim Int | Uso médico de un inhibidor de DPP-4 |
| WO2017211979A1 (en) | 2016-06-10 | 2017-12-14 | Boehringer Ingelheim International Gmbh | Combinations of linagliptin and metformin |
| PL3461819T3 (pl) | 2017-09-29 | 2020-11-30 | Probiodrug Ag | Inhibitory cyklazy glutaminylowej |
| BR112020024793A2 (pt) | 2018-07-17 | 2021-03-02 | Boehringer Ingelheim International Gmbh | terapia antidiabética cardiossegura |
| BR112020026164A2 (pt) | 2018-07-17 | 2021-03-23 | Boehringer Ingelheim International Gmbh | terapia antidiabética cardioprotetora e nefroprotetora |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1917865A (zh) * | 2004-01-22 | 2007-02-21 | 诺瓦提斯公司 | 有机化合物的组合 |
-
2005
- 2005-10-06 AU AU2005294320A patent/AU2005294320A1/en not_active Abandoned
- 2005-10-06 KR KR1020077007859A patent/KR20070099527A/ko not_active Withdrawn
- 2005-10-06 BR BRPI0516446-0A patent/BRPI0516446A/pt not_active IP Right Cessation
- 2005-10-06 US US11/576,860 patent/US20080070922A1/en not_active Abandoned
- 2005-10-06 WO PCT/US2005/035917 patent/WO2006041976A1/en not_active Ceased
- 2005-10-06 RU RU2007116869/15A patent/RU2007116869A/ru not_active Application Discontinuation
- 2005-10-06 CA CA002580266A patent/CA2580266A1/en not_active Abandoned
- 2005-10-06 JP JP2007535797A patent/JP2008515905A/ja not_active Withdrawn
- 2005-10-06 CN CNA200580033958XA patent/CN101035536A/zh active Pending
- 2005-10-06 EP EP05801149A patent/EP1802308A1/en not_active Withdrawn
- 2005-10-06 MX MX2007004021A patent/MX2007004021A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US20080070922A1 (en) | 2008-03-20 |
| RU2007116869A (ru) | 2008-11-20 |
| CA2580266A1 (en) | 2006-04-20 |
| MX2007004021A (es) | 2007-05-24 |
| EP1802308A1 (en) | 2007-07-04 |
| WO2006041976A1 (en) | 2006-04-20 |
| CN101035536A (zh) | 2007-09-12 |
| AU2005294320A1 (en) | 2006-04-20 |
| BRPI0516446A (pt) | 2008-09-02 |
| KR20070099527A (ko) | 2007-10-09 |
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