JP2008500991A5 - - Google Patents

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Publication number
JP2008500991A5
JP2008500991A5 JP2007513846A JP2007513846A JP2008500991A5 JP 2008500991 A5 JP2008500991 A5 JP 2008500991A5 JP 2007513846 A JP2007513846 A JP 2007513846A JP 2007513846 A JP2007513846 A JP 2007513846A JP 2008500991 A5 JP2008500991 A5 JP 2008500991A5
Authority
JP
Japan
Prior art keywords
bromo
phenoxy
carbonyl
pyrazole
acetic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2007513846A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008500991A (ja
Filing date
Publication date
Priority claimed from GB0412198A external-priority patent/GB0412198D0/en
Priority claimed from GB0414196A external-priority patent/GB0414196D0/en
Priority claimed from GB0424018A external-priority patent/GB0424018D0/en
Application filed filed Critical
Priority claimed from PCT/EP2005/005884 external-priority patent/WO2005115382A1/en
Publication of JP2008500991A publication Critical patent/JP2008500991A/ja
Publication of JP2008500991A5 publication Critical patent/JP2008500991A5/ja
Ceased legal-status Critical Current

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JP2007513846A 2004-05-29 2005-05-30 医学的使用のためのｃｒｔｈ２レセプターリガンド Ceased JP2008500991A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0412198A GB0412198D0 (en) 2004-05-29 2004-05-29 Medicinal use of receptor ligands
GB0414196A GB0414196D0 (en) 2004-06-24 2004-06-24 Medicinal use of receptor ligands
GB0424018A GB0424018D0 (en) 2004-10-29 2004-10-29 Medicinal use of receptor ligands
PCT/EP2005/005884 WO2005115382A1 (en) 2004-05-29 2005-05-30 Crth2 receptor ligands for medicinal uses

Publications (2)

Publication Number Publication Date
JP2008500991A JP2008500991A (ja) 2008-01-17
JP2008500991A5 true JP2008500991A5 (enExample) 2008-07-17

Family

ID=34993084

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007513846A Ceased JP2008500991A (ja) 2004-05-29 2005-05-30 医学的使用のためのｃｒｔｈ２レセプターリガンド

Country Status (14)

Country Link
US (2) US8022063B2 (enExample)
EP (2) EP1758579A1 (enExample)
JP (1) JP2008500991A (enExample)
KR (1) KR20070045153A (enExample)
AU (1) AU2005247110B2 (enExample)
BR (1) BRPI0511676A (enExample)
CA (1) CA2568766A1 (enExample)
CR (1) CR8838A (enExample)
EA (1) EA014729B1 (enExample)
IL (1) IL179694A (enExample)
MX (1) MXPA06013912A (enExample)
NO (1) NO20066048L (enExample)
NZ (1) NZ551810A (enExample)
WO (1) WO2005115382A1 (enExample)

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TWI410421B (zh) 2009-07-16 2013-10-01 Actelion Pharmaceuticals Ltd 吡啶－４－基衍生物
CN102822163B (zh) * 2009-12-23 2016-01-20 艾恩伍德医药品股份有限公司 Crth2调节剂
EP2586772A4 (en) 2010-06-23 2013-11-13 Taisho Pharmaceutical Co Ltd isoquinoline
CA2805452C (en) 2010-07-05 2018-07-31 Actelion Pharmaceuticals Ltd 1-phenyl-substituted heterocyclyl derivatives and their use as prostaglandin d2 receptor modulators
EP2457900A1 (en) 2010-11-25 2012-05-30 Almirall, S.A. New pyrazole derivatives having CRTh2 antagonistic behaviour
CA2818470C (en) 2011-01-19 2019-03-05 Actelion Pharmaceuticals Ltd 2-methoxy-pyridin-4-yl derivatives
TR201906779T4 (tr) * 2011-05-12 2019-05-21 Proteostasis Therapeutics Inc Proteostaz regülatörleri.
BR112014001265A2 (pt) 2011-07-29 2017-02-21 Taisho Pharmaceutical Co Ltd composto de amidina ou seu sal
CN104114169A (zh) 2011-12-16 2014-10-22 阿托佩斯治疗有限公司 用于治疗嗜酸细胞性食管炎的crth2拮抗剂和质子泵抑制剂的组合物
TW201331179A (zh) 2011-12-21 2013-08-01 Actelion Pharmaceuticals Ltd 雜環衍生物及其作為前列腺素ｄ２受體調節劑之用途
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TWI695831B (zh) 2014-09-13 2020-06-11 香港商南北兄弟藥業投資有限公司 Ｃｒｔｈ２拮抗劑化合物及其用途
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JPWO2022138700A1 (enExample) * 2020-12-23 2022-06-30

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