JP2007518685A5 - - Google Patents
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- Publication number
- JP2007518685A5 JP2007518685A5 JP2006519266A JP2006519266A JP2007518685A5 JP 2007518685 A5 JP2007518685 A5 JP 2007518685A5 JP 2006519266 A JP2006519266 A JP 2006519266A JP 2006519266 A JP2006519266 A JP 2006519266A JP 2007518685 A5 JP2007518685 A5 JP 2007518685A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cyclo
- aryl
- hydroxy
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000000217 alkyl group Chemical group 0.000 claims 18
- 125000000623 heterocyclic group Chemical group 0.000 claims 13
- 125000003545 alkoxy group Chemical group 0.000 claims 12
- 125000004423 acyloxy group Chemical group 0.000 claims 8
- 125000003118 aryl group Chemical group 0.000 claims 8
- 229910052736 halogen Inorganic materials 0.000 claims 8
- 150000002367 halogens Chemical class 0.000 claims 8
- -1 prostaglandin compound Chemical class 0.000 claims 8
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 6
- 125000004104 aryloxy group Chemical group 0.000 claims 6
- 229910052739 hydrogen Inorganic materials 0.000 claims 6
- 239000001257 hydrogen Substances 0.000 claims 6
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 6
- 125000004043 oxo group Chemical group O=* 0.000 claims 6
- 125000002947 alkylene group Chemical group 0.000 claims 5
- 150000001875 compounds Chemical class 0.000 claims 5
- 125000001820 oxy group Chemical group [*:1]O[*:2] 0.000 claims 5
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 4
- 125000001931 aliphatic group Chemical group 0.000 claims 4
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 4
- 150000002431 hydrogen Chemical class 0.000 claims 4
- 229910052757 nitrogen Inorganic materials 0.000 claims 4
- 229910052760 oxygen Inorganic materials 0.000 claims 4
- 239000001301 oxygen Substances 0.000 claims 4
- 229910052717 sulfur Inorganic materials 0.000 claims 4
- 239000011593 sulfur Substances 0.000 claims 4
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 2
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 claims 2
- 125000004356 hydroxy functional group Chemical group O* 0.000 claims 2
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims 2
- 229920006395 saturated elastomer Polymers 0.000 claims 2
- 239000004480 active ingredient Substances 0.000 claims 1
- 230000003779 hair growth Effects 0.000 claims 1
- 125000005842 heteroatom Chemical group 0.000 claims 1
- 230000001737 promoting effect Effects 0.000 claims 1
- 0 **C(C(BC(*)(**)**)C(C1N)N)C1I Chemical compound **C(C(BC(*)(**)**)C(C1N)N)C1I 0.000 description 4
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49412103P | 2003-08-12 | 2003-08-12 | |
| PCT/JP2004/011864 WO2005013928A1 (en) | 2003-08-12 | 2004-08-12 | Composition and method for promoting hair growth |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010226217A Division JP5318837B2 (ja) | 2003-08-12 | 2010-10-06 | 育毛を促進する組成物および方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2007518685A JP2007518685A (ja) | 2007-07-12 |
| JP2007518685A5 true JP2007518685A5 (https=) | 2007-10-04 |
| JP4642021B2 JP4642021B2 (ja) | 2011-03-02 |
Family
ID=34135320
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006519266A Expired - Fee Related JP4642021B2 (ja) | 2003-08-12 | 2004-08-12 | 育毛を促進する組成物および方法 |
| JP2010226217A Expired - Fee Related JP5318837B2 (ja) | 2003-08-12 | 2010-10-06 | 育毛を促進する組成物および方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010226217A Expired - Fee Related JP5318837B2 (ja) | 2003-08-12 | 2010-10-06 | 育毛を促進する組成物および方法 |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US8686035B2 (https=) |
| EP (2) | EP1673058B1 (https=) |
| JP (2) | JP4642021B2 (https=) |
| KR (3) | KR101166738B1 (https=) |
| CN (1) | CN1867310B (https=) |
| AT (1) | ATE526008T1 (https=) |
| CA (1) | CA2534645C (https=) |
| CY (1) | CY1112076T1 (https=) |
| DK (1) | DK1673058T3 (https=) |
| ES (1) | ES2369892T3 (https=) |
| PL (1) | PL1673058T3 (https=) |
| PT (1) | PT1673058E (https=) |
| SI (1) | SI1673058T1 (https=) |
| TW (2) | TWI495471B (https=) |
| WO (1) | WO2005013928A1 (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI495471B (zh) | 2003-08-12 | 2015-08-11 | R Tech Ueno Ltd | 促進毛髮生長之組成物及方法 |
| EP1830793A1 (en) * | 2004-12-29 | 2007-09-12 | R-Tech Ueno, Ltd. | Composition and method for scalp and hair treatment |
| US8455547B2 (en) | 2008-02-05 | 2013-06-04 | Allergan, Inc. | Substituted cyclopentanes having prostaglandin activity |
| US7964596B2 (en) * | 2008-03-07 | 2011-06-21 | Allergan, Inc. | Therapeutic compounds |
| US7732443B2 (en) * | 2008-03-18 | 2010-06-08 | Yariv Donde | Therapeutic substituted cyclopentanes |
| WO2009137345A1 (en) * | 2008-05-09 | 2009-11-12 | Allergan, Inc. | Therapeutic compounds |
| US20130067604A1 (en) * | 2010-02-24 | 2013-03-14 | Sadatoshi Sakuma | Method of Treatment or Prevention of Hair Loss or for the Enhancement of Hair Growth |
| WO2012176792A1 (ja) | 2011-06-21 | 2012-12-27 | 株式会社アールテック・ウエノ | 炎症性疾患、アレルギー性疾患および自己免疫疾患用途のための医薬組成物 |
| WO2014182908A1 (en) * | 2013-05-10 | 2014-11-13 | Topical Solutions, Inc. | Compositions and methods for treating nails, claws, and hoofs |
| US12539302B2 (en) | 2019-08-07 | 2026-02-03 | Aneira Pharma, Inc. | Methods and compositions for the treatment of hair loss |
| EP4331683A3 (en) | 2019-08-07 | 2024-08-07 | Aneira Pharma, Inc. | Methods and compositions for the treatment of hair loss |
Family Cites Families (63)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2328132A1 (de) * | 1973-05-30 | 1975-01-02 | Schering Ag | Neue prostansaeurederivate und verfahren zu ihrer herstellung |
| DE2434133C2 (de) * | 1974-07-12 | 1987-03-19 | Schering AG, 1000 Berlin und 4709 Bergkamen | 15,15-Äthylendioxy-Prostansäurederivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
| CS230650B1 (cs) | 1983-01-14 | 1984-08-13 | Jan Stanek | Způsob výroby acetalů prostanoidů |
| DE3325175A1 (de) | 1983-07-08 | 1985-01-17 | Schering AG, 1000 Berlin und 4709 Bergkamen | 11-halogen-prostanderivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
| JPH0818989B2 (ja) | 1984-01-12 | 1996-02-28 | 株式会社ミドリ十字 | 脂肪乳剤中のプロスタグランジンの安定化方法 |
| JPS61218510A (ja) * | 1985-03-22 | 1986-09-29 | Dai Ichi Seiyaku Co Ltd | 毛髪用剤 |
| CA1322749C (en) | 1987-01-28 | 1993-10-05 | Ryuzo Ueno | Prostaglandins of the d series, and tranquilizers and soporifics containing the same |
| US5166174A (en) | 1987-01-28 | 1992-11-24 | K.K. Ueno Seiyaku Oyo Kenkyujo | Prostaglandins E and anti-ulcers containing same |
| US5428062A (en) * | 1987-01-28 | 1995-06-27 | K.K. Ueno Seiyaku Oyo Kenkyujo | Prostaglandins E and anti ulcers containing same |
| CA1324129C (en) * | 1987-04-30 | 1993-11-09 | Ryuzo Ueno | Prostaglandins of the f series |
| US5591887A (en) | 1987-04-30 | 1997-01-07 | R-Tech Ueno, Ltd. | Prostaglandins of the F series |
| US5221763A (en) | 1987-04-30 | 1993-06-22 | R-Tech Ueno, Ltd. | Prostaglandins of the F series |
| US5166178B1 (en) | 1987-09-18 | 1998-07-21 | R Tech Ueno Ltd | Ocular hypotensive agents |
| DE3850676T2 (de) | 1987-09-18 | 1994-11-03 | Ueno Seiyaku Oyo Kenkyujo Kk | Hypotensive okulare Mittel. |
| US5212200A (en) | 1987-09-18 | 1993-05-18 | R-Tech Ueno, Ltd. | Ocular hypotensive agents |
| TW224942B (https=) | 1990-04-04 | 1994-06-11 | Adka Ueno Kk | |
| US5208256A (en) | 1990-05-22 | 1993-05-04 | R-Tech Ueno, Ltd. | Treatment of ocular hypertension with a synergistic combination for ocular administration |
| CA2042934C (en) | 1990-05-22 | 2002-04-23 | Ryuji Ueno | Treatment of ocular hypertension with an ocular synergistic combination |
| US5175189A (en) | 1990-05-22 | 1992-12-29 | K.K. Ueno Seiyaku Oyo Kenkyujo | Treatment of ocular hypertension with a synergistic combination for ophthalmic use |
| ES2084771T3 (es) * | 1990-05-22 | 1996-05-16 | R Tech Ueno Ltd | Tratamiento de la hipertension ocular con la ayuda de una combinacion sinergica. |
| TW210287B (https=) | 1991-03-01 | 1993-08-01 | Kabushikaisha Ueno Seiyaku Oyo Kenkyujo | |
| US5274130A (en) | 1991-09-03 | 1993-12-28 | R-Tech Ueno Ltd. | Process for production of prostaglandin intermediates |
| DE69232150T2 (de) | 1992-03-19 | 2002-03-07 | R-Tech Ueno, Ltd. | Behandlung von Augenhochdruck mit Betablockern und Prostansäurederivaten |
| EP0668076B1 (en) | 1992-08-26 | 2002-09-04 | Sucampo AG | Stabilization of a prostanoic acid compound |
| SE9303444D0 (sv) | 1993-10-20 | 1993-10-20 | Kabi Pharmacia Ab | New use of prostaglandins |
| SE9402816D0 (sv) | 1994-08-24 | 1994-08-24 | Pharmacia Ab | Method and meams for drug administration |
| WO1997047595A1 (en) | 1996-06-10 | 1997-12-18 | R-Tech Ueno, Ltd. | Endothelin antagonist |
| WO1998000100A1 (en) | 1996-07-03 | 1998-01-08 | The Board Of Regents Of The University Of Oklahoma | Enhancement of skin pigmentation by prostaglandins |
| WO1998020881A1 (en) * | 1996-11-12 | 1998-05-22 | Alcon Laboratories, Inc | 15-ketal prostaglandins for the treatment of glaucoma or ocular hypertension |
| ATE266397T1 (de) * | 1997-02-04 | 2004-05-15 | Murray A Johnstone | Verfahren zur förderung des haarwuchses und entwicklung des haarsystems |
| JP3217293B2 (ja) * | 1997-04-17 | 2001-10-09 | 株式会社アールテック・ウエノ | 発毛・育毛剤 |
| US6235781B1 (en) | 1998-07-14 | 2001-05-22 | Alcon Laboratories, Inc. | Prostaglandin product |
| US6225348B1 (en) | 1998-08-20 | 2001-05-01 | Alfred W. Paulsen | Method of treating macular degeneration with a prostaglandin derivative |
| BRPI0014869B8 (pt) | 1999-10-15 | 2021-05-25 | Sucampo Ag | prostaglandinas bicíclicas, composições estabilizadas das mesmas, bem como processo para sua estabilização |
| US20020146439A1 (en) | 2000-03-31 | 2002-10-10 | Delong Mitchell Anthony | Compositions and methods for treating hair loss using oximyl and hydroxylamino prostaglandins |
| US20020037914A1 (en) | 2000-03-31 | 2002-03-28 | Delong Mitchell Anthony | Compositions and methods for treating hair loss using C16-C20 aromatic tetrahydro prostaglandins |
| US20020172693A1 (en) | 2000-03-31 | 2002-11-21 | Delong Michell Anthony | Compositions and methods for treating hair loss using non-naturally occurring prostaglandins |
| FR2812191B1 (fr) | 2000-07-28 | 2003-10-17 | Oreal | Utilisation d'agonistes du recepteur des prostaglandines e2 (ep-3) pour attenuer, diminuer ou stopper la pousse des cheveux et des poils dans des preparations cosmetiques |
| FR2812190B1 (fr) | 2000-07-28 | 2003-01-31 | Oreal | Utilisation d'agonistes non prostanoiques des recepteurs des prostaglandines ep-2 et/ou ep-4 comme agent cosmetique permettant d'attenuer, de diminuer ou d'arreter la chute des cheveux et des poils |
| FR2812193B1 (fr) | 2000-07-28 | 2003-10-24 | Oreal | Utilisation d'antagoniste des recepteurs des prostaglandines ep-2 et/ou ep-4 pour attenuer, diminuer ou stopper la pousse des cheveux et des poils dans des preparations cosmetiques |
| FR2812192B1 (fr) | 2000-07-28 | 2003-01-31 | Oreal | Utilisation d'antagonistes de recepteur des prostaglandines ep-3 comme agent cosmetique permettant d'attenuer, de diminuer ou d'arreter la chute des cheveux et des poils |
| US6414016B1 (en) | 2000-09-05 | 2002-07-02 | Sucampo, A.G. | Anti-constipation composition |
| SE0100158D0 (sv) | 2001-01-19 | 2001-01-19 | Synphora Ab | Novel method and composition for local treatment of Meniere´s disease and tinnitus |
| EP1420794B1 (en) * | 2001-08-31 | 2017-12-27 | Sucampo AG | Prostaglandin analogs as chloride channel openers |
| JP2003155218A (ja) * | 2001-09-10 | 2003-05-27 | Lion Corp | 養育毛組成物 |
| US7351404B2 (en) | 2002-02-04 | 2008-04-01 | Allergan, Inc. | Method of enhancing hair growth |
| US20030199590A1 (en) | 2002-07-25 | 2003-10-23 | Cagle Gerald D | Prostaglandin analogues for promotion of hair growth |
| US20040115234A1 (en) | 2002-09-24 | 2004-06-17 | Gewirtz Joan T. | Cosmetic composition |
| TWI495471B (zh) | 2003-08-12 | 2015-08-11 | R Tech Ueno Ltd | 促進毛髮生長之組成物及方法 |
| US20050112075A1 (en) | 2003-11-25 | 2005-05-26 | Hwang Cheng S. | Reduction of hair growth |
| EP1830793A1 (en) | 2004-12-29 | 2007-09-12 | R-Tech Ueno, Ltd. | Composition and method for scalp and hair treatment |
| WO2006106915A1 (ja) | 2005-03-31 | 2006-10-12 | Asahi Glass Company, Limited | プロスタグランジンＦ2α誘導体を有効成分として含む網膜神経細胞保護剤 |
| WO2007023841A1 (ja) | 2005-08-25 | 2007-03-01 | Taisho Pharmaceutical Co., Ltd. | 発毛剤組成物 |
| US20070160562A1 (en) | 2006-01-06 | 2007-07-12 | Brinkenhoff Michael C | Delivery devices for hair-promoting cosmetic agent |
| US20070286890A1 (en) | 2006-06-07 | 2007-12-13 | John Garnett Walt | Eyelash applicator and method |
| US8206695B2 (en) | 2007-04-26 | 2012-06-26 | La Canada Ventures, Inc. | Eyelash enhancement composition and method of treatment |
| US20090018204A1 (en) | 2007-07-13 | 2009-01-15 | Brinkenhoff Michael C | Composition and method for enhancing hair growth |
| WO2009035565A1 (en) | 2007-09-07 | 2009-03-19 | Qlt Plug Delivery, Inc | Prostaglandin analogues for implant devices and methods |
| US20090088473A1 (en) | 2007-09-28 | 2009-04-02 | Cayman Chemical Company | Method for screening of prostaglandin compounds comprising an optimal formulation for the enhancement of hair growth and the stimulation of follicular anagen and formulations resulting therefrom |
| WO2009054787A1 (en) * | 2007-10-26 | 2009-04-30 | Astrazeneca Ab | 1,2,4-triazole carboxylic acid derivatives as modulators of mglur5 |
| EP2214482A4 (en) | 2007-10-31 | 2011-08-24 | Pamela Lipkin | COMPOSITIONS OF PROSTAGLANDIN ANALOGUES AND METHODS OF TREATING EPITHELIAL STATES |
| US20100166841A1 (en) | 2008-05-14 | 2010-07-01 | Peter Thomas Roth | Prostaglandin Based Compositions and Method of Use Thereof |
| US20080275118A1 (en) | 2008-06-12 | 2008-11-06 | Shaw Mari M | Health and cosmetic composition and regime for stimulating hair growth and thickening on the head, including the scalp, eyelashes, and eyebrows, and which discourages hair loss |
-
2004
- 2004-08-11 TW TW099126213A patent/TWI495471B/zh not_active IP Right Cessation
- 2004-08-11 TW TW093124177A patent/TWI348386B/zh not_active IP Right Cessation
- 2004-08-12 JP JP2006519266A patent/JP4642021B2/ja not_active Expired - Fee Related
- 2004-08-12 EP EP04771825A patent/EP1673058B1/en not_active Revoked
- 2004-08-12 EP EP10008142A patent/EP2243771A3/en not_active Withdrawn
- 2004-08-12 WO PCT/JP2004/011864 patent/WO2005013928A1/en not_active Ceased
- 2004-08-12 AT AT04771825T patent/ATE526008T1/de active
- 2004-08-12 DK DK04771825.9T patent/DK1673058T3/da active
- 2004-08-12 CN CN2004800298049A patent/CN1867310B/zh not_active Expired - Fee Related
- 2004-08-12 KR KR1020117017023A patent/KR101166738B1/ko not_active Expired - Fee Related
- 2004-08-12 ES ES04771825T patent/ES2369892T3/es not_active Expired - Lifetime
- 2004-08-12 CA CA2534645A patent/CA2534645C/en not_active Expired - Fee Related
- 2004-08-12 KR KR1020067002643A patent/KR101137750B1/ko not_active Expired - Fee Related
- 2004-08-12 KR KR1020117031353A patent/KR20120008080A/ko not_active Ceased
- 2004-08-12 SI SI200431752T patent/SI1673058T1/sl unknown
- 2004-08-12 US US10/567,462 patent/US8686035B2/en not_active Expired - Fee Related
- 2004-08-12 PL PL04771825T patent/PL1673058T3/pl unknown
- 2004-08-12 PT PT04771825T patent/PT1673058E/pt unknown
-
2010
- 2010-10-06 JP JP2010226217A patent/JP5318837B2/ja not_active Expired - Fee Related
-
2011
- 2011-11-21 CY CY20111101121T patent/CY1112076T1/el unknown
-
2014
- 2014-02-07 US US14/175,356 patent/US20140171496A1/en not_active Abandoned
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