JP2007514638A5 - - Google Patents

Download PDF

Info

Publication number
JP2007514638A5
JP2007514638A5 JP2006516318A JP2006516318A JP2007514638A5 JP 2007514638 A5 JP2007514638 A5 JP 2007514638A5 JP 2006516318 A JP2006516318 A JP 2006516318A JP 2006516318 A JP2006516318 A JP 2006516318A JP 2007514638 A5 JP2007514638 A5 JP 2007514638A5
Authority
JP
Japan
Prior art keywords
disorders
mixture
dmf
water
alcoholism
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2006516318A
Other languages
English (en)
Japanese (ja)
Other versions
JP4669839B2 (ja
JP2007514638A (ja
Filing date
Publication date
Priority claimed from FR0307757A external-priority patent/FR2856684B1/fr
Application filed filed Critical
Publication of JP2007514638A publication Critical patent/JP2007514638A/ja
Publication of JP2007514638A5 publication Critical patent/JP2007514638A5/ja
Application granted granted Critical
Publication of JP4669839B2 publication Critical patent/JP4669839B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2006516318A 2003-06-26 2004-06-24 ジフェニルピリジン誘導体、その製造法および治療用途 Expired - Fee Related JP4669839B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0307757A FR2856684B1 (fr) 2003-06-26 2003-06-26 Derives de diphenylpyridine, leur preparation et leur application en therapeutique
PCT/FR2004/001581 WO2005000817A2 (fr) 2003-06-26 2004-06-24 Derives de diphenylpyridine, leur preparation et leur application en therapeutique

Publications (3)

Publication Number Publication Date
JP2007514638A JP2007514638A (ja) 2007-06-07
JP2007514638A5 true JP2007514638A5 (enExample) 2007-08-30
JP4669839B2 JP4669839B2 (ja) 2011-04-13

Family

ID=33515448

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006516318A Expired - Fee Related JP4669839B2 (ja) 2003-06-26 2004-06-24 ジフェニルピリジン誘導体、その製造法および治療用途

Country Status (16)

Country Link
US (1) US7345059B2 (enExample)
EP (1) EP1641758B1 (enExample)
JP (1) JP4669839B2 (enExample)
KR (1) KR20060025191A (enExample)
CN (1) CN1832945A (enExample)
AR (1) AR044906A1 (enExample)
AT (1) ATE412635T1 (enExample)
AU (1) AU2004251914B9 (enExample)
BR (1) BRPI0411762A (enExample)
CA (1) CA2528619A1 (enExample)
DE (1) DE602004017463D1 (enExample)
FR (1) FR2856684B1 (enExample)
IL (1) IL172733A0 (enExample)
MX (1) MXPA05014222A (enExample)
TW (1) TW200504019A (enExample)
WO (1) WO2005000817A2 (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003225964B2 (en) 2002-03-28 2008-11-20 Merck Sharp & Dohme Corp. Substituted 2,3-diphenyl pyridines
WO2004029204A2 (en) 2002-09-27 2004-04-08 Merck & Co., Inc. Substituted pyrimidines
DK1868999T3 (da) 2005-04-06 2009-08-17 Hoffmann La Roche Pyridin-3-carboxamidderivater som omvendte CB1-agonister
GB0514739D0 (en) * 2005-07-19 2005-08-24 Astrazeneca Ab Therapeutic agents
WO2007039797A1 (en) * 2005-10-03 2007-04-12 Pfizer Products Inc. Use of cannabinoid receptor-1 antagonist for treating inflammation and arthritis
FR2899899A1 (fr) * 2006-04-14 2007-10-19 Sanofi Aventis Sa Derives d'aminomethyl pyridine, leur preparation et leur application en therapeutique
US7629346B2 (en) 2006-06-19 2009-12-08 Hoffmann-La Roche Inc. Pyrazinecarboxamide derivatives as CB1 antagonists
FR2904827B1 (fr) 2006-08-11 2008-09-19 Sanofi Aventis Sa Derives de 5,6-bisaryl-2-pyridine-carboxamide, leur preparation et leur application en therapeutique comme antiganistes des recepteurs a l'urotensine ii
US7781593B2 (en) 2006-09-14 2010-08-24 Hoffmann-La Roche Inc. 5-phenyl-nicotinamide derivatives
FR2927330B1 (fr) 2008-02-07 2010-02-19 Sanofi Aventis Derives de 5,6-bisaryl-2-pyridine-carboxamide, leur preparation et leur application en therapeutique comme antagonistes des recepteurs a l'urotensine ii
US8410107B2 (en) 2010-10-15 2013-04-02 Hoffmann-La Roche Inc. N-pyridin-3-yl or N-pyrazin-2-yl carboxamides
US8669254B2 (en) 2010-12-15 2014-03-11 Hoffman-La Roche Inc. Pyridine, pyridazine, pyrimidine or pyrazine carboxamides as HDL-cholesterol raising agents
CN102276517B (zh) * 2011-06-29 2012-11-28 孙光辉 二芳基吡啶类药物的合成方法
CN104837832B (zh) * 2012-10-05 2019-04-26 里格尔药品股份有限公司 Gdf-8抑制剂
EP3456716A4 (en) * 2016-05-09 2019-11-06 Nippon Soda Co., Ltd. RINGFUL AMID CONNECTION AND PESTICIDES
KR102598895B1 (ko) 2016-07-12 2023-11-07 레볼루션 메디슨즈, 인크. 다른자리 입체성 shp2 억제제로서의 2,5-이치환 3-메틸 피라진 및 2,5,6-3치환 3-메틸 피라진
JP7240319B2 (ja) 2017-01-23 2023-03-15 レヴォリューション・メディスンズ,インコーポレイテッド アロステリックshp2阻害剤としての二環式化合物
KR20190110588A (ko) 2017-01-23 2019-09-30 레볼루션 메디슨즈, 인크. 알로스테릭 shp2 억제제로서의 피리딘 화합물
WO2019051084A1 (en) 2017-09-07 2019-03-14 Revolution Medicines, Inc. SHP2 INHIBITOR COMPOSITIONS AND METHODS OF TREATING CANCER
MX2020003579A (es) 2017-10-12 2020-07-22 Revolution Medicines Inc Compuestos de piridina, pirazina, y triazina como inhibidores de shp2 alostericos.
TW201927791A (zh) 2017-12-15 2019-07-16 美商銳新醫藥公司 作為變構shp2抑制劑的多環化合物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2198737B1 (enExample) * 1972-09-13 1975-11-28 Serdex
FR2248027B2 (enExample) * 1973-10-18 1977-09-09 Serdex
FR2612189B1 (fr) * 1987-03-13 1989-06-23 Roussel Uclaf Nouveaux derives de la pyridine, leur procede de preparation et les nouveaux intermediaires obtenus, leur application a titre de medicaments et les compositions les renfermant
GB9210436D0 (en) * 1992-05-15 1992-07-01 Neave Andrew J A light projector for use in conjunction with light guides
FR2741621B1 (fr) * 1995-11-23 1998-02-13 Sanofi Sa Nouveaux derives de pyrazole, procede pour leur preparation et compositions pharmaceutiques en contenant
FR2816938B1 (fr) * 2000-11-22 2003-01-03 Sanofi Synthelabo Derives de 3-aroylindole, leur procede de preparation et les compositions pharmaceutiques en contenant
AU2003225964B2 (en) * 2002-03-28 2008-11-20 Merck Sharp & Dohme Corp. Substituted 2,3-diphenyl pyridines
FR2838438A1 (fr) * 2002-04-11 2003-10-17 Sanofi Synthelabo Derives de diphenylpyridine,leur preparation, les compositions pharmaceutiques en contenant
FR2838439B1 (fr) * 2002-04-11 2005-05-20 Sanofi Synthelabo Derives de terphenyle, leur preparation, les compositions pharmaceutqiues en contenant

Similar Documents

Publication Publication Date Title
JP2007514638A5 (enExample)
TW544453B (en) Novel guanidine mimics as factor Xa inhibitors
JP3325263B2 (ja) Cox−2のインヒビターとして有用なジアリールピリジンの製造方法
JP6724246B2 (ja) チオフェン化合物、その合成方法及び医療における応用
JP2007531756A5 (enExample)
JPH09503214A (ja) 抗炎症活性及び/又は鎮痛活性を有する硝酸エステル類及びそれらの製造方法
JP2007534638A5 (enExample)
JP2008526692A5 (enExample)
CN105384691B (zh) 一种谷氨酰胺酰基环化酶抑制剂的制备方法及应用
CN106632245B (zh) 氮取代基苯基吡唑类黄嘌呤氧化还原酶抑制剂及制备与应用
CZ293246B6 (cs) Způsob výroby 2-aryl-3-aryl-5-halogenpyridinů
CN102424659A (zh) 一种对甲砜基苯丝氨酸乙酯的合成方法
CN105384692A (zh) 一种谷氨酰胺酰基环化酶抑制剂
JP2006509781A5 (enExample)
CN106008403A (zh) 一种(E)-β-三氟甲基-烯烃磺酰胺类化合物的制备方法
JP2002529463A (ja) 化合物
JP2002510333A (ja) 1,5−ジフェニルピラゾール誘導体
TW201035050A (en) Bis aromatic compounds for use as LTC4 synthase inhibitors
KR20130119927A (ko) 이미다졸 유도체, 그의 제조 방법 및 용도
CN105601528A (zh) 一类以ent-贝叶烷型二萜为手性臂的分子钳化合物及其制备方法和应用
CN110016049A (zh) 一种磷酸吡哆醛的制备方法
CN110372614B (zh) 一种四氢喹喔啉类化合物及制备方法与应用
CN105399644A (zh) 一类以(1s,2s)-1,2-环己二胺为隔离基、以异斯特维醇为手性臂的分子钳化合物及其制备方法和应用
CN114621218B (zh) 一种唑吡坦中间体化合物
CN106496087B (zh) 一种通过脱羧偶联反应一锅法合成含硒类化合物的方法