JP2006519852A5 - - Google Patents
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- Publication number
- JP2006519852A5 JP2006519852A5 JP2006507175A JP2006507175A JP2006519852A5 JP 2006519852 A5 JP2006519852 A5 JP 2006519852A5 JP 2006507175 A JP2006507175 A JP 2006507175A JP 2006507175 A JP2006507175 A JP 2006507175A JP 2006519852 A5 JP2006519852 A5 JP 2006519852A5
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutical composition
- composition according
- salt
- carbon atoms
- less
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 *c1nc(C=C)c(C=C)[n]1 Chemical compound *c1nc(C=C)c(C=C)[n]1 0.000 description 1
- MFUFVMDJHGXUND-UHFFFAOYSA-N c1c[s]c(-c2nc3cccnc3[nH]2)c1 Chemical compound c1c[s]c(-c2nc3cccnc3[nH]2)c1 MFUFVMDJHGXUND-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US45403503P | 2003-03-12 | 2003-03-12 | |
| US45451403P | 2003-03-13 | 2003-03-13 | |
| US10/402,347 US7022712B2 (en) | 2002-03-26 | 2003-03-26 | Solubilization of weak bases |
| PCT/US2004/007786 WO2004081006A1 (en) | 2003-03-12 | 2004-03-12 | Weak base salts |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006519852A JP2006519852A (ja) | 2006-08-31 |
| JP2006519852A5 true JP2006519852A5 (enExample) | 2007-04-19 |
Family
ID=32995897
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006507175A Pending JP2006519852A (ja) | 2003-03-12 | 2004-03-12 | 弱塩基の塩 |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP1606290A1 (enExample) |
| JP (1) | JP2006519852A (enExample) |
| AU (1) | AU2004220053A1 (enExample) |
| CA (1) | CA2515289A1 (enExample) |
| MX (1) | MXPA05009564A (enExample) |
| WO (1) | WO2004081006A1 (enExample) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
| US7501426B2 (en) | 2004-02-18 | 2009-03-10 | Boehringer Ingelheim International Gmbh | 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions |
| DE102004054054A1 (de) | 2004-11-05 | 2006-05-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine |
| DE102005035891A1 (de) * | 2005-07-30 | 2007-02-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
| EP1852108A1 (en) | 2006-05-04 | 2007-11-07 | Boehringer Ingelheim Pharma GmbH & Co.KG | DPP IV inhibitor formulations |
| PE20080251A1 (es) | 2006-05-04 | 2008-04-25 | Boehringer Ingelheim Int | Usos de inhibidores de dpp iv |
| SG174054A1 (en) | 2006-05-04 | 2011-09-29 | Boehringer Ingelheim Int | Polymorphs |
| AR071175A1 (es) | 2008-04-03 | 2010-06-02 | Boehringer Ingelheim Int | Composicion farmaceutica que comprende un inhibidor de la dipeptidil-peptidasa-4 (dpp4) y un farmaco acompanante |
| KR20190016601A (ko) | 2008-08-06 | 2019-02-18 | 베링거 인겔하임 인터내셔날 게엠베하 | 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료 |
| UY32030A (es) | 2008-08-06 | 2010-03-26 | Boehringer Ingelheim Int | "tratamiento para diabetes en pacientes inapropiados para terapia con metformina" |
| KR20110067096A (ko) | 2008-09-10 | 2011-06-21 | 베링거 인겔하임 인터내셔날 게엠베하 | 당뇨병 및 관련 상태를 치료하기 위한 병용 요법 |
| US20200155558A1 (en) | 2018-11-20 | 2020-05-21 | Boehringer Ingelheim International Gmbh | Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug |
| AR074374A1 (es) * | 2008-11-19 | 2011-01-12 | Cephalon Inc | Formas de un compuesto de pirrolocarbazol fusionado, composiciones que las comprenden y su uso en el tratamiento de la angiogénesis y los tumores sólidos. |
| EA022310B1 (ru) | 2008-12-23 | 2015-12-30 | Бёрингер Ингельхайм Интернациональ Гмбх | Солевые формы органического соединения |
| AR074990A1 (es) | 2009-01-07 | 2011-03-02 | Boehringer Ingelheim Int | Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina |
| BR112012012641A2 (pt) | 2009-11-27 | 2020-08-11 | Boehringer Ingelheim International Gmbh | TRATAMENTO DE PACIENTES DIABÉTICOS GENOTIPADOS COM INIBIDORES DE DPP-lVTAL COMO LINAGLIPTINA |
| KR101927068B1 (ko) | 2010-05-05 | 2018-12-10 | 베링거 인겔하임 인터내셔날 게엠베하 | 체중 감소 치료에 후속하는 dpp-4 억제제에 의한 순차적 병용 요법 |
| CA2803504C (en) | 2010-06-24 | 2022-08-30 | Boehringer Ingelheim International Gmbh | A combination for diabetes therapy comprising linagliptin and a long-acting insulin |
| US9034883B2 (en) | 2010-11-15 | 2015-05-19 | Boehringer Ingelheim International Gmbh | Vasoprotective and cardioprotective antidiabetic therapy |
| EP3517539B1 (en) | 2011-07-15 | 2022-12-14 | Boehringer Ingelheim International GmbH | Substituted dimeric quinazoline derivative, its preparation and its use in pharmaceutical compositions for the treatment of type i and ii diabetes |
| US9555001B2 (en) | 2012-03-07 | 2017-01-31 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition and uses thereof |
| JP6224084B2 (ja) | 2012-05-14 | 2017-11-01 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 糸球体上皮細胞関連障害及び/又はネフローゼ症候群の治療に用いるdpp−4阻害薬としてのキサンチン誘導体 |
| EP4151218A1 (en) | 2012-05-14 | 2023-03-22 | Boehringer Ingelheim International GmbH | Linagliptin, a xanthine derivative as dpp-4 inhibitor, for use in the treatment of sirs and/or sepsis |
| WO2013174767A1 (en) | 2012-05-24 | 2013-11-28 | Boehringer Ingelheim International Gmbh | A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference |
| JP6615109B2 (ja) | 2014-02-28 | 2019-12-04 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Dpp−4阻害薬の医学的使用 |
| WO2017211979A1 (en) | 2016-06-10 | 2017-12-14 | Boehringer Ingelheim International Gmbh | Combinations of linagliptin and metformin |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1195180A (en) * | 1967-05-05 | 1970-06-17 | Du Pont | Use of Alkyl 2-Benzimidazole-Carbamate Salts a Fungicides |
| CA962588A (en) * | 1972-05-17 | 1975-02-11 | Her Majesty In Right Of Canada As Represented By The Minister Of The Env Ironment, And Canadian Patents And Development Limited | Method, apparatus, and fungicides for the treatment of trees subject to dutch elm disease and other fungus diseases |
| JPS5459338A (en) * | 1977-10-20 | 1979-05-12 | Takeda Chem Ind Ltd | Remedy for dermatomycosis |
| HU199431B (en) * | 1985-02-04 | 1990-02-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing carbendazim salts, and fungicide comprising such carbendazim salt as active ingredient |
| US6423734B1 (en) * | 1999-08-13 | 2002-07-23 | The Procter & Gamble Company | Method of preventing cancer |
-
2004
- 2004-03-12 MX MXPA05009564A patent/MXPA05009564A/es not_active Application Discontinuation
- 2004-03-12 CA CA002515289A patent/CA2515289A1/en not_active Abandoned
- 2004-03-12 EP EP04720454A patent/EP1606290A1/en not_active Withdrawn
- 2004-03-12 JP JP2006507175A patent/JP2006519852A/ja active Pending
- 2004-03-12 WO PCT/US2004/007786 patent/WO2004081006A1/en not_active Ceased
- 2004-03-12 AU AU2004220053A patent/AU2004220053A1/en not_active Abandoned
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