JP2011517697A5 - - Google Patents

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Publication number
JP2011517697A5
JP2011517697A5 JP2011505019A JP2011505019A JP2011517697A5 JP 2011517697 A5 JP2011517697 A5 JP 2011517697A5 JP 2011505019 A JP2011505019 A JP 2011505019A JP 2011505019 A JP2011505019 A JP 2011505019A JP 2011517697 A5 JP2011517697 A5 JP 2011517697A5
Authority
JP
Japan
Prior art keywords
aryl
alkyl
carbonyl
heterocycle
sulfinyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011505019A
Other languages
English (en)
Japanese (ja)
Other versions
JP2011517697A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2009/002344 external-priority patent/WO2009128913A1/en
Publication of JP2011517697A publication Critical patent/JP2011517697A/ja
Publication of JP2011517697A5 publication Critical patent/JP2011517697A5/ja
Pending legal-status Critical Current

Links

JP2011505019A 2008-04-14 2009-04-14 置換テトラサイクリン化合物 Pending JP2011517697A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4477308P 2008-04-14 2008-04-14
US61/044,773 2008-04-14
PCT/US2009/002344 WO2009128913A1 (en) 2008-04-14 2009-04-14 Substituted tetracycline compounds

Publications (2)

Publication Number Publication Date
JP2011517697A JP2011517697A (ja) 2011-06-16
JP2011517697A5 true JP2011517697A5 (enExample) 2013-05-23

Family

ID=41199392

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011505019A Pending JP2011517697A (ja) 2008-04-14 2009-04-14 置換テトラサイクリン化合物

Country Status (7)

Country Link
US (1) US20100022483A1 (enExample)
EP (1) EP2276342A4 (enExample)
JP (1) JP2011517697A (enExample)
AU (1) AU2009236631A1 (enExample)
CA (1) CA2721399A1 (enExample)
PE (1) PE20110069A1 (enExample)
WO (1) WO2009128913A1 (enExample)

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CN1893956A (zh) 2003-07-25 2007-01-10 沃纳奇尔科特公司 多西环素金属络合物固体剂型
CN101128206A (zh) * 2005-01-21 2008-02-20 沃纳奇尔科特公司 固体剂型形式的四环素类金属络合物
AU2009220171A1 (en) 2008-03-05 2009-09-11 Paratek Pharmaceuticals, Inc. Minocycline compounds and methods of use thereof
CN105367440A (zh) 2008-08-08 2016-03-02 四相制药公司 C7-氟取代的四环素化合物
CN102459153A (zh) 2009-05-08 2012-05-16 四相制药公司 四环素类化合物
HUE037852T2 (hu) 2009-08-28 2018-09-28 Tetraphase Pharmaceuticals Inc Tetraciklin-vegyületek
JP6522498B2 (ja) * 2012-05-30 2019-05-29 パラテック ファーマシューティカルズ インコーポレイテッド ７−二置換フェニルテトラサイクリン誘導体
EA031523B1 (ru) 2012-08-31 2019-01-31 Тетрафейз Фармасьютикалс, Инк. Тетрациклиновые соединения
HRP20240605T1 (hr) 2016-10-19 2024-07-19 Tetraphase Pharmaceuticals, Inc. Kristalni oblici eravaciklina
US10383884B2 (en) 2016-11-01 2019-08-20 Paratek Pharmaceuticals, Inc. 9-aminomethyl minocycline compounds and use thereof in treating community-acquired bacterial pneumonia (CABP)
WO2021183918A1 (en) * 2020-03-13 2021-09-16 Cmtx Biotech Inc. Methods of treating illnesses caused by coronavirus, swine flu and avian flu

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