JP2006506356A5 - - Google Patents

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Publication number
JP2006506356A5
JP2006506356A5 JP2004542551A JP2004542551A JP2006506356A5 JP 2006506356 A5 JP2006506356 A5 JP 2006506356A5 JP 2004542551 A JP2004542551 A JP 2004542551A JP 2004542551 A JP2004542551 A JP 2004542551A JP 2006506356 A5 JP2006506356 A5 JP 2006506356A5
Authority
JP
Japan
Prior art keywords
mixture
mmol
dissolved
diazabicyclo
dimethylformamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2004542551A
Other languages
English (en)
Japanese (ja)
Other versions
JP2006506356A (ja
JP4537853B2 (ja
Filing date
Publication date
Priority claimed from FR0212500A external-priority patent/FR2845388B1/fr
Application filed filed Critical
Publication of JP2006506356A publication Critical patent/JP2006506356A/ja
Publication of JP2006506356A5 publication Critical patent/JP2006506356A5/ja
Application granted granted Critical
Publication of JP4537853B2 publication Critical patent/JP4537853B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2004542551A 2002-10-08 2003-10-06 1,4−ジアザビシクロ[3.2.2]ノナンカルボキシアミド誘導体、それらの製造法およびそれらの治療用途 Expired - Fee Related JP4537853B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0212500A FR2845388B1 (fr) 2002-10-08 2002-10-08 Derives de 1,4-diazabicyclo[3.2.2]nonanecarboxamides, leur preparation et leur application en therapeutique
PCT/FR2003/002929 WO2004033456A2 (fr) 2002-10-08 2003-10-06 Derives de 1,4-diazabicyclo[3.2.2]nonanecarboxamides, leur preparation et leur application en therapeutique ayant trait au dysfonctionnement des recepteurs nicotiniques

Publications (3)

Publication Number Publication Date
JP2006506356A JP2006506356A (ja) 2006-02-23
JP2006506356A5 true JP2006506356A5 (https=) 2010-07-01
JP4537853B2 JP4537853B2 (ja) 2010-09-08

Family

ID=32011522

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004542551A Expired - Fee Related JP4537853B2 (ja) 2002-10-08 2003-10-06 1,4−ジアザビシクロ[3.2.2]ノナンカルボキシアミド誘導体、それらの製造法およびそれらの治療用途

Country Status (9)

Country Link
EP (1) EP1575960B1 (https=)
JP (1) JP4537853B2 (https=)
AR (1) AR041527A1 (https=)
AT (1) ATE425980T1 (https=)
AU (1) AU2003283500A1 (https=)
DE (1) DE60326757D1 (https=)
FR (1) FR2845388B1 (https=)
TW (1) TWI320413B (https=)
WO (1) WO2004033456A2 (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA05003317A (es) 2002-09-25 2005-07-05 Memory Pharm Corp Indazoles, benzotiazoles y benzoisotiazoles asi como preparacion y usos de los mismos.
RU2389729C2 (ru) 2003-12-22 2010-05-20 Мемори Фармасьютиклз Корпорейшн 1н-индазолы, 1, 2-бензизоксазолы и 1, 2-бензизотиазолы, их получение и применение
FR2865208B1 (fr) 2004-01-16 2009-01-16 Sanofi Synthelabo Derives de 1,4-diazabicyclo[3.2.1]octanecarboxmique, leur preparation et leur application en therapeutique
EP1735306A2 (en) 2004-03-25 2006-12-27 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof
CA2567977A1 (en) * 2004-04-22 2006-01-05 Memory Pharmaceutical Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof
NZ551712A (en) * 2004-05-07 2010-07-30 Memory Pharm Corp 1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles, 1,2-benzoisothiazoles, and chromones and preparations and uses thereof
KR20070034049A (ko) 2004-06-09 2007-03-27 글락소 그룹 리미티드 피롤로피리딘 유도체
CA2591817A1 (en) 2004-12-22 2006-06-29 Memory Pharmaceuticals Corporation Nicotinic alpha-7 receptor ligands and preparation and uses thereof
BRPI0619672A2 (pt) * 2005-11-09 2011-10-11 Memory Pharm Corp composto, composição farmacêutica, e, uso de um composto
EP1842541A1 (en) * 2006-03-29 2007-10-10 G.I.M.-Gesellschaft Für Innovative Medizin Gmbh Nfg Ohg Plant components and extracts and uses thereof
AU2008316895A1 (en) * 2007-10-22 2009-04-30 Memory Pharmaceuticals Corporation (1,4-diaza-bicyclo[3.2.2]non-6-en-4-yl)-heterocyclyl-methanone ligands for nicotinic acetylcholine receptors, useful for the treatment of disease
JP7746384B2 (ja) * 2020-12-08 2025-09-30 ディスアーム セラピューティクス, インコーポレイテッド Sarm1のベンゾピラゾール阻害剤

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ226000A (en) * 1987-09-10 1991-06-25 Merck Sharp & Dohme Oxadiazolyl-azabicycloheptanes and pharmaceutical compositions
FR2786770B1 (fr) * 1998-12-04 2001-01-19 Synthelabo Derives de 1,4-diazabicyclo[3.2.2.]nonane, leur preparation et leur application en therapeutique
FR2804430B1 (fr) * 2000-01-28 2002-03-22 Sanofi Synthelabo Derives de 4-heteroaryl-1,4-diazabicyclo[3.2.2] nonane, leur preparation et leur application en therapeutique
FR2809730B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo Derives de 1,4-diazabicyclo[3.2.2] nonanebenzoxazole, -benzothiazole et -benzimidazole, leur preparation et leur application therapeutique
US20020086871A1 (en) * 2000-12-29 2002-07-04 O'neill Brian Thomas Pharmaceutical composition for the treatment of CNS and other disorders

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