DE60326757D1 - 1,4-DIAZABICYCLOi3.2.2 NONANECARBOXAMIDES DERIVATE, DEREN HERSTELLUNG, UND DEREN THERAPEUTISCHE VERWENDUNG IM ZUSAMMENHANG MIT NIKOTINISCHEN REZEPTOR-STÖRUNGEN - Google Patents
1,4-DIAZABICYCLOi3.2.2 NONANECARBOXAMIDES DERIVATE, DEREN HERSTELLUNG, UND DEREN THERAPEUTISCHE VERWENDUNG IM ZUSAMMENHANG MIT NIKOTINISCHEN REZEPTOR-STÖRUNGENInfo
- Publication number
- DE60326757D1 DE60326757D1 DE60326757T DE60326757T DE60326757D1 DE 60326757 D1 DE60326757 D1 DE 60326757D1 DE 60326757 T DE60326757 T DE 60326757T DE 60326757 T DE60326757 T DE 60326757T DE 60326757 D1 DE60326757 D1 DE 60326757D1
- Authority
- DE
- Germany
- Prior art keywords
- nonanecarboxamides
- derivatives
- preparation
- connection
- therapeutic use
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 229960002715 nicotine Drugs 0.000 title 1
- SNICXCGAKADSCV-UHFFFAOYSA-N nicotine Natural products CN1CCCC1C1=CC=CN=C1 SNICXCGAKADSCV-UHFFFAOYSA-N 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0212500A FR2845388B1 (fr) | 2002-10-08 | 2002-10-08 | Derives de 1,4-diazabicyclo[3.2.2]nonanecarboxamides, leur preparation et leur application en therapeutique |
| PCT/FR2003/002929 WO2004033456A2 (fr) | 2002-10-08 | 2003-10-06 | Derives de 1,4-diazabicyclo[3.2.2]nonanecarboxamides, leur preparation et leur application en therapeutique ayant trait au dysfonctionnement des recepteurs nicotiniques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE60326757D1 true DE60326757D1 (de) | 2009-04-30 |
Family
ID=32011522
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE60326757T Expired - Lifetime DE60326757D1 (de) | 2002-10-08 | 2003-10-06 | 1,4-DIAZABICYCLOi3.2.2 NONANECARBOXAMIDES DERIVATE, DEREN HERSTELLUNG, UND DEREN THERAPEUTISCHE VERWENDUNG IM ZUSAMMENHANG MIT NIKOTINISCHEN REZEPTOR-STÖRUNGEN |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1575960B1 (https=) |
| JP (1) | JP4537853B2 (https=) |
| AR (1) | AR041527A1 (https=) |
| AT (1) | ATE425980T1 (https=) |
| AU (1) | AU2003283500A1 (https=) |
| DE (1) | DE60326757D1 (https=) |
| FR (1) | FR2845388B1 (https=) |
| TW (1) | TWI320413B (https=) |
| WO (1) | WO2004033456A2 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA05003317A (es) | 2002-09-25 | 2005-07-05 | Memory Pharm Corp | Indazoles, benzotiazoles y benzoisotiazoles asi como preparacion y usos de los mismos. |
| RU2389729C2 (ru) | 2003-12-22 | 2010-05-20 | Мемори Фармасьютиклз Корпорейшн | 1н-индазолы, 1, 2-бензизоксазолы и 1, 2-бензизотиазолы, их получение и применение |
| FR2865208B1 (fr) | 2004-01-16 | 2009-01-16 | Sanofi Synthelabo | Derives de 1,4-diazabicyclo[3.2.1]octanecarboxmique, leur preparation et leur application en therapeutique |
| EP1735306A2 (en) | 2004-03-25 | 2006-12-27 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof |
| CA2567977A1 (en) * | 2004-04-22 | 2006-01-05 | Memory Pharmaceutical Corporation | Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
| NZ551712A (en) * | 2004-05-07 | 2010-07-30 | Memory Pharm Corp | 1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles, 1,2-benzoisothiazoles, and chromones and preparations and uses thereof |
| KR20070034049A (ko) | 2004-06-09 | 2007-03-27 | 글락소 그룹 리미티드 | 피롤로피리딘 유도체 |
| CA2591817A1 (en) | 2004-12-22 | 2006-06-29 | Memory Pharmaceuticals Corporation | Nicotinic alpha-7 receptor ligands and preparation and uses thereof |
| BRPI0619672A2 (pt) * | 2005-11-09 | 2011-10-11 | Memory Pharm Corp | composto, composição farmacêutica, e, uso de um composto |
| EP1842541A1 (en) * | 2006-03-29 | 2007-10-10 | G.I.M.-Gesellschaft Für Innovative Medizin Gmbh Nfg Ohg | Plant components and extracts and uses thereof |
| AU2008316895A1 (en) * | 2007-10-22 | 2009-04-30 | Memory Pharmaceuticals Corporation | (1,4-diaza-bicyclo[3.2.2]non-6-en-4-yl)-heterocyclyl-methanone ligands for nicotinic acetylcholine receptors, useful for the treatment of disease |
| JP7746384B2 (ja) * | 2020-12-08 | 2025-09-30 | ディスアーム セラピューティクス, インコーポレイテッド | Sarm1のベンゾピラゾール阻害剤 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ226000A (en) * | 1987-09-10 | 1991-06-25 | Merck Sharp & Dohme | Oxadiazolyl-azabicycloheptanes and pharmaceutical compositions |
| FR2786770B1 (fr) * | 1998-12-04 | 2001-01-19 | Synthelabo | Derives de 1,4-diazabicyclo[3.2.2.]nonane, leur preparation et leur application en therapeutique |
| FR2804430B1 (fr) * | 2000-01-28 | 2002-03-22 | Sanofi Synthelabo | Derives de 4-heteroaryl-1,4-diazabicyclo[3.2.2] nonane, leur preparation et leur application en therapeutique |
| FR2809730B1 (fr) * | 2000-05-31 | 2002-07-19 | Sanofi Synthelabo | Derives de 1,4-diazabicyclo[3.2.2] nonanebenzoxazole, -benzothiazole et -benzimidazole, leur preparation et leur application therapeutique |
| US20020086871A1 (en) * | 2000-12-29 | 2002-07-04 | O'neill Brian Thomas | Pharmaceutical composition for the treatment of CNS and other disorders |
-
2002
- 2002-10-08 FR FR0212500A patent/FR2845388B1/fr not_active Expired - Fee Related
-
2003
- 2003-10-06 AT AT03775474T patent/ATE425980T1/de not_active IP Right Cessation
- 2003-10-06 EP EP03775474A patent/EP1575960B1/fr not_active Expired - Lifetime
- 2003-10-06 DE DE60326757T patent/DE60326757D1/de not_active Expired - Lifetime
- 2003-10-06 AU AU2003283500A patent/AU2003283500A1/en not_active Abandoned
- 2003-10-06 AR ARP030103628A patent/AR041527A1/es unknown
- 2003-10-06 JP JP2004542551A patent/JP4537853B2/ja not_active Expired - Fee Related
- 2003-10-06 WO PCT/FR2003/002929 patent/WO2004033456A2/fr not_active Ceased
- 2003-10-07 TW TW092127821A patent/TWI320413B/zh not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2006506356A (ja) | 2006-02-23 |
| WO2004033456A3 (fr) | 2004-05-27 |
| WO2004033456A2 (fr) | 2004-04-22 |
| AU2003283500A1 (en) | 2004-05-04 |
| ATE425980T1 (de) | 2009-04-15 |
| AR041527A1 (es) | 2005-05-18 |
| EP1575960B1 (fr) | 2009-03-18 |
| TWI320413B (en) | 2010-02-11 |
| FR2845388A1 (fr) | 2004-04-09 |
| AU2003283500A8 (en) | 2004-05-04 |
| EP1575960A2 (fr) | 2005-09-21 |
| FR2845388B1 (fr) | 2004-11-12 |
| TW200505926A (en) | 2005-02-16 |
| JP4537853B2 (ja) | 2010-09-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |