JP2005534661A5 - - Google Patents

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Publication number
JP2005534661A5
JP2005534661A5 JP2004511295A JP2004511295A JP2005534661A5 JP 2005534661 A5 JP2005534661 A5 JP 2005534661A5 JP 2004511295 A JP2004511295 A JP 2004511295A JP 2004511295 A JP2004511295 A JP 2004511295A JP 2005534661 A5 JP2005534661 A5 JP 2005534661A5
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JP
Japan
Prior art keywords
disease
injury
peripheral
alopecia
metastases
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2004511295A
Other languages
English (en)
Japanese (ja)
Other versions
JP4437075B2 (ja
JP2005534661A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/FR2003/001685 external-priority patent/WO2003104225A1/fr
Publication of JP2005534661A publication Critical patent/JP2005534661A/ja
Publication of JP2005534661A5 publication Critical patent/JP2005534661A5/ja
Application granted granted Critical
Publication of JP4437075B2 publication Critical patent/JP4437075B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2004511295A 2002-06-07 2003-06-05 ピペラジニルアシルピペリジン誘導体、それらの製造方法およびそれらの治療的用途 Expired - Fee Related JP4437075B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0207001 2002-06-07
PCT/FR2003/001685 WO2003104225A1 (fr) 2002-06-07 2003-06-05 Derives de piperazinylacylpiperidine, leur preparation et leur application en therapeutique

Publications (3)

Publication Number Publication Date
JP2005534661A JP2005534661A (ja) 2005-11-17
JP2005534661A5 true JP2005534661A5 (enExample) 2006-05-11
JP4437075B2 JP4437075B2 (ja) 2010-03-24

Family

ID=29724874

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2004511295A Expired - Fee Related JP4437075B2 (ja) 2002-06-07 2003-06-05 ピペラジニルアシルピペリジン誘導体、それらの製造方法およびそれらの治療的用途
JP2004511296A Expired - Fee Related JP4441401B2 (ja) 2002-06-07 2003-06-05 ピペラジニルアシルピペリジン誘導体、それらの製造およびそれらの治療的用途

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2004511296A Expired - Fee Related JP4441401B2 (ja) 2002-06-07 2003-06-05 ピペラジニルアシルピペリジン誘導体、それらの製造およびそれらの治療的用途

Country Status (29)

Country Link
US (2) US7294628B2 (enExample)
EP (2) EP1513835B1 (enExample)
JP (2) JP4437075B2 (enExample)
KR (1) KR100970812B1 (enExample)
CN (1) CN100448875C (enExample)
AR (2) AR040246A1 (enExample)
AT (2) ATE336491T1 (enExample)
AU (2) AU2003255645A1 (enExample)
BR (1) BR0311828A (enExample)
CA (1) CA2487840C (enExample)
CY (2) CY1107330T1 (enExample)
DE (2) DE60307632T2 (enExample)
DK (2) DK1513836T3 (enExample)
EA (1) EA007501B1 (enExample)
ES (2) ES2271637T3 (enExample)
HR (1) HRP20041157B1 (enExample)
IS (1) IS2302B (enExample)
MA (1) MA27233A1 (enExample)
ME (1) MEP11508A (enExample)
MX (1) MXPA04012341A (enExample)
NO (1) NO329669B1 (enExample)
NZ (1) NZ537044A (enExample)
PL (1) PL208711B1 (enExample)
PT (2) PT1513835E (enExample)
RS (2) RS52588B (enExample)
TW (2) TWI319400B (enExample)
UA (1) UA77526C2 (enExample)
WO (2) WO2003104226A1 (enExample)
ZA (1) ZA200409823B (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2862968B1 (fr) * 2003-12-01 2006-08-04 Sanofi Synthelabo Derives de 4-[(arylmethyl)aminomethyl]piperidine, leur preparation et leur application en therapeutique
FR2862967B1 (fr) * 2003-12-01 2006-08-04 Sanofi Synthelabo Derives de (4-phenylpiperazin-1-yl)acylpiperidine, leur preparation et leur application en therapeutique
US7723362B2 (en) * 2004-01-08 2010-05-25 Syngenta Crop Protection, Inc. Pesticidal heterocyclic dihaloallyl compounds
CN1984910A (zh) * 2004-07-16 2007-06-20 詹森药业有限公司 适用于神经变性疾病治疗的哌啶、哌嗪或者吗啉或它们的7元类似物的二聚化合物
BRPI0515483A (pt) * 2004-09-20 2008-07-22 Xenon Pharmaceuticals Inc derivados heterocìclicos para o tratamento de doenças mediadas por enzimas estearoil-coa desaturase
US7723328B2 (en) * 2005-04-15 2010-05-25 The University Of North Carolina At Chapel Hill Methods of facilitating cell survival using neurotrophin mimetics
EP2586778A3 (en) * 2007-03-15 2013-07-31 Merck Sharp & Dohme Corp. Pyridazinone derivatives useful as glucan synthase inhibitors
CA2688784A1 (en) * 2007-05-21 2008-11-27 Reviva Pharmaceuticals, Inc. Compositions, synthesis, and methods of using quinolinone based atypical antipsychotic agents
DE102007026341A1 (de) 2007-06-06 2008-12-11 Merck Patent Gmbh Benzoxazolonderivate
DE102007032507A1 (de) 2007-07-12 2009-04-02 Merck Patent Gmbh Pyridazinonderivate
FR2932481B1 (fr) * 2008-06-13 2010-10-08 Sanofi Aventis Derives de 4-{2-°4-phenyl-3,6-dihydro-2h-pyridin-1-yl!-2- oxo-alkyl}-1-piperazin-2-one, leur preparation et leur application en therapeutique.
FR2932482B1 (fr) * 2008-06-13 2010-10-08 Sanofi Aventis Nouveaux derives de (phenyl-3,6-dihydro-2h-pyridinyl)- (piperazinyl ponte)-1-alcanone et leur utilisation comme inhibiteurs de p75
CN102740856B (zh) 2009-11-12 2015-02-18 特罗菲克斯制药股份有限公司 神经营养蛋白模拟化合物及其盐的晶型
US10273219B2 (en) 2009-11-12 2019-04-30 Pharmatrophix, Inc. Crystalline forms of neurotrophin mimetic compounds and their salts
MX2012006776A (es) 2009-12-14 2012-10-05 Merck Patent Gmbh Inhibidores de la esfingosina quinasa.
FR2953839A1 (fr) * 2009-12-14 2011-06-17 Sanofi Aventis Nouveaux derives d'(heterocycle-piperidine condensee)-(piperazinyl)-1alcanone ou d'(heterocycle-pyrrolidine condensee)-(piperazinyl)-1alcanone et leur utilisation comme inhibiteurs de p75
FR2953836B1 (fr) 2009-12-14 2012-03-16 Sanofi Aventis Nouveaux derives (heterocycle-tetrahydro-pyridine)-(piperazinyl)-1-alcanone et (heterocycle-dihydro-pyrrolidine)-(piperazinyl)-1-alcanone et leur utilisation comme inhibiteurs de p75
EP2606894A1 (en) 2011-12-20 2013-06-26 Sanofi Novel therapeutic use of p75 receptor antagonists
CA3075727A1 (en) 2017-09-18 2019-03-21 Goldfinch Bio, Inc. Pyridazinones and methods of use thereof
RS65558B1 (sr) 2018-09-18 2024-06-28 Gfb Abc Llc Piridazinoni i postupci primene istih
EP3858439A1 (en) * 2020-02-03 2021-08-04 Esteve Pharmaceuticals, S.A. Amide derivatives having multimodal activity against pain

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1989003831A1 (en) * 1987-10-26 1989-05-05 Pfizer Inc. Anti-anxiety agents
FR2747041B1 (fr) * 1996-04-05 1998-05-22 Cird Galderma Utilisation de derives benzonaphtaleniques pour la fabrication de medicaments destines au traitement des neuropathies
US6468990B1 (en) * 1999-05-17 2002-10-22 Queen's University At Kingston Method of inhibiting binding of nerve growth factor to p75 NTR receptor
FR2803593B1 (fr) * 2000-01-06 2002-02-15 Sanofi Synthelabo Nouvelles tetrahydropyridines, procede pour leur preparation et compositions pharmaceutiques les contenant

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