JP2005526095A - 脆砕性の低い急速溶解投与剤型 - Google Patents

脆砕性の低い急速溶解投与剤型 Download PDF

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Publication number
JP2005526095A
JP2005526095A JP2003577853A JP2003577853A JP2005526095A JP 2005526095 A JP2005526095 A JP 2005526095A JP 2003577853 A JP2003577853 A JP 2003577853A JP 2003577853 A JP2003577853 A JP 2003577853A JP 2005526095 A JP2005526095 A JP 2005526095A
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chloride
bromide
dosage form
dimethyl
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JP2005526095A5 (enExample
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プラス,カール
ウェンデル,スーザン
ラディ,スティーブン
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エラン ファーマ インターナショナル,リミティド
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Zoology (AREA)
  • Medicinal Preparation (AREA)
JP2003577853A 2002-03-20 2003-03-20 脆砕性の低い急速溶解投与剤型 Withdrawn JP2005526095A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US36552602P 2002-03-20 2002-03-20
PCT/US2003/008544 WO2003080023A2 (en) 2002-03-20 2003-03-20 Fast dissolving dosage forms having reduced friability

Related Child Applications (1)

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JP2010178286A Division JP2010285451A (ja) 2002-03-20 2010-08-09 脆砕性の低い急速溶解投与剤型

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JP2005526095A true JP2005526095A (ja) 2005-09-02
JP2005526095A5 JP2005526095A5 (enExample) 2006-03-30

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JP2003577853A Withdrawn JP2005526095A (ja) 2002-03-20 2003-03-20 脆砕性の低い急速溶解投与剤型
JP2010178286A Pending JP2010285451A (ja) 2002-03-20 2010-08-09 脆砕性の低い急速溶解投与剤型

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JP2010178286A Pending JP2010285451A (ja) 2002-03-20 2010-08-09 脆砕性の低い急速溶解投与剤型

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US (1) US20030215502A1 (enExample)
EP (1) EP1487419A2 (enExample)
JP (2) JP2005526095A (enExample)
AU (1) AU2003222027A1 (enExample)
CA (1) CA2479735C (enExample)
WO (1) WO2003080023A2 (enExample)

Cited By (5)

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JP2009519985A (ja) * 2005-12-20 2009-05-21 レツク・フアーマシユーテイカルズ・デー・デー (e)−7−〔4−(4−フルオロフェニル)−6−イソプロピル−2−〔メチル(メチルスルホニル)アミノ〕ピリミジン−5−イル〕−(3r,5s)−3,5−ジヒドロキシヘプタ−6−エン酸を含む医薬組成物
JP2011195567A (ja) * 2010-02-26 2011-10-06 Daiichi Sankyo Co Ltd 錠剤
JP2012087104A (ja) * 2010-10-22 2012-05-10 Asahi Group Holdings Ltd 乾燥酵母を含有する錠剤
JP5373283B2 (ja) * 2005-07-08 2013-12-18 武田薬品工業株式会社 錠剤
JP2016074611A (ja) * 2014-10-02 2016-05-12 ライオン株式会社 経口投与用錠剤

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JP4547161B2 (ja) * 2004-01-22 2010-09-22 エスエス製薬株式会社 用時溶解型速溶性固形製剤
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EP1959966B1 (en) 2005-11-28 2020-06-03 Marinus Pharmaceuticals, Inc. Ganaxolone formulations and methods for the making and use thereof
BRPI0620578A2 (pt) * 2005-12-27 2011-12-06 Jubilant Organosys Ltd composição farmacêutica que dissolve na boca e processo para o preparo da mesma
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EP2151235B1 (de) * 2008-07-21 2011-02-16 Dr. Falk Pharma Gmbh Pharmazeutische Formulierung zur Behandlung des oberen Verdauungstraktes
US20100120776A1 (en) * 2008-11-12 2010-05-13 Hall Bioscience Corporation Carbocysteine medical foods
EP2253306A1 (en) 2009-05-18 2010-11-24 Royal College of Surgeons in Ireland Orodispersible dosage forms containing solid drug dispersions
EP3167875A1 (en) 2009-05-27 2017-05-17 Alkermes Pharma Ireland Limited Reduction of flake-like aggregation in nanoparticulate meloxicam compositions
US20110105441A1 (en) * 2009-10-30 2011-05-05 Fmc Corporation Stable Orally Disintegrating Tablets Having Low Superdisintegrant
US9012511B2 (en) 2010-05-19 2015-04-21 Alkermes Pharma Ireland Limited Nanoparticulate cinacalcet compositions
BR112013030093B1 (pt) * 2011-05-25 2019-12-10 Taiho Pharmaceutical Co Ltd comprimido revestido seco de desintegração oral contendo tegafur, gimeracilo e oteracilo potássico
US20140141078A1 (en) * 2012-09-15 2014-05-22 Jeffery K. Slaboden Dissolvable TableT
EP2886108B2 (de) 2013-12-23 2022-11-02 Dr. Falk Pharma Gmbh Optimierte pharmazeutische Formulierung zur Behandlung von entzündlichen Veränderungen des Ösophagus
JP6379884B2 (ja) * 2014-09-03 2018-08-29 ニプロ株式会社 口腔内崩壊錠、及び口腔内崩壊錠の製造方法
CN106822007B (zh) 2015-09-11 2021-12-31 西姆莱斯股份公司 口服制剂
US20180042903A1 (en) 2016-08-11 2018-02-15 Ovid Therapeutics Inc. Methods and compositions for treatment of epileptic disorders
US11096896B2 (en) 2018-05-17 2021-08-24 Fertin Pharma A/S Tablet dosage form for buccal absorption of active ingredients
US11096894B2 (en) * 2018-05-17 2021-08-24 Fertin Pharma A/S Oral tablet for induced saliva generation
US11135157B2 (en) 2018-05-17 2021-10-05 Fertin Pharma A/S Oral tablet for delivery of active ingredients to the throat
US20190350858A1 (en) 2018-05-17 2019-11-21 Fertin Pharma A/S Oral tablet for delivery of active ingredients to the gastrointestinal tract
US11052047B2 (en) 2018-05-17 2021-07-06 Fertin Pharma A/S Oral tablet suitable for fast release of active pharmaceutical ingredients
US11058633B2 (en) 2018-05-17 2021-07-13 Fertin Pharma A/S Disintegrating oral tablet suitable for active pharmaceutical ingredients
US11090263B2 (en) 2018-05-22 2021-08-17 Fertin Pharma A/S Tableted chewing gum suitable for active pharmaceutical ingredients
US11058641B2 (en) 2018-05-17 2021-07-13 Fertin Pharma A/S Oral tablet for taste masking of active ingredients
US11096895B2 (en) 2018-05-17 2021-08-24 Fertin Pharma A/S Oral tablet suitable for active pharmaceutical ingredients
WO2020118142A1 (en) 2018-12-07 2020-06-11 Marinus Pharmaceuticals, Inc. Ganaxolone for use in prophylaxis and treatment of pospartum depression
CA3145923A1 (en) 2019-08-05 2021-02-11 David Czekai Ganaxolone for use in treatment of status epilepticus
IL293525A (en) 2019-12-06 2022-08-01 Marinus Pharmaceuticals Inc Ganaxolone for use in the treatment of multiple sclerosis complex

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JP5373283B2 (ja) * 2005-07-08 2013-12-18 武田薬品工業株式会社 錠剤
JP2009519985A (ja) * 2005-12-20 2009-05-21 レツク・フアーマシユーテイカルズ・デー・デー (e)−7−〔4−(4−フルオロフェニル)−6−イソプロピル−2−〔メチル(メチルスルホニル)アミノ〕ピリミジン−5−イル〕−(3r,5s)−3,5−ジヒドロキシヘプタ−6−エン酸を含む医薬組成物
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JP2012087104A (ja) * 2010-10-22 2012-05-10 Asahi Group Holdings Ltd 乾燥酵母を含有する錠剤
JP2016074611A (ja) * 2014-10-02 2016-05-12 ライオン株式会社 経口投与用錠剤

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WO2003080023A2 (en) 2003-10-02
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AU2003222027A8 (en) 2003-10-08
CA2479735C (en) 2011-05-17
US20030215502A1 (en) 2003-11-20
JP2010285451A (ja) 2010-12-24
CA2479735A1 (en) 2003-10-02

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