JP2005519915A - Ｅｄｇ受容体に関連する症状の処置方法 - Google Patents

Ｅｄｇ受容体に関連する症状の処置方法 Download PDF

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JP2005519915A
JP2005519915A JP2003562260A JP2003562260A JP2005519915A JP 2005519915 A JP2005519915 A JP 2005519915A JP 2003562260 A JP2003562260 A JP 2003562260A JP 2003562260 A JP2003562260 A JP 2003562260A JP 2005519915 A JP2005519915 A JP 2005519915A
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alkyl
substituted
heteroaryl
edg
nhc
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JP2005519915A5 (fr
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ジーサ・シャンカー
デイビッド・ソロー−コルデロ
ジュリエット・ブイ・スペンサー
チャールズ・アール・グルチョウスキ
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Ceretek LLC
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Transplantation (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
JP2003562260A 2002-01-18 2003-01-21 Ｅｄｇ受容体に関連する症状の処置方法 Pending JP2005519915A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US35044502P 2002-01-18 2002-01-18
US35044602P 2002-01-18 2002-01-18
US35044802P 2002-01-18 2002-01-18
US35044702P 2002-01-18 2002-01-18
PCT/US2003/001881 WO2003062392A2 (fr) 2002-01-18 2003-01-21 Procedes pour traiter des pathologies associees a un recepteur d'edg

Publications (2)

Publication Number Publication Date
JP2005519915A true JP2005519915A (ja) 2005-07-07
JP2005519915A5 JP2005519915A5 (fr) 2006-04-20

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JP2003562260A Pending JP2005519915A (ja) 2002-01-18 2003-01-21 Ｅｄｇ受容体に関連する症状の処置方法

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EP (1) EP1513522A2 (fr)
JP (1) JP2005519915A (fr)
AU (1) AU2003214873A1 (fr)
CA (1) CA2473740A1 (fr)
WO (1) WO2003062392A2 (fr)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006511488A (ja) * 2002-10-15 2006-04-06 レノビス， インコーポレイテッド 炎症および神経障害性疼痛を処置するための、ニトロン化合物、同化合物を含有する薬学的化合物ならびに方法
WO2006137514A1 (fr) * 2005-06-23 2006-12-28 Locomogene, Inc. Agent thérapeutique pour le cancer qui comprend une substance capable d'inhiber l’expression ou la fonction de la synovioline comme principe actif et méthode pour dépister l'agent thérapeutique pour le cancer
JP2010524955A (ja) * 2007-04-16 2010-07-22 アボット・ラボラトリーズ ７−置換されていないインドール系Ｍｃｌ−１阻害薬
JP2011527286A (ja) * 2008-05-08 2011-10-27 アラーガン インコーポレイテッド 治療的に有効な置換ヒドロピリド［３，２，１−ｉｊ］キノリン化合物
JP2014152148A (ja) * 2013-02-12 2014-08-25 Kumamoto Health Science Univ ポリフェノール化合物
JP2015527378A (ja) * 2012-09-05 2015-09-17 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ Ｌｐａｒ置換シアノピラゾール化合物

Families Citing this family (119)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6953787B2 (en) 2002-04-12 2005-10-11 Arena Pharmaceuticals, Inc. 5HT2C receptor modulators
GB2397301A (en) * 2003-01-14 2004-07-21 Novo Pharmaceuticals Ltd De Substituted 1,3,5-triazine derivatives
US20070027190A1 (en) * 2003-01-17 2007-02-01 Moir Donald T Antibacterial fab i inhibitors
RU2358716C2 (ru) 2003-04-08 2009-06-20 Новартис Аг Органические соединения
SI2332921T1 (sl) 2003-06-17 2016-06-30 Arena Pharmaceuticals, Inc. 8-kloro-1-metil-2,3,4,5-tetrahidro-1H-3-benzazapin hidroklorid
CN101792417A (zh) 2003-06-17 2010-08-04 艾尼纳制药公司 用于治疗5ht2c受体相关疾病的苯并氮杂卓衍生物
US20060074124A1 (en) 2003-09-12 2006-04-06 Andrew Napper Methods of treating a disorder
WO2005026112A2 (fr) * 2003-09-12 2005-03-24 Elixir Pharmaceuticals, Inc. Procedes de traitement de troubles
CA2543918A1 (fr) * 2003-10-28 2005-05-12 Dean Wilson Benzimidazoles convenant comme modulateurs des canaux ioniques
JP2007523957A (ja) * 2004-02-25 2007-08-23 スミスクライン・ビーチャム・コーポレイション 新規化学化合物
KR100843526B1 (ko) 2004-02-27 2008-07-03 에프. 호프만-라 로슈 아게 피라졸의 접합 유도체
BRPI0508220A (pt) 2004-02-27 2007-07-17 Hoffmann La Roche derivados de pirazol heteroarila fundidos
CA2557268A1 (fr) 2004-02-27 2005-09-15 F. Hoffmann-La Roche Ag Derives d'indazole et compositions pharmaceutiques renfermant ceux-ci
GB0406867D0 (en) * 2004-03-26 2004-04-28 F2G Ltd Antifungal agents
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