JP2005509634A - マクロライドを含む医薬組成物 - Google Patents
マクロライドを含む医薬組成物 Download PDFInfo
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- JP2005509634A JP2005509634A JP2003537635A JP2003537635A JP2005509634A JP 2005509634 A JP2005509634 A JP 2005509634A JP 2003537635 A JP2003537635 A JP 2003537635A JP 2003537635 A JP2003537635 A JP 2003537635A JP 2005509634 A JP2005509634 A JP 2005509634A
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/133—Amines having hydroxy groups, e.g. sphingosine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
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- Pulmonology (AREA)
- Diabetes (AREA)
- Dermatology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Emergency Medicine (AREA)
- Urology & Nephrology (AREA)
- Transplantation (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0125443.2A GB0125443D0 (en) | 2001-10-23 | 2001-10-23 | Organic Compounds |
| GB0127341A GB0127341D0 (en) | 2001-11-14 | 2001-11-14 | Organic compounds |
| PCT/EP2002/011799 WO2003035068A1 (en) | 2001-10-23 | 2002-10-22 | Macrolides containing pharmaceutical compositions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005509634A true JP2005509634A (ja) | 2005-04-14 |
| JP2005509634A5 JP2005509634A5 (https=) | 2008-04-10 |
Family
ID=26246689
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003537635A Pending JP2005509634A (ja) | 2001-10-23 | 2002-10-22 | マクロライドを含む医薬組成物 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US7259170B2 (https=) |
| EP (1) | EP1439838A1 (https=) |
| JP (1) | JP2005509634A (https=) |
| KR (2) | KR100978971B1 (https=) |
| CN (1) | CN1307993C (https=) |
| AU (1) | AU2002346859C1 (https=) |
| BR (1) | BR0213463A (https=) |
| CA (1) | CA2458690C (https=) |
| EC (1) | ECSP045086A (https=) |
| GB (1) | GB0125443D0 (https=) |
| HU (1) | HUP0402108A3 (https=) |
| IL (1) | IL160973A0 (https=) |
| MX (1) | MXPA04003738A (https=) |
| NO (1) | NO20042074L (https=) |
| NZ (1) | NZ532412A (https=) |
| PL (1) | PL368533A1 (https=) |
| RU (1) | RU2321402C2 (https=) |
| WO (1) | WO2003035068A1 (https=) |
| ZA (1) | ZA200401711B (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005512946A (ja) * | 2001-05-09 | 2005-05-12 | ノバルティス アクチエンゲゼルシャフト | 選択的免疫調節法 |
| BR0306811A (pt) | 2002-01-11 | 2004-10-26 | Sankyo Co | Composto, éster farmacologicamente aceitável do mesmo, composição farmacêutica e métodos para prevenção ou tratamento de doenças autoimunes, da artrite reumatóide e da rejeição causada pelo transplante de vários órgãos em um mamìfero |
| GB0307867D0 (en) * | 2003-04-04 | 2003-05-14 | Novartis Ag | Pharmaceutical composition |
| JP2005272453A (ja) | 2004-02-24 | 2005-10-06 | Sankyo Co Ltd | アミノアルコール化合物 |
Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0427680A1 (en) * | 1989-11-09 | 1991-05-15 | Sandoz Ltd. | Heteroatoms-containing tricyclic compounds |
| GB2252041A (en) * | 1991-01-23 | 1992-07-29 | Fujisawa Pharmaceutical Co | Use of macrolide compounds in treatment of autoimmune myocarditis |
| EP0627406A1 (en) * | 1992-10-21 | 1994-12-07 | Yoshitomi Pharmaceutical Industries, Ltd. | 2-amino-1,3-propanediol compound and immunosuppressant |
| US5482965A (en) * | 1991-03-19 | 1996-01-09 | Rajadhyaksha; Vithal J. | Compositions and method comprising aminoalcohol derivatives as membrane penetration enhancers for physiological active agents |
| EP0778263A1 (en) * | 1994-08-22 | 1997-06-11 | Yoshitomi Pharmaceutical Industries, Ltd. | Benzene compound and medicinal use thereof |
| EP1002792A1 (en) * | 1997-04-04 | 2000-05-24 | Yoshitomi Pharmaceutical Industries, Ltd. | 2-aminopropane-1,3-diol compounds, medicinal use thereof, and intermediates in synthesizing the same |
| JP2001072585A (ja) * | 1999-06-30 | 2001-03-21 | Akira Matsumori | ウイルス性心筋炎の予防または治療薬剤 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE68921934T2 (de) | 1988-06-29 | 1995-10-19 | Merck & Co Inc | Immunsuppressives Agens. |
| US5352671A (en) * | 1989-11-09 | 1994-10-04 | Sandoz Ltd. | Heteroatoms-containing tricyclic compounds |
| US5247076A (en) * | 1991-09-09 | 1993-09-21 | Merck & Co., Inc. | Imidazolidyl macrolides having immunosuppressive activity |
| GB9203636D0 (en) * | 1992-02-19 | 1992-04-08 | Lucas Ind Plc | Fuel pumping apparatus |
| JPH08507789A (ja) | 1993-03-17 | 1996-08-20 | アボツト・ラボラトリーズ | 大環状アミド及び尿素免疫調節剤 |
| US5590460A (en) * | 1994-07-19 | 1997-01-07 | Tessera, Inc. | Method of making multilayer circuit |
| GB9521322D0 (en) | 1995-10-17 | 1995-12-20 | Sandoz Ltd | Organic compounds |
| JPH11209277A (ja) | 1998-01-19 | 1999-08-03 | Yoshitomi Pharmaceut Ind Ltd | 医薬組成物 |
| GB9624038D0 (en) | 1996-11-19 | 1997-01-08 | Sandoz Ltd | Organic compounds |
| GB9713730D0 (en) * | 1997-06-30 | 1997-09-03 | Ciba Geigy Ag | Organic compounds |
| GB0003932D0 (en) | 2000-02-18 | 2000-04-12 | Novartis Ag | Pharmaceutical compositions |
| EP1355588B1 (en) | 2000-12-22 | 2007-08-15 | Avantec Vascular Corporation | Device for delivery of therepeutic agents |
-
2001
- 2001-10-23 GB GBGB0125443.2A patent/GB0125443D0/en not_active Ceased
-
2002
- 2002-10-22 NZ NZ532412A patent/NZ532412A/en unknown
- 2002-10-22 RU RU2004116067/15A patent/RU2321402C2/ru not_active IP Right Cessation
- 2002-10-22 KR KR1020047005958A patent/KR100978971B1/ko not_active Expired - Fee Related
- 2002-10-22 EP EP02782975A patent/EP1439838A1/en not_active Withdrawn
- 2002-10-22 WO PCT/EP2002/011799 patent/WO2003035068A1/en not_active Ceased
- 2002-10-22 MX MXPA04003738A patent/MXPA04003738A/es active IP Right Grant
- 2002-10-22 CA CA2458690A patent/CA2458690C/en not_active Expired - Fee Related
- 2002-10-22 CN CNB028211588A patent/CN1307993C/zh not_active Expired - Fee Related
- 2002-10-22 JP JP2003537635A patent/JP2005509634A/ja active Pending
- 2002-10-22 IL IL16097302A patent/IL160973A0/xx unknown
- 2002-10-22 AU AU2002346859A patent/AU2002346859C1/en not_active Ceased
- 2002-10-22 HU HU0402108A patent/HUP0402108A3/hu unknown
- 2002-10-22 BR BR0213463-2A patent/BR0213463A/pt not_active IP Right Cessation
- 2002-10-22 PL PL02368533A patent/PL368533A1/xx not_active Application Discontinuation
- 2002-10-22 US US10/492,439 patent/US7259170B2/en not_active Expired - Fee Related
- 2002-10-22 KR KR1020097021354A patent/KR20090114483A/ko not_active Ceased
-
2004
- 2004-03-02 ZA ZA200401711A patent/ZA200401711B/en unknown
- 2004-04-23 EC EC2004005086A patent/ECSP045086A/es unknown
- 2004-05-19 NO NO20042074A patent/NO20042074L/no not_active Application Discontinuation
Patent Citations (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0427680A1 (en) * | 1989-11-09 | 1991-05-15 | Sandoz Ltd. | Heteroatoms-containing tricyclic compounds |
| GB2252041A (en) * | 1991-01-23 | 1992-07-29 | Fujisawa Pharmaceutical Co | Use of macrolide compounds in treatment of autoimmune myocarditis |
| US5482965A (en) * | 1991-03-19 | 1996-01-09 | Rajadhyaksha; Vithal J. | Compositions and method comprising aminoalcohol derivatives as membrane penetration enhancers for physiological active agents |
| EP0627406A1 (en) * | 1992-10-21 | 1994-12-07 | Yoshitomi Pharmaceutical Industries, Ltd. | 2-amino-1,3-propanediol compound and immunosuppressant |
| JP2579602B2 (ja) * | 1992-10-21 | 1997-02-05 | 吉富製薬株式会社 | ２−アミノ−１，３−プロパンジオール化合物および免疫抑制剤 |
| EP0778263A1 (en) * | 1994-08-22 | 1997-06-11 | Yoshitomi Pharmaceutical Industries, Ltd. | Benzene compound and medicinal use thereof |
| EP1002792A1 (en) * | 1997-04-04 | 2000-05-24 | Yoshitomi Pharmaceutical Industries, Ltd. | 2-aminopropane-1,3-diol compounds, medicinal use thereof, and intermediates in synthesizing the same |
| JP2001072585A (ja) * | 1999-06-30 | 2001-03-21 | Akira Matsumori | ウイルス性心筋炎の予防または治療薬剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20040192716A1 (en) | 2004-09-30 |
| CA2458690A1 (en) | 2003-05-01 |
| CA2458690C (en) | 2011-01-25 |
| ECSP045086A (es) | 2004-06-28 |
| PL368533A1 (en) | 2005-04-04 |
| KR20090114483A (ko) | 2009-11-03 |
| KR100978971B1 (ko) | 2010-08-30 |
| WO2003035068A1 (en) | 2003-05-01 |
| BR0213463A (pt) | 2004-11-09 |
| ZA200401711B (en) | 2004-10-21 |
| HUP0402108A3 (en) | 2008-02-28 |
| IL160973A0 (en) | 2004-08-31 |
| AU2002346859C1 (en) | 2008-07-10 |
| NO20042074L (no) | 2004-05-19 |
| MXPA04003738A (es) | 2004-07-23 |
| CN1307993C (zh) | 2007-04-04 |
| AU2002346859B2 (en) | 2006-03-02 |
| RU2321402C2 (ru) | 2008-04-10 |
| CN1575173A (zh) | 2005-02-02 |
| US7259170B2 (en) | 2007-08-21 |
| KR20040052250A (ko) | 2004-06-22 |
| EP1439838A1 (en) | 2004-07-28 |
| RU2004116067A (ru) | 2005-04-20 |
| NZ532412A (en) | 2006-01-27 |
| HUP0402108A2 (hu) | 2005-02-28 |
| GB0125443D0 (en) | 2001-12-12 |
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