JP2005502608A - 抗コリン作用剤とコルチコステロイドとβ刺激剤を含む新規な医薬組成物 - Google Patents
抗コリン作用剤とコルチコステロイドとβ刺激剤を含む新規な医薬組成物 Download PDFInfo
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- JP2005502608A JP2005502608A JP2003506888A JP2003506888A JP2005502608A JP 2005502608 A JP2005502608 A JP 2005502608A JP 2003506888 A JP2003506888 A JP 2003506888A JP 2003506888 A JP2003506888 A JP 2003506888A JP 2005502608 A JP2005502608 A JP 2005502608A
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- 238000003756 stirring Methods 0.000 description 1
- 229960004793 sucrose Drugs 0.000 description 1
- 238000000967 suction filtration Methods 0.000 description 1
- HGKLFYLYWZXWPO-UHFFFAOYSA-N sulfo benzoate Chemical compound OS(=O)(=O)OC(=O)C1=CC=CC=C1 HGKLFYLYWZXWPO-UHFFFAOYSA-N 0.000 description 1
- 229950007862 sulfonterol Drugs 0.000 description 1
- 125000000472 sulfonyl group Chemical group *S(*)(=O)=O 0.000 description 1
- 150000003467 sulfuric acid derivatives Chemical class 0.000 description 1
- 230000001975 sympathomimetic effect Effects 0.000 description 1
- 230000002195 synergetic effect Effects 0.000 description 1
- 238000011287 therapeutic dose Methods 0.000 description 1
- JOXIMZWYDAKGHI-UHFFFAOYSA-N toluene-4-sulfonic acid Chemical compound CC1=CC=C(S(O)(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-N 0.000 description 1
- 239000002699 waste material Substances 0.000 description 1
- 229950000339 xinafoate Drugs 0.000 description 1
- 239000000811 xylitol Substances 0.000 description 1
- 235000010447 xylitol Nutrition 0.000 description 1
- HEBKCHPVOIAQTA-SCDXWVJYSA-N xylitol Chemical compound OC[C@H](O)[C@@H](O)[C@H](O)CO HEBKCHPVOIAQTA-SCDXWVJYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/537—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines spiro-condensed or forming part of bridged ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10130371A DE10130371A1 (de) | 2001-06-23 | 2001-06-23 | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika, Corticosteroiden und Betamimetika |
| PCT/EP2002/005896 WO2003000241A2 (de) | 2001-06-23 | 2002-05-29 | Neue arzneimittelkompositionen auf der basis von anticholinergika; corticosteroiden und betamimetika zur behandlung von entzündlichen und/oder obstruktiven atemwegserkrankungen |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005502608A true JP2005502608A (ja) | 2005-01-27 |
| JP2005502608A5 JP2005502608A5 (https=) | 2006-01-05 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003506888A Pending JP2005502608A (ja) | 2001-06-23 | 2002-05-29 | 抗コリン作用剤とコルチコステロイドとβ刺激剤を含む新規な医薬組成物 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20090088408A1 (https=) |
| EP (1) | EP1408967B1 (https=) |
| JP (1) | JP2005502608A (https=) |
| AT (1) | ATE446756T1 (https=) |
| AU (1) | AU2002316935A1 (https=) |
| CA (1) | CA2455167C (https=) |
| CY (1) | CY1109712T1 (https=) |
| DE (2) | DE10130371A1 (https=) |
| DK (1) | DK1408967T3 (https=) |
| ES (1) | ES2332883T3 (https=) |
| MX (1) | MXPA03011515A (https=) |
| PT (1) | PT1408967E (https=) |
| SI (1) | SI1408967T1 (https=) |
| WO (1) | WO2003000241A2 (https=) |
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| JP2005539046A (ja) * | 2002-08-29 | 2005-12-22 | シプラ・リミテッド | 特異的な抗コリン作用薬、β−２アゴニスト、および副腎皮質ステロイドを含む、治療薬および組成物 |
| JP2006508044A (ja) * | 2002-07-31 | 2006-03-09 | ザ・リージエンツ・オブ・ザ・ユニバーシテイ・オブ・カリフオルニア | 腫瘍の治療方法 |
| JP2008528565A (ja) * | 2005-01-31 | 2008-07-31 | ブレス リミテッド | ネブライザー処方物 |
| JP2008530176A (ja) * | 2005-02-19 | 2008-08-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 呼吸系疾患を治療するための新規な長く作用するベータミメチックス |
| JP2008532973A (ja) * | 2005-03-09 | 2008-08-21 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 抗コリン作用薬とｐｄｅ５−阻害剤に基づく新規な医薬組成物 |
| JP2008534611A (ja) * | 2005-03-30 | 2008-08-28 | シェーリング コーポレイション | 抗コリン作用薬、コルチコステロイドおよび長時間作用性βアゴニストを合わせる薬物および方法 |
| JP2008538758A (ja) * | 2005-04-23 | 2008-11-06 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 抗コリン作用薬に加えてベータ受容体刺激薬及びステロイドを含有する吸入用の医薬組成物 |
| JP2010500318A (ja) * | 2006-08-07 | 2010-01-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 呼吸器疾患の治療用医薬組成物 |
| JP2010501022A (ja) * | 2006-08-18 | 2010-01-14 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | βアゴニストの吸入用エアロゾル製剤 |
| JP2013531056A (ja) * | 2010-07-16 | 2013-08-01 | シプラ・リミテッド | Ｒ（＋）ブデソニド及び１以上の気管支拡張剤を含む医薬組成物 |
| JP2017515835A (ja) * | 2014-05-12 | 2017-06-15 | テバ ファーマシューティカルズ ヨーロッパ ベスローテン ベンノートシャップ | Ｃｏｐｄの治療のためのチオトロピウムブロミド、フォルモテロール及びブデソニドの組み合わせ |
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| ES2165768B1 (es) | 1999-07-14 | 2003-04-01 | Almirall Prodesfarma Sa | Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen. |
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| JP2006508044A (ja) * | 2002-07-31 | 2006-03-09 | ザ・リージエンツ・オブ・ザ・ユニバーシテイ・オブ・カリフオルニア | 腫瘍の治療方法 |
| JP2005539046A (ja) * | 2002-08-29 | 2005-12-22 | シプラ・リミテッド | 特異的な抗コリン作用薬、β−２アゴニスト、および副腎皮質ステロイドを含む、治療薬および組成物 |
| JP2008528565A (ja) * | 2005-01-31 | 2008-07-31 | ブレス リミテッド | ネブライザー処方物 |
| JP2008530176A (ja) * | 2005-02-19 | 2008-08-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 呼吸系疾患を治療するための新規な長く作用するベータミメチックス |
| JP2008532973A (ja) * | 2005-03-09 | 2008-08-21 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 抗コリン作用薬とｐｄｅ５−阻害剤に基づく新規な医薬組成物 |
| JP2008534611A (ja) * | 2005-03-30 | 2008-08-28 | シェーリング コーポレイション | 抗コリン作用薬、コルチコステロイドおよび長時間作用性βアゴニストを合わせる薬物および方法 |
| JP2008538758A (ja) * | 2005-04-23 | 2008-11-06 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 抗コリン作用薬に加えてベータ受容体刺激薬及びステロイドを含有する吸入用の医薬組成物 |
| JP2010500318A (ja) * | 2006-08-07 | 2010-01-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 呼吸器疾患の治療用医薬組成物 |
| JP2010501022A (ja) * | 2006-08-18 | 2010-01-14 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | βアゴニストの吸入用エアロゾル製剤 |
| JP2013531056A (ja) * | 2010-07-16 | 2013-08-01 | シプラ・リミテッド | Ｒ（＋）ブデソニド及び１以上の気管支拡張剤を含む医薬組成物 |
| JP2017039736A (ja) * | 2010-07-16 | 2017-02-23 | シプラ・リミテッド | Ｒ（＋）ブデソニド及び１以上の気管支拡張剤を含む医薬組成物 |
| JP2018199684A (ja) * | 2010-07-16 | 2018-12-20 | シプラ・リミテッド | Ｒ（＋）ブデソニド及び１以上の気管支拡張剤を含む医薬組成物 |
| US11077124B2 (en) | 2010-07-16 | 2021-08-03 | Cipla Limited | Pharmaceutical compositions |
| US12472190B2 (en) | 2010-07-16 | 2025-11-18 | Cipla Limited | Pharmaceutical compositions |
| JP2017515835A (ja) * | 2014-05-12 | 2017-06-15 | テバ ファーマシューティカルズ ヨーロッパ ベスローテン ベンノートシャップ | Ｃｏｐｄの治療のためのチオトロピウムブロミド、フォルモテロール及びブデソニドの組み合わせ |
Also Published As
| Publication number | Publication date |
|---|---|
| DE50213966D1 (de) | 2009-12-10 |
| EP1408967B1 (de) | 2009-10-28 |
| DE10130371A1 (de) | 2003-01-02 |
| ES2332883T3 (es) | 2010-02-15 |
| CY1109712T1 (el) | 2014-08-13 |
| SI1408967T1 (sl) | 2010-02-26 |
| AU2002316935A1 (en) | 2003-01-08 |
| WO2003000241A2 (de) | 2003-01-03 |
| WO2003000241A3 (de) | 2003-12-11 |
| CA2455167C (en) | 2010-10-05 |
| CA2455167A1 (en) | 2003-01-03 |
| PT1408967E (pt) | 2009-11-25 |
| DK1408967T3 (da) | 2010-03-08 |
| US20090088408A1 (en) | 2009-04-02 |
| MXPA03011515A (es) | 2004-03-18 |
| ATE446756T1 (de) | 2009-11-15 |
| EP1408967A2 (de) | 2004-04-21 |
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