JP2004520335A - 興奮性アミノ酸レセプターアンタゴニスト - Google Patents
興奮性アミノ酸レセプターアンタゴニスト Download PDFInfo
- Publication number
- JP2004520335A JP2004520335A JP2002554680A JP2002554680A JP2004520335A JP 2004520335 A JP2004520335 A JP 2004520335A JP 2002554680 A JP2002554680 A JP 2002554680A JP 2002554680 A JP2002554680 A JP 2002554680A JP 2004520335 A JP2004520335 A JP 2004520335A
- Authority
- JP
- Japan
- Prior art keywords
- pharmaceutically acceptable
- compound
- alkyl
- acceptable salt
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- AZNNFRBTUPHBIE-WIJBJCKWSA-N CCOC([C@H](C1)N(CC(CC2)CC(C3)C2CN[C@@H]3C(OCC)=O)CC1(F)F)=O Chemical compound CCOC([C@H](C1)N(CC(CC2)CC(C3)C2CN[C@@H]3C(OCC)=O)CC1(F)F)=O AZNNFRBTUPHBIE-WIJBJCKWSA-N 0.000 description 1
- OXQXJYQSWZFDBB-IUCVHNFVSA-N OC([C@H](C1)N(CC(CC2)CC(C3)[C@@H]2CN[C@@H]3C(O)=O)CC1(F)F)=O Chemical compound OC([C@H](C1)N(CC(CC2)CC(C3)[C@@H]2CN[C@@H]3C(O)=O)CC1(F)F)=O OXQXJYQSWZFDBB-IUCVHNFVSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US26001401P | 2001-01-05 | 2001-01-05 | |
| PCT/US2001/044715 WO2002053561A1 (en) | 2001-01-05 | 2001-12-20 | Excitatory amino acid receptor antagonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004520335A true JP2004520335A (ja) | 2004-07-08 |
| JP2004520335A5 JP2004520335A5 (pl) | 2005-12-22 |
Family
ID=22987455
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002554680A Pending JP2004520335A (ja) | 2001-01-05 | 2001-12-20 | 興奮性アミノ酸レセプターアンタゴニスト |
Country Status (23)
| Country | Link |
|---|---|
| EP (1) | EP1351955A1 (pl) |
| JP (1) | JP2004520335A (pl) |
| KR (1) | KR20030066797A (pl) |
| CN (1) | CN1484642A (pl) |
| AR (1) | AR035679A1 (pl) |
| BR (1) | BR0116672A (pl) |
| CA (1) | CA2431545A1 (pl) |
| CZ (1) | CZ20031856A3 (pl) |
| DZ (1) | DZ3460A1 (pl) |
| EA (1) | EA200300770A1 (pl) |
| EC (1) | ECSP034682A (pl) |
| HR (1) | HRP20030544A2 (pl) |
| HU (1) | HUP0302528A2 (pl) |
| IL (1) | IL156138A0 (pl) |
| MX (1) | MXPA03005981A (pl) |
| NO (1) | NO20032973D0 (pl) |
| NZ (1) | NZ525821A (pl) |
| PE (1) | PE20020792A1 (pl) |
| PL (1) | PL361934A1 (pl) |
| SK (1) | SK8242003A3 (pl) |
| TW (1) | TW591023B (pl) |
| WO (1) | WO2002053561A1 (pl) |
| ZA (1) | ZA200304311B (pl) |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5284957A (en) * | 1992-09-03 | 1994-02-08 | Eli Lilly And Company | Excitatory amino acid receptor antagonists |
| KR20010040711A (ko) * | 1998-02-06 | 2001-05-15 | 피터 기딩스 | 파록세틴의 염 |
| GB9908175D0 (en) * | 1999-04-09 | 1999-06-02 | Lilly Co Eli | Method of treating neurological disorders |
| EP1200073B1 (en) * | 1999-07-06 | 2007-01-10 | Eli Lilly And Company | SELECTIVE iGluR 5? RECEPTOR ANTAGONISTS FOR THE TREATMENT OF MIGRAINE |
-
2001
- 2001-12-20 EA EA200300770A patent/EA200300770A1/ru unknown
- 2001-12-20 CN CNA018217508A patent/CN1484642A/zh active Pending
- 2001-12-20 SK SK824-2003A patent/SK8242003A3/sk unknown
- 2001-12-20 PL PL01361934A patent/PL361934A1/pl not_active Application Discontinuation
- 2001-12-20 MX MXPA03005981A patent/MXPA03005981A/es unknown
- 2001-12-20 EP EP01995980A patent/EP1351955A1/en not_active Withdrawn
- 2001-12-20 HU HU0302528A patent/HUP0302528A2/hu unknown
- 2001-12-20 BR BR0116672-7A patent/BR0116672A/pt not_active IP Right Cessation
- 2001-12-20 NZ NZ525821A patent/NZ525821A/en unknown
- 2001-12-20 KR KR10-2003-7008977A patent/KR20030066797A/ko not_active Application Discontinuation
- 2001-12-20 WO PCT/US2001/044715 patent/WO2002053561A1/en not_active Application Discontinuation
- 2001-12-20 IL IL15613801A patent/IL156138A0/xx unknown
- 2001-12-20 CZ CZ20031856A patent/CZ20031856A3/cs unknown
- 2001-12-20 CA CA002431545A patent/CA2431545A1/en not_active Abandoned
- 2001-12-20 JP JP2002554680A patent/JP2004520335A/ja active Pending
- 2001-12-20 DZ DZ013460A patent/DZ3460A1/fr active
-
2002
- 2002-01-04 PE PE2002000003A patent/PE20020792A1/es not_active Application Discontinuation
- 2002-01-04 TW TW091100071A patent/TW591023B/zh not_active IP Right Cessation
- 2002-01-04 AR ARP020100030A patent/AR035679A1/es not_active Application Discontinuation
-
2003
- 2003-06-02 ZA ZA200304311A patent/ZA200304311B/en unknown
- 2003-06-27 NO NO20032973A patent/NO20032973D0/no not_active Application Discontinuation
- 2003-07-03 HR HR20030544A patent/HRP20030544A2/hr not_active Application Discontinuation
- 2003-07-03 EC EC2003004682A patent/ECSP034682A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20030066797A (ko) | 2003-08-09 |
| PL361934A1 (pl) | 2004-10-18 |
| SK8242003A3 (en) | 2004-01-08 |
| CZ20031856A3 (cs) | 2003-09-17 |
| CA2431545A1 (en) | 2002-07-11 |
| MXPA03005981A (es) | 2003-09-10 |
| IL156138A0 (en) | 2003-12-23 |
| HRP20030544A2 (en) | 2004-08-31 |
| ZA200304311B (en) | 2004-09-02 |
| PE20020792A1 (es) | 2002-09-06 |
| HUP0302528A2 (hu) | 2003-11-28 |
| NO20032973L (no) | 2003-06-27 |
| ECSP034682A (es) | 2003-08-29 |
| BR0116672A (pt) | 2003-09-23 |
| TW591023B (en) | 2004-06-11 |
| NO20032973D0 (no) | 2003-06-27 |
| NZ525821A (en) | 2004-07-30 |
| EA200300770A1 (ru) | 2003-10-30 |
| DZ3460A1 (fr) | 2002-07-11 |
| WO2002053561A1 (en) | 2002-07-11 |
| AR035679A1 (es) | 2004-06-23 |
| EP1351955A1 (en) | 2003-10-15 |
| CN1484642A (zh) | 2004-03-24 |
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| JP2004520335A5 (pl) | ||
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20040831 |
|
| A621 | Written request for application examination |
Free format text: JAPANESE INTERMEDIATE CODE: A621 Effective date: 20040831 |
|
| A131 | Notification of reasons for refusal |
Free format text: JAPANESE INTERMEDIATE CODE: A131 Effective date: 20080325 |
|
| A02 | Decision of refusal |
Free format text: JAPANESE INTERMEDIATE CODE: A02 Effective date: 20080819 |