JP2003532724A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2003532724A5 JP2003532724A5 JP2001582319A JP2001582319A JP2003532724A5 JP 2003532724 A5 JP2003532724 A5 JP 2003532724A5 JP 2001582319 A JP2001582319 A JP 2001582319A JP 2001582319 A JP2001582319 A JP 2001582319A JP 2003532724 A5 JP2003532724 A5 JP 2003532724A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compounds
- compound
- pharmaceutically acceptable
- acid addition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 C*1C2=CC=S(*)=CC=C2*=C1 Chemical compound C*1C2=CC=S(*)=CC=C2*=C1 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0011071.8 | 2000-05-08 | ||
| GBGB0011071.8A GB0011071D0 (en) | 2000-05-08 | 2000-05-08 | Organic compounds |
| PCT/EP2001/005162 WO2001085718A1 (en) | 2000-05-08 | 2001-05-07 | Hydantoin derivatives with affinity for somatostatin receptors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2003532724A JP2003532724A (ja) | 2003-11-05 |
| JP2003532724A5 true JP2003532724A5 (https=) | 2008-06-19 |
Family
ID=9891182
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001582319A Pending JP2003532724A (ja) | 2000-05-08 | 2001-05-07 | ソマトスタチン誘導体に親和性を有する、ヒダントイン誘導体 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US7019004B2 (https=) |
| EP (1) | EP1282617B1 (https=) |
| JP (1) | JP2003532724A (https=) |
| AT (1) | ATE441642T1 (https=) |
| AU (1) | AU7399801A (https=) |
| CA (1) | CA2405968A1 (https=) |
| DE (1) | DE60139770D1 (https=) |
| ES (1) | ES2330305T3 (https=) |
| GB (1) | GB0011071D0 (https=) |
| PT (1) | PT1282617E (https=) |
| WO (1) | WO2001085718A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7186855B2 (en) | 2001-06-11 | 2007-03-06 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| US8048917B2 (en) | 2005-04-06 | 2011-11-01 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| US7232924B2 (en) | 2001-06-11 | 2007-06-19 | Xenoport, Inc. | Methods for synthesis of acyloxyalkyl derivatives of GABA analogs |
| US6818787B2 (en) | 2001-06-11 | 2004-11-16 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| AU2002363655A1 (en) * | 2001-11-14 | 2003-05-26 | Novartis Ag | Non-peptide somatostatin receptor ligands |
| US7189856B2 (en) | 2001-12-28 | 2007-03-13 | Gideon Shapiro | Non-peptide somatostatin receptor ligands |
| SI2384753T1 (sl) | 2003-08-29 | 2016-06-30 | The Brigham And Women's Hospital, Inc. | Hidantoinski derivati kot inhibitorji celične nekroze |
| CA2772760A1 (en) | 2008-12-23 | 2010-07-01 | President And Fellows Of Harvard College | Small molecule inhibitors of necroptosis |
| US9725452B2 (en) | 2013-03-15 | 2017-08-08 | Presidents And Fellows Of Harvard College | Substituted indoles and pyrroles as RIP kinase inhibitors |
| EP3229807A4 (en) | 2014-12-11 | 2018-10-17 | President and Fellows of Harvard College | Inhibitors of cellular necrosis and related methods |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5859190A (en) * | 1997-02-04 | 1999-01-12 | Trega Biosciences, Inc. | Combinatorial libraries of hydantoin and thiohydantoin derivatives, methods of making the libraries and compounds therein |
| FR2796945B1 (fr) * | 1999-07-30 | 2002-06-28 | Sod Conseils Rech Applic | Nouveaux derives d'hydantoines, de thiohydantoines, de pyrimidinediones et de thioxopyrimidinones, leurs procedes de preparation et leur application a titre de medicaments |
| AU2002363655A1 (en) * | 2001-11-14 | 2003-05-26 | Novartis Ag | Non-peptide somatostatin receptor ligands |
| US7189856B2 (en) * | 2001-12-28 | 2007-03-13 | Gideon Shapiro | Non-peptide somatostatin receptor ligands |
-
2000
- 2000-05-08 GB GBGB0011071.8A patent/GB0011071D0/en not_active Ceased
-
2001
- 2001-05-07 PT PT01940412T patent/PT1282617E/pt unknown
- 2001-05-07 ES ES01940412T patent/ES2330305T3/es not_active Expired - Lifetime
- 2001-05-07 WO PCT/EP2001/005162 patent/WO2001085718A1/en not_active Ceased
- 2001-05-07 CA CA002405968A patent/CA2405968A1/en not_active Abandoned
- 2001-05-07 AT AT01940412T patent/ATE441642T1/de not_active IP Right Cessation
- 2001-05-07 US US10/333,388 patent/US7019004B2/en not_active Expired - Fee Related
- 2001-05-07 DE DE60139770T patent/DE60139770D1/de not_active Expired - Fee Related
- 2001-05-07 EP EP01940412A patent/EP1282617B1/en not_active Expired - Lifetime
- 2001-05-07 AU AU73998/01A patent/AU7399801A/en not_active Abandoned
- 2001-05-07 JP JP2001582319A patent/JP2003532724A/ja active Pending
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EP4148050B1 (en) | Novel acid secretion inhibitor and use thereof | |
| JPWO2003037881A1 (ja) | 酢酸アニリド誘導体のα型又はβ型結晶 | |
| CN112898345A (zh) | 核苷酸类似物 | |
| CA2511479A1 (en) | Histone deacetylase inhibitors of novel benzamide derivatives with potent differentiation and anti-proliferation activity | |
| CA2694567A1 (en) | Pharmaceutical composition containing optically active compound having thrombopoietin receptor agonist activity and intermediate thereof | |
| JP2003532724A5 (https=) | ||
| KR20110013411A (ko) | (ｆ-19)-표지된 ｌ-글루탐산 및 ｌ-글루타민 유도체 (ⅲ), 그의 용도 및 그의 수득 방법 | |
| TWI432423B (zh) | ３－二取代吲哚－２－酮衍生物，其製備及其治療用途 | |
| JP2010512355A (ja) | 癌の処置のためのジフェニルオキシ−インドール−２−オン化合物のプロドラッグ | |
| JP4393376B2 (ja) | フェニルシクロヘキシルプロパノールアミン誘導体、その製造法、およびその治療的適用 | |
| EP1282617B1 (en) | Hydantoin derivatives with affinity for somatostatin receptors | |
| TW448176B (en) | Phenylcyclohexylcarboxamides, their preparation and pharmaceutical composition containing the same | |
| US6919379B2 (en) | Compounds useful in reflux disease | |
| WO2000009115A1 (en) | Grp receptor ligands | |
| JP4567889B2 (ja) | （（アミノイミノメチル）アミノ）アルカンカルボキシアミドおよび治療におけるその適用 | |
| JP4927566B2 (ja) | Ｐａｒ−２アゴニスト | |
| US20070004777A1 (en) | Methods for treating or preventing acute myelogenous leukemia | |
| HUP0204476A2 (en) | Therapeutically useful new salts of cck inhibitors, process for the preparation thereof and pharmaceutical compositions containing them | |
| WO2006035936A1 (ja) | Ｐａｒ－２アンタゴニスト | |
| CN111094259A (zh) | 止痛化合物 | |
| JPH06506451A (ja) | Ｇｅｍ−ジホスホン酸ニトロソカルバモイル誘導体、その製造方法およびそれを含む医薬組成物 | |
| JP2001181251A (ja) | アスピリン誘導体、その製造方法、並びにこれを有効成分として含有する抗炎症剤 | |
| RU2263669C2 (ru) | Замещенные 8,8a-дигидро-3ah-индено [1,2-d] тиазолы, способ их получения и их применение в качестве лекарственных средств | |
| JPS5857349A (ja) | ジペプチド誘導体 | |
| EP0270292A2 (en) | Radiation sensitizers |