JP2003530433A5 - - Google Patents

Download PDF

Info

Publication number
JP2003530433A5
JP2003530433A5 JP2001576013A JP2001576013A JP2003530433A5 JP 2003530433 A5 JP2003530433 A5 JP 2003530433A5 JP 2001576013 A JP2001576013 A JP 2001576013A JP 2001576013 A JP2001576013 A JP 2001576013A JP 2003530433 A5 JP2003530433 A5 JP 2003530433A5
Authority
JP
Japan
Prior art keywords
alkoxy
sulfamyl
amino
acetoxy
phosphonate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2001576013A
Other languages
English (en)
Japanese (ja)
Other versions
JP2003530433A (ja
JP4677162B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2001/012134 external-priority patent/WO2001078712A1/en
Publication of JP2003530433A publication Critical patent/JP2003530433A/ja
Publication of JP2003530433A5 publication Critical patent/JP2003530433A5/ja
Application granted granted Critical
Publication of JP4677162B2 publication Critical patent/JP4677162B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

JP2001576013A 2000-04-14 2001-04-13 増殖性障害を治療するための置換スチリルベンジルスルホン Expired - Lifetime JP4677162B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US19784900P 2000-04-14 2000-04-14
US60/197,849 2000-04-14
US23470700P 2000-09-22 2000-09-22
US60/234,707 2000-09-22
US27164001P 2001-02-27 2001-02-27
US60/271,640 2001-02-27
PCT/US2001/012134 WO2001078712A1 (en) 2000-04-14 2001-04-13 Substituted styryl benzylsulfones for treating proliferative disorders

Publications (3)

Publication Number Publication Date
JP2003530433A JP2003530433A (ja) 2003-10-14
JP2003530433A5 true JP2003530433A5 (enExample) 2008-05-29
JP4677162B2 JP4677162B2 (ja) 2011-04-27

Family

ID=27393791

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001576013A Expired - Lifetime JP4677162B2 (ja) 2000-04-14 2001-04-13 増殖性障害を治療するための置換スチリルベンジルスルホン

Country Status (13)

Country Link
US (2) US6486210B2 (enExample)
EP (2) EP1305015B1 (enExample)
JP (1) JP4677162B2 (enExample)
KR (1) KR100768415B1 (enExample)
AU (2) AU2001251615C1 (enExample)
CA (1) CA2406212C (enExample)
DK (1) DK1305015T3 (enExample)
ES (1) ES2427088T3 (enExample)
IL (2) IL152190A0 (enExample)
NZ (1) NZ522551A (enExample)
PT (1) PT1305015E (enExample)
SI (1) SI1305015T1 (enExample)
WO (1) WO2001078712A1 (enExample)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6762207B1 (en) * 1999-04-02 2004-07-13 Temple University - Of The Commonwealth System Of Higher Education (E)-styryl sulfone anticancer agents
CA2424884C (en) 2000-10-05 2009-12-15 E. Premkumar Reddy Substituted (e)-styryl benzylsulfones for treating proliferative disorders
US6833480B2 (en) * 2001-02-27 2004-12-21 Temple University - Of The Commonwealth System Of Higher Education (Z)-styrylbenzylsulfones and pharmaceutical uses thereof
ATE406881T1 (de) 2001-02-28 2008-09-15 Univ Temple Verwendung von alpha, beta ungesättigten arylsulfonen zum schutz von zellen und geweben vor toxizität ionischer strahlung
MXPA04008356A (es) * 2002-02-28 2005-09-12 Univ Temple (e)-2,6-dialcoxiestiril bencilsulfonas sustituidas con un grupo amino y en la posicion 4 para tratar trastornos poliferativos.
ATE517626T1 (de) * 2002-02-28 2011-08-15 Univ Temple Aminosubstituierte sulphonanilide und ihre derivate zur behandlung von proliferativen erkrankungen
JP4182844B2 (ja) * 2003-09-03 2008-11-19 株式会社島津製作所 質量分析装置
HUE032523T2 (en) * 2003-11-14 2017-09-28 Temple Univ - Of The Commonwealth System Of Higher Education Alpha, beta-unsaturated sulfoxides for the treatment of proliferative disorders
ES2609084T3 (es) * 2004-03-16 2017-04-18 Temple University - Of The Commonwealth System Of Higher Education Derivados de fenoxi y feniltio sustituidos para tratar trastornos proliferativos
CA2577309C (en) 2004-06-24 2013-10-22 Temple University - Of The Commonwealth System Of Higher Education Alpha, beta-unsaturated sulfones, sulfoxides, sulfonimides, sulfinimides, acylsulfonamides and acylsulfinamides and therapeutic uses thereof
AU2006204103B2 (en) * 2005-01-05 2011-11-24 Temple University Of The Commonwealth System Of Higher Education Treatment of drug-resistant proliferative disorders
PT1896401E (pt) * 2005-02-25 2013-07-17 Univ Temple Síntese de sulfuretos, sulfonas, sulfóxidos e sulfonamidas não saturados
WO2006104668A2 (en) * 2005-03-11 2006-10-05 Temple University - Of The Commonwealth System Of Higher Education Composition and methods for the treatment of proliferative diseases
JP5278968B2 (ja) * 2006-08-30 2013-09-04 テンプル・ユニバーシティ−オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション 骨髄異形性症候群及び急性骨髄性白血病の治療のための組成物及び方法
US8273787B2 (en) * 2006-09-15 2012-09-25 Onconova Therapeutics, Inc Activated cytotoxic compounds for attachment to targeting molecules for the treatment of mammalian disease conditions
US8735620B2 (en) * 2008-12-17 2014-05-27 Epr Pharmaceuticals Pvt. Ltd Processes for preparing (E)-styrylbenzylsulfone compounds and uses thereof for treating proliferative disorders
US10207989B2 (en) 2012-09-20 2019-02-19 Temple University—Of the Commonwealth System of Higher Education Substituted alkyl diaryl derivatives, methods of preparation and uses
WO2014089483A1 (en) 2012-12-07 2014-06-12 Onconova Therapeutics, Inc. Methods and compositions for treatment of cancer
US10383831B2 (en) 2015-08-03 2019-08-20 Temple University—Of the Commonwealth System of Higher Education 2,4,6-trialkoxystryl aryl sulfones, sulfonamides and carboxamides, and methods of preparation and use
WO2024186641A1 (en) * 2023-03-03 2024-09-12 Onconova Therapeutics, Inc. Methods and compositions for treating cancer

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2532612A (en) 1945-08-29 1950-12-05 Union Oil Co Preparation of unsaturated thio-ethers
US3185743A (en) 1960-08-24 1965-05-25 Union Carbide Corp Production of olefinic compounds from allyl sulfones
US3418101A (en) 1965-12-15 1968-12-24 Pennsalt Chemicals Corp Process for plant desiccation
US3514386A (en) 1967-12-11 1970-05-26 Exxon Research Engineering Co Stereoselective addition of thiols to acetylenic compounds
US3917714A (en) 1972-09-06 1975-11-04 American Cyanamid Co Bis(alkylsulfonyl)vinylbenzenes
US4161407A (en) 1977-10-06 1979-07-17 Eastman Kodak Company Crosslinkable polymers having vinylsulfonyl groups or styrylsulfonyl groups and their use as hardeners for gelatin
US4386221A (en) 1981-10-28 1983-05-31 Eastman Kodak Company Process for the preparation of aryl alkyl sulfones and aryl vinyl sulfones
US4937388A (en) 1985-08-09 1990-06-26 Imperial Chemical Industries Plc Insecticidal ethers
YU213587A (en) * 1986-11-28 1989-06-30 Orion Yhtymae Oy Process for obtaining new pharmacologic active cateholic derivatives
FR2621038B1 (fr) * 1987-09-28 1989-12-29 Rhone Poulenc Sante Derives d'alcadienes, leurs preparations, les medicaments les contenant et produits intermediaires
GB8902409D0 (en) * 1989-02-03 1989-03-22 Ici Plc Aliphatic compounds
US5659087A (en) 1995-06-07 1997-08-19 Eli Lilly And Company Diarylvinyl sulfoxides
JP3660395B2 (ja) * 1995-06-22 2005-06-15 大鵬薬品工業株式会社 フェニルスルホン誘導体及びその製造方法
CZ290756B6 (cs) * 1995-10-19 2002-10-16 Ciba Specialty Chemicals Holding Inc. Substituované fenoly působící jako antioxidanty, kompozice, které je obsahují, a jejich pouľití
ATE284386T1 (de) 1997-10-03 2004-12-15 Univ Temple Styrolsulfone als antikrebsmittel
US6201154B1 (en) * 1999-03-31 2001-03-13 Temple University-Of The Commonwealth Of Higher Education Z-styryl sulfone anticancer agents
JP2002541101A (ja) * 1999-04-02 2002-12-03 テンプル・ユニバーシティ−オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイション スチリルスルホン抗癌剤
CA2366750C (en) * 1999-04-02 2010-06-01 Temple University - Of The Commonwealth System Of Higher Education (e)-styryl sulfone anticancer agents
AU780844B2 (en) * 1999-10-12 2005-04-21 Temple University-Of The Commonwealth System Of Higher Education Method for protecting normal cells from cytotoxicity of chemotherapeutic agents

Similar Documents

Publication Publication Date Title
JP2003530433A5 (enExample)
JP2002332234A5 (enExample)
JP2019512478A5 (enExample)
JP2004505047A5 (enExample)
JP2005511697A5 (enExample)
JP2001247459A5 (enExample)
CA2406212A1 (en) Substituted styryl benzylsulfones for treating proliferative disorders
JP2005528325A5 (enExample)
JP2005525323A5 (enExample)
JP2004537516A5 (enExample)
JP2006502283A5 (enExample)
JP2002531498A5 (enExample)
JP2002540152A5 (enExample)
JP2003522198A5 (enExample)
JP2003532640A5 (enExample)
JP2004503564A5 (enExample)
JP2004531612A5 (enExample)
JP2005530779A5 (enExample)
JP2002505323A5 (enExample)
JP2012513390A5 (enExample)
JP2001515881A5 (enExample)
JP2003502367A5 (enExample)
JP2008520662A5 (enExample)
JP2001097975A5 (enExample)
JP2005504696A5 (enExample)