JP2003513090A5 - - Google Patents

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Publication number
JP2003513090A5
JP2003513090A5 JP2001534803A JP2001534803A JP2003513090A5 JP 2003513090 A5 JP2003513090 A5 JP 2003513090A5 JP 2001534803 A JP2001534803 A JP 2001534803A JP 2001534803 A JP2001534803 A JP 2001534803A JP 2003513090 A5 JP2003513090 A5 JP 2003513090A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2001534803A
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Japanese (ja)
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JP3787307B2 (ja
JP2003513090A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2000/010524 external-priority patent/WO2001032652A2/en
Publication of JP2003513090A publication Critical patent/JP2003513090A/ja
Publication of JP2003513090A5 publication Critical patent/JP2003513090A5/ja
Application granted granted Critical
Publication of JP3787307B2 publication Critical patent/JP3787307B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2001534803A 1999-11-02 2000-10-25 N置換カルバモイルオキシアルキルアゾリウム誘導体 Expired - Lifetime JP3787307B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP99121694 1999-11-02
EP99121694.6 1999-11-02
PCT/EP2000/010524 WO2001032652A2 (en) 1999-11-02 2000-10-25 N-substituted carbamoyloxyalkyl-azolium derivatives

Publications (3)

Publication Number Publication Date
JP2003513090A JP2003513090A (ja) 2003-04-08
JP2003513090A5 true JP2003513090A5 (https=) 2005-12-22
JP3787307B2 JP3787307B2 (ja) 2006-06-21

Family

ID=8239312

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001534803A Expired - Lifetime JP3787307B2 (ja) 1999-11-02 2000-10-25 N置換カルバモイルオキシアルキルアゾリウム誘導体

Country Status (22)

Country Link
EP (1) EP1280795B1 (https=)
JP (1) JP3787307B2 (https=)
KR (1) KR100449797B1 (https=)
CN (1) CN1185230C (https=)
AR (1) AR029403A1 (https=)
AT (1) ATE291575T1 (https=)
AU (1) AU777859B2 (https=)
BE (1) BE2016C007I2 (https=)
BR (1) BRPI0015254C1 (https=)
CA (2) CA2680292C (https=)
CY (1) CY2016002I2 (https=)
DE (1) DE60018989T2 (https=)
DK (1) DK1280795T3 (https=)
ES (1) ES2238341T3 (https=)
FR (1) FR15C0096I2 (https=)
LU (1) LU92939I2 (https=)
MX (1) MXPA02004145A (https=)
NL (1) NL300791I2 (https=)
PT (1) PT1280795E (https=)
TR (1) TR200201205T2 (https=)
WO (1) WO2001032652A2 (https=)
ZA (1) ZA200203003B (https=)

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MY148805A (en) 2002-10-16 2013-05-31 Takeda Pharmaceutical Controlled release preparation
JP5576279B2 (ja) 2007-08-21 2014-08-20 バジリア ファルマスーチカ アーゲー 抗真菌組成物
CN103857440B (zh) 2011-06-22 2018-09-25 维奥姆生物科学有限公司 基于缀合物的抗真菌和抗细菌前药
US20160128944A1 (en) 2013-06-04 2016-05-12 Vyome Biosciences Pvt. Ltd. Coated particles and compositions comprising same
CN104230894B (zh) * 2013-06-06 2016-08-24 南京华威医药科技开发有限公司 三唑类化合物
US20170290333A1 (en) 2014-12-30 2017-10-12 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
CN106032356B (zh) * 2015-03-13 2018-09-14 江苏正大丰海制药有限公司 一种[n-甲基-吡啶-2-基]氨基甲酸-1-氯乙酯的制备方法
CN104974143A (zh) * 2015-05-12 2015-10-14 深圳致君制药有限公司 一种季铵盐类化合物、其制备方法以及用途
CN106467534B (zh) * 2015-08-17 2019-10-11 江苏奥赛康药业有限公司 一种硫酸艾沙康唑鎓化合物及其药物组合物
CN106467519B (zh) * 2015-08-17 2019-08-13 南京华威医药科技集团有限公司 一种水溶性三唑化合物
CN106565699B (zh) * 2015-10-10 2019-07-26 江苏正大丰海制药有限公司 一种艾沙康唑硫酸盐晶体及其制备方法
US10683387B2 (en) 2016-10-04 2020-06-16 Massachusetts Institute Of Technology Bottlebrush copolymers and uses thereof
WO2018149359A1 (zh) * 2017-02-17 2018-08-23 武汉朗来科技发展有限公司 三氮唑抗菌衍生物、其药物组合物和用途
CN106916152B (zh) * 2017-04-27 2019-09-17 扬子江药业集团有限公司 氧化还原反应制备艾沙康唑鎓单硫酸盐的方法
WO2019006425A1 (en) 2017-06-30 2019-01-03 Massachusetts Institute Of Technology IMAGING AGENTS OF BRUSH ARRAY STAR POLYMERS AND USES THEREOF
JP7187048B2 (ja) 2017-06-30 2022-12-12 マサチューセッツ インスティテュート オブ テクノロジー 分枝多官能性マクロモノマーおよび関連ポリマーならびにそれらの使用
US10368502B2 (en) 2017-09-25 2019-08-06 Multiple Energy Technologies Llc Bioceramic and carbon-based hydroponic systems, methods and devices
CN110317165A (zh) * 2018-03-28 2019-10-11 上海医药工业研究院 一种药物中间体2-甲胺基-3-吡啶甲醇的制备方法
US12414997B2 (en) 2018-04-13 2025-09-16 Massachusetts Institute Of Technology Brush prodrugs and uses thereof
CN110551064B (zh) * 2018-06-01 2021-01-01 重庆世森医药科技有限公司 艾沙康唑硫酸酯及其中间体的制备方法
AU2019313525A1 (en) 2018-08-01 2021-01-07 Basilea Pharmaceutica International AG Methods for purifying isavuconazonium sulfate
US10988491B2 (en) 2018-08-17 2021-04-27 Massachusetts Institute Of Technology Degradable polymers of a cyclic silyl ether and uses thereof
CN110128420A (zh) * 2019-05-08 2019-08-16 阴启明 硫酸氢根/硫酸根型阴离子交换技术制备艾沙康唑鎓单硫酸盐的方法
EP4021576A1 (en) 2019-08-26 2022-07-06 Synthon B.V. Isavuconazonium salts and process for preparing thereof
EP4045562A2 (en) * 2019-10-16 2022-08-24 Massachusetts Institute of Technology Brush prodrugs and uses thereof
WO2021141662A1 (en) 2020-01-10 2021-07-15 Massachusetts Institute Of Technology Proteolysis targeting chimeric molecules (protacs) with functional handles and uses thereof
JP7570382B2 (ja) 2021-09-28 2024-10-21 旭化成ファーマ株式会社 エアベント付き輸液フィルタを備える点滴静脈投与用輸液セット
JP7454905B2 (ja) * 2021-09-28 2024-03-25 旭化成ファーマ株式会社 有効成分であるイサブコナゾール又はそのプロドラッグを含有する真菌症治療及び/又は予防剤
US12084415B2 (en) 2021-12-20 2024-09-10 Massachusetts Institute Of Technology Biomolecule-polymer-pharmaceutical agent conjugates for delivering the pharmaceutical agent
EP4289840A1 (en) 2022-06-07 2023-12-13 Zaklady Farmaceutyczne Polpharma S.A. A process for preparing isavuconazonium sulfate
WO2024094329A1 (en) 2022-11-01 2024-05-10 Basilea Pharmaceutica International Ag, Allschwil Blister-packaged capsule preparation containing isavuconazonium sulfate
WO2024189550A1 (en) * 2023-03-13 2024-09-19 Apitoria Pharma Private Limited Process for the preparation of isavuconazonium sulfate and its crystalline forms
TW202541814A (zh) 2023-11-30 2025-11-01 瑞士商巴塞利亞阿爾斯維爾藥業國際股份有限公司 用於治療真菌感染的藥物組合

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Publication number Priority date Publication date Assignee Title
JP3108997B2 (ja) * 1997-03-31 2000-11-13 武田薬品工業株式会社 アゾール化合物、その製造法および用途
CN1251098A (zh) * 1997-03-31 2000-04-19 武田药品工业株式会社 吡咯化合物,其制备及其用途
AU2931399A (en) * 1998-03-06 1999-09-20 F. Hoffmann-La Roche Ag 3-(4-(4-cyanophenyl)thiazol-2-y))-1-(1h-1,2,4-triazol-1-yl) -butan-2-ol derivatives having antifungal activity

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