JP2003342259A - 光学活性シスピペリジン誘導体の製造法 - Google Patents

光学活性シスピペリジン誘導体の製造法

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Publication number
JP2003342259A
JP2003342259A JP2002369405A JP2002369405A JP2003342259A JP 2003342259 A JP2003342259 A JP 2003342259A JP 2002369405 A JP2002369405 A JP 2002369405A JP 2002369405 A JP2002369405 A JP 2002369405A JP 2003342259 A JP2003342259 A JP 2003342259A
Authority
JP
Japan
Prior art keywords
optically active
group
derivative
cispiperidine
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002369405A
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English (en)
Japanese (ja)
Other versions
JP2003342259A5 (https=
Inventor
Toshihiro Fujino
年弘 藤野
Seiji Morii
清二 森井
Haruyo Sato
治代 佐藤
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Toray Industries Inc
Original Assignee
Toray Industries Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Toray Industries Inc filed Critical Toray Industries Inc
Priority to JP2002369405A priority Critical patent/JP2003342259A/ja
Publication of JP2003342259A publication Critical patent/JP2003342259A/ja
Publication of JP2003342259A5 publication Critical patent/JP2003342259A5/ja
Pending legal-status Critical Current

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  • Hydrogenated Pyridines (AREA)
JP2002369405A 2001-12-21 2002-12-20 光学活性シスピペリジン誘導体の製造法 Pending JP2003342259A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2002369405A JP2003342259A (ja) 2001-12-21 2002-12-20 光学活性シスピペリジン誘導体の製造法

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2001-388633 2001-12-21
JP2001388633 2001-12-21
JP2002074160 2002-03-18
JP2002-74160 2002-03-18
JP2002369405A JP2003342259A (ja) 2001-12-21 2002-12-20 光学活性シスピペリジン誘導体の製造法

Publications (2)

Publication Number Publication Date
JP2003342259A true JP2003342259A (ja) 2003-12-03
JP2003342259A5 JP2003342259A5 (https=) 2005-04-07

Family

ID=29783080

Family Applications (1)

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JP2002369405A Pending JP2003342259A (ja) 2001-12-21 2002-12-20 光学活性シスピペリジン誘導体の製造法

Country Status (1)

Country Link
JP (1) JP2003342259A (https=)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012211174A (ja) * 2004-11-05 2012-11-01 Boehringer Ingelheim Internatl Gmbh キラル８−（３−アミノ−ピペリジン−１−イル）−キサンチンの製造方法
JP2021515029A (ja) * 2017-12-22 2021-06-17 ジークフリート アクチェンゲゼルシャフトＳｉｅｇｆｒｉｅｄ Ａｇ Ｏ，ｏ’−二置換酒石酸エナンチオマーの添加によるラセミ体ニコチンのエナンチオマー分離
US11407730B2 (en) 2017-12-22 2022-08-09 Siegfried Ag Preparation of racemic nicotine by reaction of ethyl nicotinate with N-vinylpyrrolidone in the presence of an alcoholate base and subsequent process steps

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012211174A (ja) * 2004-11-05 2012-11-01 Boehringer Ingelheim Internatl Gmbh キラル８−（３−アミノ−ピペリジン−１−イル）−キサンチンの製造方法
JP2021515029A (ja) * 2017-12-22 2021-06-17 ジークフリート アクチェンゲゼルシャフトＳｉｅｇｆｒｉｅｄ Ａｇ Ｏ，ｏ’−二置換酒石酸エナンチオマーの添加によるラセミ体ニコチンのエナンチオマー分離
JP7030208B2 (ja) 2017-12-22 2022-03-04 ジークフリート アクチェンゲゼルシャフト Ｏ，ｏ’－二置換酒石酸エナンチオマーの添加によるラセミ体ニコチンのエナンチオマー分離
US11279685B2 (en) 2017-12-22 2022-03-22 Siegfried Ag Enantiomeric separation of racemic nicotine by addition of an O,O″-disubstituted tartaric acid enantiomer
US11407730B2 (en) 2017-12-22 2022-08-09 Siegfried Ag Preparation of racemic nicotine by reaction of ethyl nicotinate with N-vinylpyrrolidone in the presence of an alcoholate base and subsequent process steps

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