JP2002506880A - テトラペプチドの製法 - Google Patents

テトラペプチドの製法

Info

Publication number
JP2002506880A
JP2002506880A JP2000536740A JP2000536740A JP2002506880A JP 2002506880 A JP2002506880 A JP 2002506880A JP 2000536740 A JP2000536740 A JP 2000536740A JP 2000536740 A JP2000536740 A JP 2000536740A JP 2002506880 A JP2002506880 A JP 2002506880A
Authority
JP
Japan
Prior art keywords
derivative
ester
phe
protected
solvent
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2000536740A
Other languages
English (en)
Japanese (ja)
Inventor
ヘンリ・フラーンセン
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
Original Assignee
AstraZeneca AB
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AstraZeneca AB filed Critical AstraZeneca AB
Publication of JP2002506880A publication Critical patent/JP2002506880A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1027—Tetrapeptides containing heteroatoms different from O, S, or N

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2000536740A 1998-03-16 1999-03-16 テトラペプチドの製法 Pending JP2002506880A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9800865-9 1998-03-16
SE9800865A SE9800865D0 (sv) 1998-03-16 1998-03-16 New Process
PCT/SE1999/000414 WO1999047548A1 (en) 1998-03-16 1999-03-16 Process for the preparation of a tetrapeptide

Publications (1)

Publication Number Publication Date
JP2002506880A true JP2002506880A (ja) 2002-03-05

Family

ID=20410566

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000536740A Pending JP2002506880A (ja) 1998-03-16 1999-03-16 テトラペプチドの製法

Country Status (19)

Country Link
EP (1) EP1062231A1 (is)
JP (1) JP2002506880A (is)
KR (1) KR20010041888A (is)
CN (1) CN1300293A (is)
AU (1) AU2968899A (is)
BR (1) BR9908765A (is)
CA (1) CA2323678A1 (is)
EE (1) EE200000540A (is)
HU (1) HUP0102877A3 (is)
ID (1) ID26938A (is)
IL (1) IL138244A0 (is)
IS (1) IS5612A (is)
NO (1) NO20004613L (is)
PL (1) PL343277A1 (is)
SE (1) SE9800865D0 (is)
SK (1) SK13442000A3 (is)
TR (1) TR200002652T2 (is)
WO (1) WO1999047548A1 (is)
ZA (1) ZA200004376B (is)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011508727A (ja) * 2007-12-13 2011-03-17 サイトジェル ファーマ リミテッド ライアビリティ カンパニー μ−オピエート受容体ペプチドの有利な塩

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9903291D0 (sv) * 1999-09-15 1999-09-15 Astra Ab New process
CN104371002B (zh) * 2013-06-20 2017-10-10 重庆理工大学 一种非蛋白氨基酸抗菌肽及其应用
CN104478993B (zh) * 2013-06-20 2017-10-10 重庆理工大学 一种非蛋白氨基酸抗菌肽及其应用
CN103319568B (zh) * 2013-06-20 2015-01-21 重庆理工大学 一种非蛋白氨基酸抗菌肽及其应用
CN104783298A (zh) * 2015-03-24 2015-07-22 湖州珍贝羊绒制品有限公司 一种生物灭菌组合物及其纳米乳的制备与应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9503924D0 (sv) * 1995-08-18 1995-11-07 Astra Ab Novel opioid peptides
GB9516994D0 (en) * 1995-08-18 1995-10-18 Iaf Biochem Int Solution synthesis of peripheral acting analgestic opioid tetrapeptides

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011508727A (ja) * 2007-12-13 2011-03-17 サイトジェル ファーマ リミテッド ライアビリティ カンパニー μ−オピエート受容体ペプチドの有利な塩

Also Published As

Publication number Publication date
NO20004613L (no) 2000-10-30
NO20004613D0 (no) 2000-09-15
HUP0102877A3 (en) 2002-02-28
IL138244A0 (en) 2001-10-31
TR200002652T2 (tr) 2000-11-21
PL343277A1 (en) 2001-08-13
KR20010041888A (ko) 2001-05-25
HUP0102877A2 (hu) 2002-01-28
WO1999047548A1 (en) 1999-09-23
BR9908765A (pt) 2000-11-07
IS5612A (is) 2000-08-30
CA2323678A1 (en) 1999-09-23
SK13442000A3 (sk) 2001-04-09
ID26938A (id) 2001-02-22
SE9800865D0 (sv) 1998-03-16
CN1300293A (zh) 2001-06-20
ZA200004376B (en) 2001-10-31
EE200000540A (et) 2002-02-15
AU2968899A (en) 1999-10-11
EP1062231A1 (en) 2000-12-27

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