IT1196751B - Alogeno e ciano derivati dell'acido glutammico ed aspartico ad attivita antagonista su polipeptidi bioattivi e procedimento per la loro preparazione - Google Patents
Alogeno e ciano derivati dell'acido glutammico ed aspartico ad attivita antagonista su polipeptidi bioattivi e procedimento per la loro preparazioneInfo
- Publication number
- IT1196751B IT1196751B IT68070/84A IT6807084A IT1196751B IT 1196751 B IT1196751 B IT 1196751B IT 68070/84 A IT68070/84 A IT 68070/84A IT 6807084 A IT6807084 A IT 6807084A IT 1196751 B IT1196751 B IT 1196751B
- Authority
- IT
- Italy
- Prior art keywords
- new
- aspartic acid
- acid amide
- acyl glutamic
- alkyl
- Prior art date
Links
- WHUUTDBJXJRKMK-UHFFFAOYSA-N Glutamic acid Natural products OC(=O)C(N)CCC(O)=O WHUUTDBJXJRKMK-UHFFFAOYSA-N 0.000 title 1
- PMLJIHNCYNOQEQ-REOHCLBHSA-N L-aspartic 1-amide Chemical compound NC(=O)[C@@H](N)CC(O)=O PMLJIHNCYNOQEQ-REOHCLBHSA-N 0.000 title 1
- 235000013922 glutamic acid Nutrition 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- -1 morpholino, piperidino Chemical group 0.000 abstract 2
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 2
- 125000004189 3,4-dichlorophenyl group Chemical group [H]C1=C([H])C(Cl)=C(Cl)C([H])=C1* 0.000 abstract 1
- 125000004801 4-cyanophenyl group Chemical group [H]C1=C([H])C(C#N)=C([H])C([H])=C1* 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (17)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT68070/84A IT1196751B (it) | 1984-10-26 | 1984-10-26 | Alogeno e ciano derivati dell'acido glutammico ed aspartico ad attivita antagonista su polipeptidi bioattivi e procedimento per la loro preparazione |
| IE1502/85A IE57892B1 (en) | 1984-06-25 | 1985-06-17 | Glutamic and aspartic acid derivatives |
| NZ212436A NZ212436A (en) | 1984-06-25 | 1985-06-17 | D,l-glutamic and d,l-aspartic acid derivatives and pharmaceutical compositions |
| CA000484341A CA1325633C (en) | 1984-06-25 | 1985-06-18 | Derivatives of glutamic acid and aspartic acid having antagonistic activities towards bioactive polypeptides and method for their preparation |
| US06/746,065 US4791215A (en) | 1984-06-25 | 1985-06-18 | Derivatives of glutamic acid and aspartic acid |
| GB08515555A GB2160869B (en) | 1984-06-25 | 1985-06-19 | Glutamic and aspartic acid derivatives |
| FR8509383A FR2566397B1 (fr) | 1984-06-25 | 1985-06-20 | Derives de l'acide glutamique et de l'acide aspartique ayant des activites antagonistes vis-a-vis de polypeptides bioactifs et procede pour leur preparation |
| SE8503097A SE503111C2 (sv) | 1984-06-25 | 1985-06-20 | Farmaceutiskt aktiva derivat av D,L-glutaminsyra och D,L- asparaginsyra samt förfarande för dess framställning |
| CH2617/85A CH674203A5 (it) | 1984-06-25 | 1985-06-20 | |
| BE0/215244A BE902726A (fr) | 1984-06-25 | 1985-06-21 | Derives de l'acide glutamique et de l'acide aspartique ayant des activites antagonistes vis-a-vis de polypeptides bioactifs. |
| ES544462A ES8604859A1 (es) | 1984-06-25 | 1985-06-22 | Metodo para la preparacion de derivados de acido glutamico yacido aspartico |
| AU44109/85A AU566601B2 (en) | 1984-06-25 | 1985-06-24 | Derivatives of glutamic and aspartic acids |
| DE19853522506 DE3522506A1 (de) | 1984-06-25 | 1985-06-24 | Derivate von glutaminsaeure und asparaginsaeure mit antagonistischer wirkung gegen bioaktive polypeptide und verfahren zu ihrer herstellung |
| PT8069285A PT80692B (pt) | 1984-06-25 | 1985-06-24 | Processo para a preparacao de derivados de acido glutamico e de acido aspartico possuindo actividades antagonisticas em relacao a polipeptidos bioactivos |
| DK285685A DK285685A (da) | 1984-06-25 | 1985-06-24 | Farmaceutisk aktive derivater af d,l-glutaminsyre og d,l-asparaginsyre og farmaceutisk acceptable salte deraf, deres fremstilling og anvendelse |
| AT0186985A AT390949B (de) | 1984-06-25 | 1985-06-24 | Verfahren zur herstellung von neuen glutaminsaeure- und asparaginsaeurederivaten und ihren salzen |
| NL8501829A NL8501829A (nl) | 1984-06-25 | 1985-06-25 | Glutaminezuur- respectievelijk asparaginezuurderivaten, werkwijze voor de bereiding ervan alsmede de toepassing ervan in preparaten. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT68070/84A IT1196751B (it) | 1984-10-26 | 1984-10-26 | Alogeno e ciano derivati dell'acido glutammico ed aspartico ad attivita antagonista su polipeptidi bioattivi e procedimento per la loro preparazione |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT8468070A0 IT8468070A0 (it) | 1984-10-26 |
| IT1196751B true IT1196751B (it) | 1988-11-25 |
Family
ID=11307627
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT68070/84A IT1196751B (it) | 1984-06-25 | 1984-10-26 | Alogeno e ciano derivati dell'acido glutammico ed aspartico ad attivita antagonista su polipeptidi bioattivi e procedimento per la loro preparazione |
Country Status (1)
| Country | Link |
|---|---|
| IT (1) | IT1196751B (it) |
-
1984
- 1984-10-26 IT IT68070/84A patent/IT1196751B/it active
Also Published As
| Publication number | Publication date |
|---|---|
| IT8468070A0 (it) | 1984-10-26 |
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