IT1156791B - Derivati di acidi tiazolidincarbos silici utili in particolare come inibitori enzimatici - Google Patents
Derivati di acidi tiazolidincarbos silici utili in particolare come inibitori enzimaticiInfo
- Publication number
- IT1156791B IT1156791B IT49660/78A IT4966078A IT1156791B IT 1156791 B IT1156791 B IT 1156791B IT 49660/78 A IT49660/78 A IT 49660/78A IT 4966078 A IT4966078 A IT 4966078A IT 1156791 B IT1156791 B IT 1156791B
- Authority
- IT
- Italy
- Prior art keywords
- thiazolidincarbos
- derivatives
- useful
- enzymatic inhibitors
- silic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D277/06—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
- C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/907,452 US4192878A (en) | 1976-12-03 | 1978-05-22 | Derivatives of thiazolidinecarboxylic acids and related acids |
Publications (2)
Publication Number | Publication Date |
---|---|
IT7849660A0 IT7849660A0 (it) | 1978-06-01 |
IT1156791B true IT1156791B (it) | 1987-02-04 |
Family
ID=25424116
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT49660/78A IT1156791B (it) | 1978-05-22 | 1978-06-01 | Derivati di acidi tiazolidincarbos silici utili in particolare come inibitori enzimatici |
Country Status (18)
Country | Link |
---|---|
JP (1) | JPS54151965A (ru) |
AU (1) | AU521516B2 (ru) |
BE (1) | BE867776R (ru) |
CA (1) | CA1102812A (ru) |
CH (1) | CH633782A5 (ru) |
DE (1) | DE2823352A1 (ru) |
DK (1) | DK242378A (ru) |
FR (1) | FR2426685A2 (ru) |
HU (1) | HU179780B (ru) |
IE (1) | IE47075B1 (ru) |
IT (1) | IT1156791B (ru) |
NZ (1) | NZ187390A (ru) |
PH (1) | PH14405A (ru) |
PL (1) | PL207332A3 (ru) |
SE (1) | SE7806468L (ru) |
SU (2) | SU730303A3 (ru) |
YU (1) | YU131478A (ru) |
ZA (1) | ZA783013B (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4347371A (en) * | 1978-12-30 | 1982-08-31 | Santen Pharmaceutical Co., Ltd. | Disulfide compounds |
US4692458A (en) * | 1980-03-05 | 1987-09-08 | University Of Miami | Anti-hypertensive agents |
RU2526619C2 (ru) * | 2012-12-12 | 2014-08-27 | Федеральное государственное бюджетное учреждение науки Институт высокомолекулярных соединений Российской академии наук | Способ получения (2r,4r)-2-алкил-3-(2-меркаптобензоил)-1,3-тиазолидин-4-карбоновых кислот |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2404635A1 (fr) * | 1977-09-28 | 1979-04-27 | Science Union & Cie | Nouveaux thioproprionylamides, leurs procedures d'obtention et leur emploi en therapeutique |
-
1978
- 1978-05-25 CA CA304,036A patent/CA1102812A/en not_active Expired
- 1978-05-25 ZA ZA00783013A patent/ZA783013B/xx unknown
- 1978-05-26 NZ NZ187390A patent/NZ187390A/xx unknown
- 1978-05-29 AU AU36602/78A patent/AU521516B2/en not_active Expired
- 1978-05-29 DE DE19782823352 patent/DE2823352A1/de not_active Withdrawn
- 1978-05-31 IE IE1098/78A patent/IE47075B1/en unknown
- 1978-05-31 CH CH596978A patent/CH633782A5/fr not_active IP Right Cessation
- 1978-05-31 DK DK242378A patent/DK242378A/da not_active Application Discontinuation
- 1978-06-01 FR FR7816377A patent/FR2426685A2/fr active Granted
- 1978-06-01 YU YU01314/78A patent/YU131478A/xx unknown
- 1978-06-01 IT IT49660/78A patent/IT1156791B/it active
- 1978-06-01 SE SE7806468A patent/SE7806468L/xx not_active Application Discontinuation
- 1978-06-02 PH PH21226A patent/PH14405A/en unknown
- 1978-06-02 JP JP6715778A patent/JPS54151965A/ja active Pending
- 1978-06-02 HU HU78SU976A patent/HU179780B/hu not_active IP Right Cessation
- 1978-06-02 SU SU782624853A patent/SU730303A3/ru active
- 1978-06-02 BE BE188292A patent/BE867776R/xx not_active IP Right Cessation
- 1978-06-02 PL PL20733278A patent/PL207332A3/xx unknown
-
1979
- 1979-04-13 SU SU792749103A patent/SU816400A3/ru active
Also Published As
Publication number | Publication date |
---|---|
CH633782A5 (en) | 1982-12-31 |
PL207332A3 (ru) | 1980-01-28 |
ZA783013B (en) | 1979-06-27 |
PH14405A (en) | 1981-06-25 |
BE867776R (fr) | 1978-12-04 |
HU179780B (en) | 1982-12-28 |
DE2823352A1 (de) | 1979-11-29 |
SU730303A3 (ru) | 1980-04-25 |
IE781098L (en) | 1979-11-22 |
NZ187390A (en) | 1980-05-27 |
DK242378A (da) | 1979-11-23 |
FR2426685A2 (fr) | 1979-12-21 |
IT7849660A0 (it) | 1978-06-01 |
FR2426685B2 (ru) | 1981-09-04 |
AU3660278A (en) | 1979-12-06 |
CA1102812A (en) | 1981-06-09 |
JPS54151965A (en) | 1979-11-29 |
AU521516B2 (en) | 1982-04-08 |
SU816400A3 (ru) | 1981-03-23 |
YU131478A (en) | 1984-06-30 |
IE47075B1 (en) | 1983-12-14 |
SE7806468L (sv) | 1979-11-23 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IT1120977B (it) | Derivati di acidi fenossialchilcar bossilici particolarmente utili come medicamenti | |
IT1149259B (it) | Derivati di acidi 6 beta-idrossialchilpenicillanici come inibitori della beta-lattamasi | |
IT1058202B (it) | Composizioni di cianoacrilato utili in particolare come adesivi | |
BG33296A3 (en) | Method for obtaining the derivatives of 4- dezacetyl- vincalevcoblastine c- 3- carboxyhydrazid | |
DE3162660D1 (de) | Amides of 4-oxo-5-amidohexanoic acid derivatives | |
IT1121786B (it) | Composizione e metodo per inibire la formazione di incroststazioni | |
IT1162481B (it) | Acidi 4-(5-fluorometil-2-piridil-ossi)-fenossi-valerici e loro derivti composizioni erbicide che li contengono e procedimento per applicarli | |
IT1173663B (it) | Derivati di acidi fenossialchilcabossilici | |
IT1121045B (it) | Derivati di acidi imminocarbossilici ciclici | |
IT1156791B (it) | Derivati di acidi tiazolidincarbos silici utili in particolare come inibitori enzimatici | |
IT1130301B (it) | Acidi penicillanici 6-beta-sostituiti come inibitori della-beta-lattamasi | |
IT1122180B (it) | Derivati di 1-fenil-1-propanolo | |
IT1228934B (it) | Derivati dell'acido 7-ossabiciclo (2.2.1.) eptan idrossammico utili come inibitori duplici | |
IT1118846B (it) | Derivati di acidi idrossammici | |
IT1085699B (it) | Processo di idrofugazione di manufatti in gesso | |
IT1126510B (it) | Derivati mercaptoacilici di acidi 4,5-diidro-1h-pirrol-2-carbossilici e di acidi 1,4,5,6-tetraidropiridin-2-carbussilici | |
IT7925221A0 (it) | Derivati di acidi idrossialcanoici. | |
BG34460A3 (en) | Method of obtaining derivatives of 7 beta-amino- thiazolylacetamido-3-cephem-4-carbonic acid | |
IT1131841B (it) | Derivati di acidi acilamminobenzoici | |
BG43187A3 (en) | Method for preparing of auronic derivatives | |
IT1085323B (it) | Composizioni e metodo per la sgrassatura di substrati | |
IT1164694B (it) | Derivati esterei di acidi chinolopiran-4-on-2-carbossilici e composizioni antiasmatiche che li contengono | |
IT7948195A0 (it) | Derivati di amminoaldeidi utili in particolare per inibire la proliferazione cellulare | |
IT1113377B (it) | Derivati di n-ciano-azometini | |
IT7826520A0 (it) | Derivati dell'acido citrico utili come ammorbidenti. |