IT1156791B - DERIVATIVES OF SILIC ACID THIAZOLIDINCARBOS USEFUL IN PARTICULAR AS ENZYMATIC INHIBITORS - Google Patents

DERIVATIVES OF SILIC ACID THIAZOLIDINCARBOS USEFUL IN PARTICULAR AS ENZYMATIC INHIBITORS

Info

Publication number
IT1156791B
IT1156791B IT49660/78A IT4966078A IT1156791B IT 1156791 B IT1156791 B IT 1156791B IT 49660/78 A IT49660/78 A IT 49660/78A IT 4966078 A IT4966078 A IT 4966078A IT 1156791 B IT1156791 B IT 1156791B
Authority
IT
Italy
Prior art keywords
thiazolidincarbos
derivatives
useful
enzymatic inhibitors
silic acid
Prior art date
Application number
IT49660/78A
Other languages
Italian (it)
Other versions
IT7849660A0 (en
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/907,452 external-priority patent/US4192878A/en
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of IT7849660A0 publication Critical patent/IT7849660A0/en
Application granted granted Critical
Publication of IT1156791B publication Critical patent/IT1156791B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/041,3-Thiazines; Hydrogenated 1,3-thiazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/121,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
IT49660/78A 1978-05-22 1978-06-01 DERIVATIVES OF SILIC ACID THIAZOLIDINCARBOS USEFUL IN PARTICULAR AS ENZYMATIC INHIBITORS IT1156791B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/907,452 US4192878A (en) 1976-12-03 1978-05-22 Derivatives of thiazolidinecarboxylic acids and related acids

Publications (2)

Publication Number Publication Date
IT7849660A0 IT7849660A0 (en) 1978-06-01
IT1156791B true IT1156791B (en) 1987-02-04

Family

ID=25424116

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49660/78A IT1156791B (en) 1978-05-22 1978-06-01 DERIVATIVES OF SILIC ACID THIAZOLIDINCARBOS USEFUL IN PARTICULAR AS ENZYMATIC INHIBITORS

Country Status (18)

Country Link
JP (1) JPS54151965A (en)
AU (1) AU521516B2 (en)
BE (1) BE867776R (en)
CA (1) CA1102812A (en)
CH (1) CH633782A5 (en)
DE (1) DE2823352A1 (en)
DK (1) DK242378A (en)
FR (1) FR2426685A2 (en)
HU (1) HU179780B (en)
IE (1) IE47075B1 (en)
IT (1) IT1156791B (en)
NZ (1) NZ187390A (en)
PH (1) PH14405A (en)
PL (1) PL207332A3 (en)
SE (1) SE7806468L (en)
SU (2) SU730303A3 (en)
YU (1) YU131478A (en)
ZA (1) ZA783013B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4347371A (en) * 1978-12-30 1982-08-31 Santen Pharmaceutical Co., Ltd. Disulfide compounds
US4692458A (en) * 1980-03-05 1987-09-08 University Of Miami Anti-hypertensive agents
RU2526619C2 (en) * 2012-12-12 2014-08-27 Федеральное государственное бюджетное учреждение науки Институт высокомолекулярных соединений Российской академии наук Method of obtaining (2r,4r)-2-alkyl-3-(2-mercaptobenzoyl)-1,3-thiazolidine-4-carboxylic acids

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2404635A1 (en) * 1977-09-28 1979-04-27 Science Union & Cie NEW THIOPROPRIONYLAMIDES, THEIR OBTAINING PROCEDURES AND THEIR USE IN THERAPEUTICS

Also Published As

Publication number Publication date
CH633782A5 (en) 1982-12-31
ZA783013B (en) 1979-06-27
AU3660278A (en) 1979-12-06
FR2426685A2 (en) 1979-12-21
IE781098L (en) 1979-11-22
SU816400A3 (en) 1981-03-23
FR2426685B2 (en) 1981-09-04
PH14405A (en) 1981-06-25
HU179780B (en) 1982-12-28
IT7849660A0 (en) 1978-06-01
PL207332A3 (en) 1980-01-28
BE867776R (en) 1978-12-04
SU730303A3 (en) 1980-04-25
DK242378A (en) 1979-11-23
IE47075B1 (en) 1983-12-14
YU131478A (en) 1984-06-30
CA1102812A (en) 1981-06-09
DE2823352A1 (en) 1979-11-29
JPS54151965A (en) 1979-11-29
AU521516B2 (en) 1982-04-08
NZ187390A (en) 1980-05-27
SE7806468L (en) 1979-11-23

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