IT1098216B - Derivati della 3-(1-pirazolil)-piridazina e procedimento per la loro preparazione - Google Patents

Derivati della 3-(1-pirazolil)-piridazina e procedimento per la loro preparazione

Info

Publication number
IT1098216B
IT1098216B IT24490/78A IT2449078A IT1098216B IT 1098216 B IT1098216 B IT 1098216B IT 24490/78 A IT24490/78 A IT 24490/78A IT 2449078 A IT2449078 A IT 2449078A IT 1098216 B IT1098216 B IT 1098216B
Authority
IT
Italy
Prior art keywords
pyridazin
pyrazolyl
derivatives
procedure
preparation
Prior art date
Application number
IT24490/78A
Other languages
English (en)
Other versions
IT7824490A0 (it
Inventor
Geza Szilagyi
Endre Kasztreiner
Laszlo Tardos
Edit Kosa
Laszlo Jaszlits
Gyorgy Cseh
Andras Divald
Pal Tolnay
Sandor Elek
Istvan Elekes
Istvan Polgari
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of IT7824490A0 publication Critical patent/IT7824490A0/it
Application granted granted Critical
Publication of IT1098216B publication Critical patent/IT1098216B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IT24490/78A 1977-06-13 1978-06-13 Derivati della 3-(1-pirazolil)-piridazina e procedimento per la loro preparazione IT1098216B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU77GO1373A HU175471B (hu) 1977-06-13 1977-06-13 Sposob poluchenija novykh proizvodnykh 3-skobka-1-pirazolil-skobka zakryta-piridazina

Publications (2)

Publication Number Publication Date
IT7824490A0 IT7824490A0 (it) 1978-06-13
IT1098216B true IT1098216B (it) 1985-09-07

Family

ID=10996834

Family Applications (1)

Application Number Title Priority Date Filing Date
IT24490/78A IT1098216B (it) 1977-06-13 1978-06-13 Derivati della 3-(1-pirazolil)-piridazina e procedimento per la loro preparazione

Country Status (25)

Country Link
US (1) US4251658A (it)
JP (1) JPS5416487A (it)
AT (1) AT357548B (it)
AU (1) AU521394B2 (it)
BE (1) BE867967A (it)
BG (1) BG28709A3 (it)
CA (1) CA1095912A (it)
CH (1) CH638202A5 (it)
CS (1) CS204029B2 (it)
DD (1) DD140043A5 (it)
DE (1) DE2825906A1 (it)
DK (1) DK263078A (it)
ES (1) ES470750A1 (it)
FI (1) FI64156C (it)
FR (1) FR2394542A1 (it)
GB (1) GB1603958A (it)
HU (1) HU175471B (it)
IL (1) IL54816A (it)
IT (1) IT1098216B (it)
NL (1) NL7806380A (it)
NO (1) NO149210C (it)
PL (1) PL111252B1 (it)
SE (1) SE437517B (it)
SU (2) SU797577A3 (it)
YU (1) YU140078A (it)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU176100B (en) * 1977-10-25 1980-12-28 Gyogyszerkutato Intezet Process for preparing new 3-/1-pyrazolyl/-pyridazine derivatives
DE2935359A1 (de) * 1979-09-01 1981-03-26 Basf Ag, 67063 Ludwigshafen 6-imidazolyl-3-hydrazino-pyridazine
DE3130251A1 (de) * 1981-07-31 1983-02-17 A. Nattermann & Cie GmbH, 5000 Köln 6-(4-((omega)-(1-imidazolyl)-alkyl)-phenyl)-3-oxo -2,3,4,5-tetrahydro-pyridazine und deren saeureadditionssalze, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
US4353905A (en) * 1981-09-17 1982-10-12 Warner-Lambert Company Substituted 4,5-dihydro-6-[4-(1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinones and 6-[4-(1H-imidazol-1-yl)phenyl]-3(2H)-pyridazinones
US4590194A (en) * 1981-10-05 1986-05-20 Sterling Drug Inc. 3-[methyl or dimethyl)amino]-6-(pyridinyl)pyridazines and their cardiotonic use
US4503056A (en) * 1982-03-02 1985-03-05 Abbott Laboratories 1-(Pyridazinyl)pyrazoline derivatives
DE3825867A1 (de) * 1988-03-04 1989-09-14 Bayer Ag Heterocyclisch substituierte sulfonylaminoazole und ihre verwendung als herbizide
US5536701A (en) * 1994-10-11 1996-07-16 Monsanto Company 3-pyrazolyloxypyridazines, herbicidal compositions and uses thereof
FR2847160A1 (fr) * 2002-11-20 2004-05-21 Oreal Composition capillaire contenant un compose pyrasol-carboxamide, son utilisation pour stimuler la pousse des cheveux et/ou freiner leur chute
AU2003295041A1 (en) * 2002-11-20 2004-06-18 L'oreal Composition for hair care or eyelashes containing a pyrazol-carboxamide, its use for stimulating hair and eyelash growth and/or for preventing loss thereof
RU2442775C2 (ru) * 2005-07-04 2012-02-20 Хай Пойнт Фармасьютикалс, ЛЛС Антагонисты гистаминовых н3-рецепторов
RU2499795C2 (ru) 2005-07-04 2013-11-27 Хай Пойнт Фармасьютикалс, ЛЛС Антагонисты гистаминовых н3-рецепторов
JP2009537596A (ja) * 2006-05-23 2009-10-29 ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー 6−(4−シクロプロピルピペリジン−1−イル)−2’−メチル−[3,4’]−ビピリジン及びその医薬としての使用
WO2007137968A1 (en) * 2006-05-29 2007-12-06 High Point Pharmaceuticals, Llc 3- (1, 3-benz0di0x0l-5-yl) -6- (4-cyclopropylpiperazin-1-yl) -pyridazine, its salts and solvates and its use as histamine h3 receptor antagonist
EP2014656A3 (en) * 2007-06-11 2011-08-24 High Point Pharmaceuticals, LLC New heteocyclic h3 antagonists
AR081626A1 (es) * 2010-04-23 2012-10-10 Cytokinetics Inc Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos
EP2560488B1 (en) 2010-04-23 2015-10-28 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
AR081331A1 (es) 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1595920B2 (de) * 1964-11-04 1978-08-10 Merck Patent Gmbh, 6100 Darmstadt 4-(co-Piperazinoalkyl)-pyrazole, ihre Salze und Verfahren zu ihrer Herstellung
JPS5831347B2 (ja) * 1975-09-05 1983-07-05 中外製薬株式会社 ピラゾリルピリダジンユウドウタイノ セイホウ

Also Published As

Publication number Publication date
CA1095912A (en) 1981-02-17
NO149210B (no) 1983-11-28
AU3683678A (en) 1979-12-06
IL54816A0 (en) 1978-07-31
BE867967A (fr) 1978-12-11
US4251658A (en) 1981-02-17
JPS5416487A (en) 1979-02-07
CH638202A5 (de) 1983-09-15
AT357548B (de) 1980-07-10
SU797577A3 (ru) 1981-01-15
NO782043L (no) 1978-12-14
FI64156B (fi) 1983-06-30
BG28709A3 (en) 1980-06-16
CS204029B2 (en) 1981-03-31
YU140078A (en) 1983-01-21
NO149210C (no) 1984-03-07
IT7824490A0 (it) 1978-06-13
ATA414478A (de) 1979-12-15
FI64156C (fi) 1983-10-10
IL54816A (en) 1981-09-13
GB1603958A (en) 1981-12-02
NL7806380A (nl) 1978-12-15
PL207570A1 (pl) 1979-05-21
DE2825906A1 (de) 1979-01-18
FI781856A (fi) 1978-12-14
SE7806576L (sv) 1978-12-14
SU860703A1 (ru) 1981-08-30
AU521394B2 (en) 1982-04-01
PL111252B1 (en) 1980-08-30
ES470750A1 (es) 1979-01-16
DK263078A (da) 1978-12-14
HU175471B (hu) 1980-08-28
SE437517B (sv) 1985-03-04
DD140043A5 (de) 1980-02-06
FR2394542B1 (it) 1980-12-05
JPS569506B2 (it) 1981-03-02
FR2394542A1 (fr) 1979-01-12

Similar Documents

Publication Publication Date Title
IT1199976B (it) Derivati della camptotecima e processi per la loro preparazione
IT1166917B (it) Derivati delle aldeidi della peptidil-arginina e procediemento per la loro preparazione
IT1088554B (it) Procedimento sellettivo per la preparazione di derivati della 7-indrossi cumarina
IT1098216B (it) Derivati della 3-(1-pirazolil)-piridazina e procedimento per la loro preparazione
IT1160264B (it) Derivati della prostaciclina e procedimento per la loro preparazione
IT7849939A0 (it) Derivati della diidropiridina loro preparazione e loro impiego quali medicamenti
IT1188970B (it) Derivati della moranolina e procedimento per la loro preparazione
IT1075373B (it) Derivati della prostaglandina e procedimento per la loro preparazione
IT7847729A0 (it) Derivati amminoalcossifenilici eprocedimento per la loro preparazione
IT1192621B (it) Derivati della maleinimmide e succinimmide e procedimento per la loro preparazione
IT7968190A0 (it) Derivati della piperidina e procedimento per la loro preparazione
IT1097156B (it) Derivati della 3-(1-pirazolil)-piridazina e procedimento per la loro preparazione
IT1109400B (it) Derivati di 2-amminometil-fenolo e procedimento per la loro preparazione
IT1092747B (it) Derivati solfonilidrazonici e procedimento per la loro preparazione
IT1094864B (it) Derivati della bromexina e procedimento per la loro preparazione
IT1113203B (it) Derivati steroideo-spiro-ossazolidinonici sostituiti e procedimento per la loro preparazione
IT1107844B (it) Derivati della benzammidina procedimento per la loro preparazione e loro impiego terapeutico
IT7847687A0 (it) Derivati della benzo(f)isochinolina loro preparazione e loro applicazione quali medicamenti
IT1212412B (it) Derivati della benzo-as-triazina e procedimento per la loro preparazione.
IT1094209B (it) Derivati di eritromicina semisintetici e procedimento per la loro preparazione
IT1149882B (it) Derivati della pirazolo chinazolina e procedimento per la loro preparazione
IT1148812B (it) Derivati della fenotiazina, e procedimento per la loro preparazione
IT1113251B (it) Derivati della ellebrigenina e procedimento per la loro produzione
IT1156738B (it) Derivati della coriolina e procedimento per la loro produzione
IT1090772B (it) Derivati della rifamicina e procedimento per la loro preparazione