IN2015DN02542A - - Google Patents

Info

Publication number
IN2015DN02542A
IN2015DN02542A IN2542DEN2015A IN2015DN02542A IN 2015DN02542 A IN2015DN02542 A IN 2015DN02542A IN 2542DEN2015 A IN2542DEN2015 A IN 2542DEN2015A IN 2015DN02542 A IN2015DN02542 A IN 2015DN02542A
Authority
IN
India
Prior art keywords
preparation
pyrrolidines
pyridyl
optionally substituted
substituted aryl
Prior art date
Application number
Other languages
English (en)
Inventor
Friedrich August Mühlthau
Mark James Ford
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of IN2015DN02542A publication Critical patent/IN2015DN02542A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • C07C317/02Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms
    • C07C317/10Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • C07C317/14Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • C07C317/16Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C317/18Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/01Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton
    • C07C323/02Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/07Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/10Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C323/11Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/16Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IN2542DEN2015 2012-09-27 2013-09-25 IN2015DN02542A (cs)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12186243 2012-09-27
PCT/EP2013/069919 WO2014048958A1 (en) 2012-09-27 2013-09-25 Process for the preparation of optionally substituted phenyl and pyridyl pyrrolidines

Publications (1)

Publication Number Publication Date
IN2015DN02542A true IN2015DN02542A (cs) 2015-09-11

Family

ID=47044827

Family Applications (1)

Application Number Title Priority Date Filing Date
IN2542DEN2015 IN2015DN02542A (cs) 2012-09-27 2013-09-25

Country Status (13)

Country Link
US (1) US9447036B2 (cs)
EP (1) EP2900634B1 (cs)
JP (1) JP6251749B2 (cs)
KR (1) KR20150059778A (cs)
CN (1) CN104619683B (cs)
BR (1) BR112015006825A2 (cs)
DK (1) DK2900634T3 (cs)
ES (1) ES2625547T3 (cs)
IL (1) IL237749A (cs)
IN (1) IN2015DN02542A (cs)
MX (1) MX350575B (cs)
TW (1) TWI601713B (cs)
WO (1) WO2014048958A1 (cs)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111032617B (zh) * 2017-08-09 2023-02-24 阿尔萨达股份公司 制备4-(七氟-2-丙基)苯胺的方法

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4092349A (en) 1976-11-10 1978-05-30 Pfizer Inc. 11-Desoxy-15-thiaprostaglandins
US4173463A (en) 1978-10-31 1979-11-06 Shell Oil Company Phosphonium salts as herbicides
DK0393424T3 (da) 1989-04-17 1996-02-05 Bayer Ag Fremgangsmåde til fremstilling af 2,7-diazabicyclo(3.3.0)octaner
IT1274021B (it) 1994-02-28 1997-07-14 Italfarmaco Spa Diesteri dell'acido carbonico ad attivita' antivirale ed antinfiammatoria
AU7699196A (en) 1995-11-23 1997-06-11 Rhodia Chimie Perfluoroalkylation method and reagent therefor
JP2000516234A (ja) * 1996-08-16 2000-12-05 デュポン ファーマシューティカルズ カンパニー アミジノフェニル―ピロリジン類、アミジノフェニル―ピロリン類、およびアミジノフェニル―イソオキサゾリジン類およびそれらの誘導体
BR0311419A (pt) 2002-05-28 2005-04-05 Dimensional Pharm Inc Amidinas de tiofeno suas composições e métodos de tratamento de doenças e condições mediadas por complemento
US7230119B2 (en) 2004-08-25 2007-06-12 Biocryst Pharmaceuticals, Inc. Process for the preparation of substituted pyrrolidine derivatives and intermediates
US7521427B2 (en) 2004-11-09 2009-04-21 Georgia Tech Research Corporation Peptidyl allyl sulfones
AR057032A1 (es) 2005-05-27 2007-11-14 Wyeth Corp Tigeciclina y metodos de preparacion
EP1928460A2 (en) 2005-08-01 2008-06-11 Pfizer Limited Mc4r-agonists for the treatment of urinary tract dysfunction
US7750167B2 (en) 2006-07-05 2010-07-06 N.V. Organon Process for the preparation of asenapine and intermediate products used in said process
JP5164510B2 (ja) * 2006-10-06 2013-03-21 日本曹達株式会社 含窒素複素環化合物および有害生物防除剤
GB0623209D0 (en) 2006-11-21 2007-01-03 F2G Ltd Antifungal agents
WO2008129811A1 (ja) 2007-03-23 2008-10-30 Panasonic Corporation 無線送信装置及び無線受信装置
JP2010116389A (ja) 2008-10-17 2010-05-27 Bayer Cropscience Ag 殺虫性アリールピロリジン類
JP2008266230A (ja) 2007-04-23 2008-11-06 Bayer Cropscience Ag 殺虫性アリールピロリジン類
ATE527266T1 (de) 2008-01-04 2011-10-15 Organon Nv Herstellungsverfahren für asenapin und in diesem verfahren verwendete zwischenprodukte
CZ305085B6 (cs) 2008-03-14 2015-04-29 Zentiva, K.S. Způsob přípravy dabigatranu
WO2010086820A1 (en) 2009-02-02 2010-08-05 Pfizer Inc. 4-amino-5-oxo-7, 8-dihydropyrimido [5,4-f] [1,4] oxazepin-6 (5h) -yl) phenyl derivatives, pharmaceutical compositions and uses thereof
HRP20140174T1 (hr) 2009-02-27 2014-04-25 Ambit Biosciences Corporation Derivati kinazolina kao modulatori jak-kinaze i postupci njihove upotrebe
BRPI1014641A2 (pt) 2009-04-30 2019-09-24 Bayer Cropscience Ag arilpirrolidinas pesticidas
SG176100A1 (en) * 2009-05-22 2011-12-29 Abbott Lab Modulators of 5-ht receptors and methods of use thereof
MX2012000583A (es) 2009-07-16 2012-02-13 Bayer Cropscience Ag Procedimiento para la preparacion de derivados de 3-triazolil-sulfoxido quirales.
JP2011136928A (ja) 2009-12-28 2011-07-14 Bayer Cropscience Ag 殺虫性アリールピロリジン類
JP2012082186A (ja) 2010-09-15 2012-04-26 Bayer Cropscience Ag 殺虫性アリールピロリジン類
BR112015004826A2 (pt) * 2012-09-07 2017-07-04 Zoetis Llc derivados espirocíclicos como agentes antiparasíticos

Also Published As

Publication number Publication date
US9447036B2 (en) 2016-09-20
EP2900634B1 (en) 2017-02-22
TW201418215A (zh) 2014-05-16
MX350575B (es) 2017-09-11
WO2014048958A1 (en) 2014-04-03
EP2900634A1 (en) 2015-08-05
CN104619683A (zh) 2015-05-13
TWI601713B (zh) 2017-10-11
BR112015006825A2 (pt) 2017-08-08
IL237749A (en) 2017-09-28
JP6251749B2 (ja) 2017-12-20
ES2625547T3 (es) 2017-07-19
KR20150059778A (ko) 2015-06-02
JP2015535835A (ja) 2015-12-17
MX2015003902A (es) 2015-07-17
US20150246880A1 (en) 2015-09-03
CN104619683B (zh) 2017-05-10
DK2900634T3 (en) 2017-05-22

Similar Documents

Publication Publication Date Title
JOP20180103A1 (ar) مركب صيدلاني
PH12014502613A1 (en) Synthesis of heterocyclic compound
IL235767A0 (en) Converted pyrrolidines as factor xia inhibitors for the treatment of thromboembolic diseases
MD20150091A2 (ro) Compuşi antivirali
UA110813C2 (uk) Лікування ліподистрофії
IN2015DN00847A (cs)
EP3674320A3 (en) Production of heterodimeric proteins
MY177031A (en) Tetrahydropyridopyrazines modulators of gpr6
GEP20247677B (en) Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds
IN2015DN00598A (cs)
IN2015DN01061A (cs)
DK3395357T3 (da) Sammensætning til kontrolleret ovariestimulering
ZA201406494B (en) Methods of producing sulfilimine compounds
CR20140495A (es) 5-amino[1,4]thiazines como inhibidores de bace1
TW201613934A (en) Methods for the preparation of 1,3-benzodioxole heterocyclic compounds
IN2014DN06192A (cs)
WO2013168176A3 (en) Process for preparation of fosaprepitant and salt thereof
IL238545A0 (en) Plants for the production of medical proteins
IN2014DN09451A (cs)
MX2015005739A (es) Compuestos novedosos de bencil sulfonamida utiles como inhibidores de mogat-2.
MX2012010443A (es) Proceso para la preparacion de 1-alquiltetrazoles 5-sustituidos.
MX348841B (es) Derivados de pirimidooxazocina como inhibidores de mtor.
MX2014002378A (es) Proceso para la preparacion de (r)-2-acetamido-n-bencil-3-metoxipr opionamida e intermediarios de la misma.
IN2015DN02542A (cs)
NZ702523A (en) Production of n-substituted sulfoximine pyridine n-oxides