IN2014MN02467A - - Google Patents
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- Publication number
- IN2014MN02467A IN2014MN02467A IN2467MUN2014A IN2014MN02467A IN 2014MN02467 A IN2014MN02467 A IN 2014MN02467A IN 2467MUN2014 A IN2467MUN2014 A IN 2467MUN2014A IN 2014MN02467 A IN2014MN02467 A IN 2014MN02467A
- Authority
- IN
- India
- Prior art keywords
- tetrahydrothieno
- thiazol
- dioxo
- pyrimidin
- difluoro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
- C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/60—Three or more oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
- Y10T428/00—Stock material or miscellaneous articles
- Y10T428/29—Coated or structually defined flake, particle, cell, strand, strand portion, rod, filament, macroscopic fiber or mass thereof
- Y10T428/2982—Particulate matter [e.g., sphere, flake, etc.]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN2467MUN2014 IN2014MN02467A (fr) | 2012-06-08 | 2013-06-08 |
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1687MU2012 | 2012-06-08 | ||
US201261665282P | 2012-06-27 | 2012-06-27 | |
IN3519MU2012 | 2012-12-13 | ||
US201261748016P | 2012-12-31 | 2012-12-31 | |
IN2467MUN2014 IN2014MN02467A (fr) | 2012-06-08 | 2013-06-08 | |
PCT/IB2013/054703 WO2013183035A2 (fr) | 2012-06-08 | 2013-06-08 | Amides de composés de 2-amino-4-arylthiazole et leurs sels |
Publications (1)
Publication Number | Publication Date |
---|---|
IN2014MN02467A true IN2014MN02467A (fr) | 2015-07-10 |
Family
ID=54193746
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IN2467MUN2014 IN2014MN02467A (fr) | 2012-06-08 | 2013-06-08 |
Country Status (22)
Country | Link |
---|---|
US (1) | US9458173B2 (fr) |
EP (1) | EP2858999B1 (fr) |
JP (1) | JP5989900B2 (fr) |
KR (1) | KR20150015488A (fr) |
CN (1) | CN104350058A (fr) |
AP (1) | AP3546A (fr) |
AU (1) | AU2013273118B2 (fr) |
BR (1) | BR112014029155A2 (fr) |
CA (1) | CA2873570C (fr) |
CL (1) | CL2014003317A1 (fr) |
EA (1) | EA031334B1 (fr) |
HK (1) | HK1207643A1 (fr) |
IL (1) | IL236084A0 (fr) |
IN (1) | IN2014MN02467A (fr) |
MX (1) | MX354014B (fr) |
MY (1) | MY165622A (fr) |
NZ (1) | NZ701721A (fr) |
PE (1) | PE20142306A1 (fr) |
PH (1) | PH12014502685B1 (fr) |
SG (1) | SG11201408093PA (fr) |
WO (1) | WO2013183035A2 (fr) |
ZA (1) | ZA201500082B (fr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR091279A1 (es) | 2012-06-08 | 2015-01-21 | Gilead Sciences Inc | Inhibidores macrociclicos de virus flaviviridae |
JP6209601B2 (ja) | 2012-06-08 | 2017-10-04 | ギリアード サイエンシーズ, インコーポレイテッド | フラビウイルス科ウイルスの大環状阻害剤 |
WO2014203210A1 (fr) | 2013-06-20 | 2014-12-24 | Glenmark Pharmaceuticals S.A. | Formulation nanoparticulaire comprenant un antagoniste de trpa1 |
JP6573968B2 (ja) * | 2014-08-11 | 2019-09-11 | ハイドラ バイオサイエンシズ インコーポレイテッドHydra Biosciences,Inc. | TRPC5調節因子としての、精神神経障害の処置のためのチエノおよびフロ[2,3−d]ピリミジン−2,4[1H,3H]−ジオン誘導体 |
WO2016042501A1 (fr) * | 2014-09-16 | 2016-03-24 | Glenmark Pharmaceuticals S.A. | Antagoniste de trpa1 permettant le traitement de la douleur associée à la douleur neuropathique diabétique |
TW202321229A (zh) | 2021-08-18 | 2023-06-01 | 美商富曼西公司 | 殺真菌的取代的雜環化合物 |
CN114671875A (zh) * | 2022-04-27 | 2022-06-28 | 成都施贝康生物医药科技有限公司 | 新型二氢嘧啶类化合物、异构体或盐及其制备方法和用途 |
Family Cites Families (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2248231A1 (de) | 1972-10-02 | 1974-04-11 | Basf Ag | 3-aminoisothiazolo eckige klammer auf 3,4-d eckige klammer zu pyrimidine |
SE9701398D0 (sv) | 1997-04-15 | 1997-04-15 | Astra Pharma Prod | Novel compounds |
ES2193839B1 (es) | 2001-06-22 | 2005-02-16 | Almirall Prodesfarma, S.A. | Nuevos derivados de 6-fenildihidropirrolpirimidindiona. |
AU2003253165A1 (en) * | 2002-08-13 | 2004-02-25 | Warner-Lambert Company Llc | Pyrimidine fused bicyclic metalloproteinase inhibitors |
US6890923B2 (en) | 2002-12-16 | 2005-05-10 | Astrazeneca Ab | Compounds |
US7465581B2 (en) | 2002-12-18 | 2008-12-16 | The Scripps Research Institute | ANKTM1, a cold-activated TRP-like channel expressed in nociceptive neurons |
CA2536313A1 (fr) | 2003-08-22 | 2005-03-03 | Takeda Pharmaceutical Company Limited | Derive de pyrimidine fusionne et utilisation associee |
EP1713815A4 (fr) | 2004-02-11 | 2009-03-11 | Smithkline Beecham Corp | Agonistes de pth |
US20070196866A1 (en) | 2004-03-13 | 2007-08-23 | Irm Llc | Modulators of ion channel trpa1 |
JPWO2006083005A1 (ja) | 2005-02-03 | 2008-06-26 | 武田薬品工業株式会社 | 縮合ピリミジン誘導体およびその用途 |
WO2007019251A2 (fr) | 2005-08-04 | 2007-02-15 | Apogee Biotechnology Corporation | Inhibiteurs de la sphingosine kinase et leurs methodes d'utilisation |
US20070105920A1 (en) | 2005-11-08 | 2007-05-10 | Akzo Nobel N.V. | 2-(Benzimidazol-1-Yl)-N-(4-phenylthiazol-2-yl) acetamide derivatives |
JP5858557B2 (ja) * | 2005-12-22 | 2016-02-10 | ハイドラ バイオサイエンシズ インコーポレイテッドHydra Biosciences,Inc. | 疼痛を処置するためのtrpa1阻害剤 |
TW200800997A (en) | 2006-03-22 | 2008-01-01 | Astrazeneca Ab | Chemical compounds |
CN101454318A (zh) * | 2006-03-22 | 2009-06-10 | 阿斯利康(瑞典)有限公司 | 吡啶并嘧啶衍生物及其作为pde4抑制剂的用途 |
JP2011201776A (ja) | 2008-07-23 | 2011-10-13 | Mochida Pharmaceut Co Ltd | ヘテロシクリデン−n−(3,4−ジヒドロ−2(1h)−キナゾリノン−5−イル)アセトアミド誘導体 |
AR065081A1 (es) | 2007-01-29 | 2009-05-13 | Xenon Pharmaceuticals Inc | Compuestos de quinazolinona y pirimidona fusionados y composicion farmaceutica |
EP3663295A1 (fr) | 2007-06-22 | 2020-06-10 | Eli Lilly And Co. | Composés de 2,6-dioxo,-2,3-dihydro-1h-purines utiles pour le traitement de troubles liés à l'activité du canal trpa1 |
US7951814B2 (en) * | 2008-06-17 | 2011-05-31 | Glenmark Pharmaceuticals, S.A. | Quinazolinedione derivatives as TRPA1 modulators |
WO2009158719A2 (fr) | 2008-06-27 | 2009-12-30 | Hydra Biosciences, Inc. | Méthodes et compositions de traitement de troubles |
PT2411395E (pt) * | 2009-03-23 | 2013-06-06 | Glenmark Pharmaceuticals Sa | Derivados de furopirimidinadiona como moduladores de trpa1 |
AP2011005888A0 (en) | 2009-03-23 | 2011-10-31 | Glenmark Pharmaceuticals Sa | Isothiazolo-pyrimidinedione derivatives as TRPA1 modulators. |
US8623880B2 (en) | 2009-03-23 | 2014-01-07 | Glenmark Pharmaceuticals S.A. | Fused pyrimidine-dione derivatives as TRPA1 modulators |
ES2551085T3 (es) | 2009-03-23 | 2015-11-16 | Glenmark Pharmaceuticals S.A. | Proceso para preparar derivados de pirimidina-diona condensados, útiles como moduladores de TRPA1 |
EA023141B1 (ru) | 2010-12-20 | 2016-04-29 | Гленмарк Фармасьютикалс С.А. | Соединения 2-амино-4-арилтиазола в качестве антагонистов trpa1 |
-
2013
- 2013-06-08 KR KR1020147033855A patent/KR20150015488A/ko active IP Right Grant
- 2013-06-08 MY MYPI2014003389A patent/MY165622A/en unknown
- 2013-06-08 US US14/402,608 patent/US9458173B2/en active Active
- 2013-06-08 WO PCT/IB2013/054703 patent/WO2013183035A2/fr active Application Filing
- 2013-06-08 CA CA2873570A patent/CA2873570C/fr active Active
- 2013-06-08 EA EA201492054A patent/EA031334B1/ru unknown
- 2013-06-08 BR BR112014029155A patent/BR112014029155A2/pt not_active Application Discontinuation
- 2013-06-08 MX MX2014014482A patent/MX354014B/es active IP Right Grant
- 2013-06-08 AP AP2014008076A patent/AP3546A/xx active
- 2013-06-08 IN IN2467MUN2014 patent/IN2014MN02467A/en unknown
- 2013-06-08 AU AU2013273118A patent/AU2013273118B2/en not_active Ceased
- 2013-06-08 CN CN201380030184.XA patent/CN104350058A/zh active Pending
- 2013-06-08 EP EP13742279.6A patent/EP2858999B1/fr active Active
- 2013-06-08 PE PE2014002226A patent/PE20142306A1/es not_active Application Discontinuation
- 2013-06-08 JP JP2015515642A patent/JP5989900B2/ja not_active Expired - Fee Related
- 2013-06-08 SG SG11201408093PA patent/SG11201408093PA/en unknown
- 2013-06-08 NZ NZ701721A patent/NZ701721A/en not_active IP Right Cessation
-
2014
- 2014-12-02 PH PH12014502685A patent/PH12014502685B1/en unknown
- 2014-12-04 CL CL2014003317A patent/CL2014003317A1/es unknown
- 2014-12-04 IL IL236084A patent/IL236084A0/en unknown
-
2015
- 2015-01-07 ZA ZA2015/00082A patent/ZA201500082B/en unknown
- 2015-08-27 HK HK15108333.2A patent/HK1207643A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
CA2873570A1 (fr) | 2013-12-12 |
AP2014008076A0 (en) | 2014-11-30 |
ZA201500082B (en) | 2015-12-23 |
NZ701721A (en) | 2016-03-31 |
MY165622A (en) | 2018-04-18 |
AP3546A (en) | 2016-01-14 |
EA201492054A1 (ru) | 2016-08-31 |
BR112014029155A2 (pt) | 2017-06-27 |
MX2014014482A (es) | 2015-06-05 |
AU2013273118B2 (en) | 2015-11-05 |
PE20142306A1 (es) | 2015-01-16 |
PH12014502685A1 (en) | 2015-01-26 |
JP2015520183A (ja) | 2015-07-16 |
KR20150015488A (ko) | 2015-02-10 |
IL236084A0 (en) | 2015-02-01 |
US9458173B2 (en) | 2016-10-04 |
CL2014003317A1 (es) | 2015-02-13 |
AU2013273118A1 (en) | 2014-11-27 |
CN104350058A (zh) | 2015-02-11 |
PH12014502685B1 (en) | 2015-01-26 |
US20150111038A1 (en) | 2015-04-23 |
WO2013183035A3 (fr) | 2014-02-27 |
EA031334B1 (ru) | 2018-12-28 |
EP2858999A2 (fr) | 2015-04-15 |
EP2858999B1 (fr) | 2017-05-10 |
MX354014B (es) | 2018-02-08 |
SG11201408093PA (en) | 2015-01-29 |
CA2873570C (fr) | 2016-11-01 |
WO2013183035A2 (fr) | 2013-12-12 |
JP5989900B2 (ja) | 2016-09-07 |
HK1207643A1 (en) | 2016-02-05 |
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