IL99062A - Gondolibrin antagonists their preparation and use - Google Patents

Gondolibrin antagonists their preparation and use

Info

Publication number
IL99062A
IL99062A IL9906291A IL9906291A IL99062A IL 99062 A IL99062 A IL 99062A IL 9906291 A IL9906291 A IL 9906291A IL 9906291 A IL9906291 A IL 9906291A IL 99062 A IL99062 A IL 99062A
Authority
IL
Israel
Prior art keywords
ser
phe
leu
trp
rha
Prior art date
Application number
IL9906291A
Other languages
English (en)
Hebrew (he)
Other versions
IL99062A0 (en
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of IL99062A0 publication Critical patent/IL99062A0/xx
Publication of IL99062A publication Critical patent/IL99062A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/23Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL9906291A 1990-08-04 1991-08-02 Gondolibrin antagonists their preparation and use IL99062A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4024779 1990-08-04

Publications (2)

Publication Number Publication Date
IL99062A0 IL99062A0 (en) 1992-07-15
IL99062A true IL99062A (en) 1995-07-31

Family

ID=6411646

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9906291A IL99062A (en) 1990-08-04 1991-08-02 Gondolibrin antagonists their preparation and use

Country Status (17)

Country Link
US (1) US5434138A (no)
EP (1) EP0477499B1 (no)
JP (1) JP3164844B2 (no)
KR (1) KR100191700B1 (no)
AT (1) ATE100822T1 (no)
AU (1) AU641035B2 (no)
CA (1) CA2048407C (no)
DE (1) DE59100945D1 (no)
DK (1) DK0477499T3 (no)
ES (1) ES2062628T3 (no)
IE (1) IE65965B1 (no)
IL (1) IL99062A (no)
NO (1) NO309429B1 (no)
NZ (1) NZ239233A (no)
PT (1) PT98533B (no)
TW (1) TW205046B (no)
ZA (1) ZA916097B (no)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5691314A (en) * 1996-03-18 1997-11-25 The Medical College Of Hampton Roads Adjunctive therapy
CN1301771A (zh) * 1999-12-27 2001-07-04 上海博德基因开发有限公司 一种新的多肽——人促性腺释放激素11和编码这种多肽的多核苷酸
US11805833B1 (en) * 2019-05-10 2023-11-07 Julie Vahos Flexible hair extension with form retention capability
WO2023101490A1 (ko) * 2021-12-01 2023-06-08 애니젠 주식회사 가니렐릭스의 신규한 제조방법

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54148722A (en) * 1978-05-12 1979-11-21 Takeda Chem Ind Ltd Nonapeptide and its preparation
US5073624A (en) * 1985-04-09 1991-12-17 Administrators Of The Tulane Educational Fund Therapeutic decapeptides
US4661472A (en) * 1985-05-09 1987-04-28 The Salk Institute For Biological Studies GnRH antagonists IX
DE3634435A1 (de) * 1986-10-09 1988-04-14 Hoechst Ag Analoga von gonadoliberin mit verbesserter loeslichkeit, verfahren zu deren herstellung, diese enthaltende mittel und ihre verwendung
US4801577A (en) * 1987-02-05 1989-01-31 Syntex (U.S.A.) Inc. Nonapeptide and decapeptide analogs of LHRH useful as LHRH antagonists
US5110904A (en) * 1989-08-07 1992-05-05 Abbott Laboratories Lhrh analogs
DK163689A (da) * 1988-04-08 1989-10-30 Sandoz Ag Peptidderivater

Also Published As

Publication number Publication date
NZ239233A (en) 1993-09-27
AU8154891A (en) 1992-02-06
ES2062628T3 (es) 1994-12-16
IE65965B1 (en) 1995-11-29
IL99062A0 (en) 1992-07-15
JPH05148299A (ja) 1993-06-15
EP0477499A1 (de) 1992-04-01
NO913020L (no) 1992-02-05
NO913020D0 (no) 1991-08-02
DE59100945D1 (de) 1994-03-10
US5434138A (en) 1995-07-18
IE912769A1 (en) 1992-02-12
AU641035B2 (en) 1993-09-09
JP3164844B2 (ja) 2001-05-14
CA2048407C (en) 2001-10-23
ATE100822T1 (de) 1994-02-15
NO309429B1 (no) 2001-01-29
CA2048407A1 (en) 1992-02-05
TW205046B (no) 1993-05-01
PT98533B (pt) 1999-01-29
DK0477499T3 (da) 1994-05-30
KR100191700B1 (ko) 1999-06-15
EP0477499B1 (de) 1994-01-26
PT98533A (pt) 1992-06-30
KR920004417A (ko) 1992-03-27
ZA916097B (en) 1992-04-29

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Legal Events

Date Code Title Description
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees