IL97828A - Substituted 4-amino-thieno¬2,3-b¾thiopyran-(and thiepin)-2-sulfonamides and pharmaceutical compositions containing them - Google Patents
Substituted 4-amino-thieno¬2,3-b¾thiopyran-(and thiepin)-2-sulfonamides and pharmaceutical compositions containing themInfo
- Publication number
- IL97828A IL97828A IL9782891A IL9782891A IL97828A IL 97828 A IL97828 A IL 97828A IL 9782891 A IL9782891 A IL 9782891A IL 9782891 A IL9782891 A IL 9782891A IL 97828 A IL97828 A IL 97828A
- Authority
- IL
- Israel
- Prior art keywords
- thieno
- sulfonamides
- substituted
- thiepin
- amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Lubricants (AREA)
- Non-Silver Salt Photosensitive Materials And Non-Silver Salt Photography (AREA)
- Photosensitive Polymer And Photoresist Processing (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US50780590A | 1990-04-12 | 1990-04-12 |
Publications (2)
Publication Number | Publication Date |
---|---|
IL97828A0 IL97828A0 (en) | 1992-06-21 |
IL97828A true IL97828A (en) | 2000-06-01 |
Family
ID=24020208
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL9782891A IL97828A (en) | 1990-04-12 | 1991-04-11 | Substituted 4-amino-thieno¬2,3-b¾thiopyran-(and thiepin)-2-sulfonamides and pharmaceutical compositions containing them |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP0452151B1 (no) |
KR (1) | KR0182610B1 (no) |
AT (1) | ATE155468T1 (no) |
AU (1) | AU645075B2 (no) |
CA (1) | CA2040312C (no) |
DE (1) | DE69126814T2 (no) |
DK (1) | DK0452151T3 (no) |
ES (1) | ES2104663T3 (no) |
FI (1) | FI98371C (no) |
GR (1) | GR3024818T3 (no) |
IE (1) | IE911192A1 (no) |
IL (1) | IL97828A (no) |
NO (1) | NO180680C (no) |
NZ (1) | NZ237783A (no) |
PT (1) | PT97359B (no) |
ZA (1) | ZA912703B (no) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP3031498B2 (ja) * | 1990-04-12 | 2000-04-10 | メルク エンド カムパニー インコーポレーテッド | 抗緑内障剤としての置換芳香族スルホンアミド類 |
CA2129037C (en) * | 1992-02-21 | 1998-03-24 | Thomas Robert Dean | Topical antiglaucoma compositions comprising carbonic anhydrase inhibitors and beta-blockers |
US5932572A (en) * | 1992-02-21 | 1999-08-03 | Alcon Laboratories, Inc. | Topical anti-glaucoma compositions |
US5276025A (en) * | 1992-09-09 | 1994-01-04 | Merck & Co., Inc. | Heterobicyclic sulfonamides |
AU3722793A (en) * | 1992-09-17 | 1994-04-12 | Alcon Laboratories, Inc. | Topical carbonic anhydrase inhibitor composition |
US5646142A (en) * | 1994-07-08 | 1997-07-08 | Alcon Laboratories, Inc. | Thiophene sulfonamides useful as carbonic anhydrase inhibitors |
US5510347A (en) * | 1994-09-09 | 1996-04-23 | Alcon Laboratories, Inc. | Thienothiadiazine sulfonamides useful as carbonic anhydrase inhibitors |
US5464831A (en) * | 1994-09-09 | 1995-11-07 | Alcon Laboratories, Inc. | Thienothiadiazine sulfonamides useful as carbonic anhydrase inhibitors |
FR2754712B1 (fr) | 1996-10-17 | 1999-09-03 | Merck Sharp Dohme Chibret Lab | Compositions ophtalmiques |
ES2177415B1 (es) * | 2000-09-04 | 2004-10-16 | Ragactives, S.L. | Procedimiento para la obtencion de 4-alquilamino-5, 6-dihidro-4h-tieno-(2,3b)-tiopiran-2-sulfonamida-7-dioxidos, e intermedios. |
EP1918293A1 (en) * | 2006-10-02 | 2008-05-07 | Sandoz AG | Process for the preparation of 6-substituted-4-oxo-thieno [2,3b]thiopyran-2-sulfonic acid |
EA030535B1 (ru) | 2013-10-17 | 2018-08-31 | Сентисс Фарма Прайвет Лимитед | Не содержащий консерванта офтальмологический фармацевтический состав |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4797413A (en) * | 1986-05-14 | 1989-01-10 | Merck & Co., Inc. | Thieno thiopyran sulfonamide derivatives, pharmaceutical compositions and use |
US4863922A (en) * | 1984-12-12 | 1989-09-05 | Merck & Co., Inc. | Substituted aromatic sulfonamides as antiglaucoma agents, compositions and use |
US4677115A (en) * | 1984-12-12 | 1987-06-30 | Merck & Co., Inc. | Antiglaucoma thieno-thiopyran and thieno-thiepin sulfonamide derivatives, compositions, and method of use thereof |
EP0193132B1 (en) * | 1985-03-01 | 1991-04-17 | Hoechst-Roussel Pharmaceuticals Incorporated | Labdan-derivatives, a process for their preparation and their use as medicaments |
US4816474A (en) * | 1987-02-27 | 1989-03-28 | Ciba-Geigy Corporation | Amino substituted thienothiopyran derivatives, composition containing them, and method of using them to stimulate presynaptic dopamine receptors |
US5120757A (en) * | 1989-07-31 | 1992-06-09 | Merck & Co., Inc. | Substituted aromatic sulfonamides as antiglaucoma agents |
IL96507A0 (en) * | 1989-12-08 | 1991-08-16 | Merck & Co Inc | Nitrogen-containing spirocycles and pharmaceutical compositions containing them |
-
1991
- 1991-04-09 IE IE119291A patent/IE911192A1/en unknown
- 1991-04-10 NZ NZ237783A patent/NZ237783A/en unknown
- 1991-04-11 AU AU74343/91A patent/AU645075B2/en not_active Ceased
- 1991-04-11 NO NO911420A patent/NO180680C/no not_active IP Right Cessation
- 1991-04-11 ZA ZA912703A patent/ZA912703B/xx unknown
- 1991-04-11 FI FI911747A patent/FI98371C/fi not_active IP Right Cessation
- 1991-04-11 IL IL9782891A patent/IL97828A/xx not_active IP Right Cessation
- 1991-04-12 KR KR1019910005824A patent/KR0182610B1/ko not_active IP Right Cessation
- 1991-04-12 ES ES91303269T patent/ES2104663T3/es not_active Expired - Lifetime
- 1991-04-12 DE DE69126814T patent/DE69126814T2/de not_active Expired - Fee Related
- 1991-04-12 CA CA002040312A patent/CA2040312C/en not_active Expired - Fee Related
- 1991-04-12 DK DK91303269.4T patent/DK0452151T3/da active
- 1991-04-12 PT PT97359A patent/PT97359B/pt not_active IP Right Cessation
- 1991-04-12 AT AT91303269T patent/ATE155468T1/de not_active IP Right Cessation
- 1991-04-12 EP EP91303269A patent/EP0452151B1/en not_active Expired - Lifetime
-
1997
- 1997-09-24 GR GR970402452T patent/GR3024818T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
IE911192A1 (en) | 1991-10-23 |
ATE155468T1 (de) | 1997-08-15 |
PT97359A (pt) | 1991-12-31 |
AU645075B2 (en) | 1994-01-06 |
NO911420L (no) | 1991-10-14 |
DE69126814T2 (de) | 1998-02-12 |
ES2104663T3 (es) | 1997-10-16 |
NO180680B (no) | 1997-02-17 |
DK0452151T3 (da) | 1997-09-08 |
KR910018386A (ko) | 1991-11-30 |
ZA912703B (en) | 1991-12-24 |
CA2040312C (en) | 2001-06-12 |
FI911747A0 (fi) | 1991-04-11 |
FI98371C (fi) | 1997-06-10 |
NO911420D0 (no) | 1991-04-11 |
AU7434391A (en) | 1991-10-17 |
CA2040312A1 (en) | 1991-10-13 |
IL97828A0 (en) | 1992-06-21 |
GR3024818T3 (en) | 1998-01-30 |
FI911747A (fi) | 1991-10-13 |
EP0452151B1 (en) | 1997-07-16 |
DE69126814D1 (de) | 1997-08-21 |
PT97359B (pt) | 1998-08-31 |
KR0182610B1 (ko) | 1999-05-01 |
NO180680C (no) | 1997-05-28 |
FI98371B (fi) | 1997-02-28 |
EP0452151A1 (en) | 1991-10-16 |
NZ237783A (en) | 1994-05-26 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IL97828A (en) | Substituted 4-amino-thieno¬2,3-b¾thiopyran-(and thiepin)-2-sulfonamides and pharmaceutical compositions containing them | |
IL86822A (en) | 6-alkyl-4-amino-5,6-dihydro-4h-thieno(2,3-b)thiopyran-2-sulfonamide-7,7-dioxides and antiglaucoma compositions containing them | |
GB2211407B (en) | 4h-benz[4,5]cyclohepta[1,2-b]thiophene derivatives as il-1 inhibitors | |
IL96367A (en) | 5,11-dihydro-6H-dipyrido [3,2-b:2', 3'-e][1,4] diazepine-6-(thi)ones their preparation and pharmaceutical compositions containing them | |
IE830331L (en) | Thiophene derivatives | |
NZ218207A (en) | Hexahydro-(1)-benzo(pyrano and thiopyrano)(4,3-c)- pyridines and pharmaceutical compositions | |
EP0204129A3 (en) | Use of calcium channel blockers in the production of compositions for reconstructive surgery | |
DK429788A (da) | Thieno(2,3-beta)thiophen-2-sulfonamid og farmaceutisk praeparat indeholdende en saadan forbindelse | |
AU626861B2 (en) | 2-(2-nitrovinyl) thiophene reduction and synthesis of thieno (3,2-c) pyridine derivatives | |
IL80906A0 (en) | 4h-benzo(4,5)cyclohepta(1,2-b)-thiophene derivatives,their production and pharmaceutical compositions containing them | |
DE68910950D1 (de) | Substituierte Thieno(3,2-B)thiophen-2-sulfonamide als topisch aktive Kohlensäureanhydraseinhibitoren. | |
GB9324727D0 (en) | Children's amusement ride | |
IL121373A0 (en) | A molecular marker for the gene determining the fructose to glucose ratio in mature tomato fruit | |
CS257089A1 (en) | /dimethylaminomethyl/phenyl derivatives 6,11-dihydrodibenzo /b,e/ thiepin's and their salts | |
EP0354013A3 (en) | Improvements in or relating to ram units in transmissions of the toroidal race, rolling traction type | |
FR2655551B1 (fr) | Portique de gymnastique sportive a cablerie de suspension d'anneaux rigide. | |
IT8505115V0 (it) | Variazione della posizione di corpi disposti in modo compatto all'interno di un contenitore mediante la loro rotazione,realizzazione di nuovi giochi di abilita'e di strategia | |
IT8604704V0 (it) | Variazione della posizione di corpi disposti in modo compatto traloro e formanti una sfera cava, mediante la loro rotazione realizzazione di nuovi giochi di abilita' e strategia | |
IL93381A0 (en) | Ophthalmic compositions comprising a carbonic anhydrase inhibitor | |
IE842615L (en) | BENZOCYCLOHEPTA (1,2-b) THIOPHENE DERIVATIVES | |
CS342088A1 (en) | N,m-disubstituted amino of n-(2-/cyan-4,5,6,7-tetrahydrobenzo/b/thienyl)/thiocarbamic acid and method of their production | |
IT8647559A0 (it) | Dispositivo applicabile a piste sportive e simili, per la visualizzazione dell'avanzamento su ritmi programmati | |
IE883735L (en) | Thieno (3,4-b) benzodiazepinones | |
HUT66017A (en) | 1-phenyl-1a,2,3,4,6,7,12,12ba-octahydro-pyrimido[1',6',:1,2]pyrido[3,4-b] indole-derivatives and pharmaceutical composition containing them and process for their production | |
NZ242777A (en) | Benzene- or thiophene- carboxylic acid derivatives |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FF | Patent granted | ||
KB | Patent renewed | ||
KB | Patent renewed | ||
MM9K | Patent not in force due to non-payment of renewal fees |