ES2104663T3 - Sulfonamidas aromaticas sustituidas como agentes antiglaucoma. - Google Patents
Sulfonamidas aromaticas sustituidas como agentes antiglaucoma.Info
- Publication number
- ES2104663T3 ES2104663T3 ES91303269T ES91303269T ES2104663T3 ES 2104663 T3 ES2104663 T3 ES 2104663T3 ES 91303269 T ES91303269 T ES 91303269T ES 91303269 T ES91303269 T ES 91303269T ES 2104663 T3 ES2104663 T3 ES 2104663T3
- Authority
- ES
- Spain
- Prior art keywords
- aromatic sulfonamides
- antiglaucoma agents
- substituted
- sulfonamides substituted
- thiopyran
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Lubricants (AREA)
- Non-Silver Salt Photosensitive Materials And Non-Silver Salt Photography (AREA)
- Photosensitive Polymer And Photoresist Processing (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
SULFONAMIDAS-2-TIENO[2,3-B]TIOPIRAN Y ANILLOS HOMOLOGOS CON UN GRUPO DE ALQUILO SUSTITUIDO HIDROFILICO ADYACENTE AL SULFURO TIOPIRANO SON INHIBIDORES DE ANHIDRASA CARBONICA TOPICAMENTE EFECTIVOS EN BAJAR LA PRESION INTRAOCULAR.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US50780590A | 1990-04-12 | 1990-04-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2104663T3 true ES2104663T3 (es) | 1997-10-16 |
Family
ID=24020208
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES91303269T Expired - Lifetime ES2104663T3 (es) | 1990-04-12 | 1991-04-12 | Sulfonamidas aromaticas sustituidas como agentes antiglaucoma. |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP0452151B1 (es) |
KR (1) | KR0182610B1 (es) |
AT (1) | ATE155468T1 (es) |
AU (1) | AU645075B2 (es) |
CA (1) | CA2040312C (es) |
DE (1) | DE69126814T2 (es) |
DK (1) | DK0452151T3 (es) |
ES (1) | ES2104663T3 (es) |
FI (1) | FI98371C (es) |
GR (1) | GR3024818T3 (es) |
IE (1) | IE911192A1 (es) |
IL (1) | IL97828A (es) |
NO (1) | NO180680C (es) |
NZ (1) | NZ237783A (es) |
PT (1) | PT97359B (es) |
ZA (1) | ZA912703B (es) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP3031498B2 (ja) * | 1990-04-12 | 2000-04-10 | メルク エンド カムパニー インコーポレーテッド | 抗緑内障剤としての置換芳香族スルホンアミド類 |
US5932572A (en) * | 1992-02-21 | 1999-08-03 | Alcon Laboratories, Inc. | Topical anti-glaucoma compositions |
ATE169499T1 (de) * | 1992-02-21 | 1998-08-15 | Alcon Lab Inc | Topische antiglaukoma zusammensetzungen, enthaltend karbonhydrasehemmer und beta-blocker |
US5276025A (en) * | 1992-09-09 | 1994-01-04 | Merck & Co., Inc. | Heterobicyclic sulfonamides |
JPH08501303A (ja) * | 1992-09-17 | 1996-02-13 | アルコン ラボラトリーズ,インコーポレイテッド | 局所用炭酸脱水酵素阻害剤組成物 |
US5646142A (en) * | 1994-07-08 | 1997-07-08 | Alcon Laboratories, Inc. | Thiophene sulfonamides useful as carbonic anhydrase inhibitors |
US5510347A (en) * | 1994-09-09 | 1996-04-23 | Alcon Laboratories, Inc. | Thienothiadiazine sulfonamides useful as carbonic anhydrase inhibitors |
US5464831A (en) * | 1994-09-09 | 1995-11-07 | Alcon Laboratories, Inc. | Thienothiadiazine sulfonamides useful as carbonic anhydrase inhibitors |
FR2754712B1 (fr) | 1996-10-17 | 1999-09-03 | Merck Sharp Dohme Chibret Lab | Compositions ophtalmiques |
ES2177415B1 (es) * | 2000-09-04 | 2004-10-16 | Ragactives, S.L. | Procedimiento para la obtencion de 4-alquilamino-5, 6-dihidro-4h-tieno-(2,3b)-tiopiran-2-sulfonamida-7-dioxidos, e intermedios. |
EP1918293A1 (en) * | 2006-10-02 | 2008-05-07 | Sandoz AG | Process for the preparation of 6-substituted-4-oxo-thieno [2,3b]thiopyran-2-sulfonic acid |
UA116273C2 (uk) | 2013-10-17 | 2018-02-26 | Сентісс Фарма Прайвет Лімітед | Офтальмологічний фармацевтичний склад, що не містить консерванта |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4863922A (en) * | 1984-12-12 | 1989-09-05 | Merck & Co., Inc. | Substituted aromatic sulfonamides as antiglaucoma agents, compositions and use |
US4677115A (en) * | 1984-12-12 | 1987-06-30 | Merck & Co., Inc. | Antiglaucoma thieno-thiopyran and thieno-thiepin sulfonamide derivatives, compositions, and method of use thereof |
US4797413A (en) * | 1986-05-14 | 1989-01-10 | Merck & Co., Inc. | Thieno thiopyran sulfonamide derivatives, pharmaceutical compositions and use |
ATE62683T1 (de) * | 1985-03-01 | 1991-05-15 | Hoechst Roussel Pharma | Labdanderivate, verfahren zu deren herstellung und deren verwendung als arzneimittel. |
US4816474A (en) * | 1987-02-27 | 1989-03-28 | Ciba-Geigy Corporation | Amino substituted thienothiopyran derivatives, composition containing them, and method of using them to stimulate presynaptic dopamine receptors |
US5120757A (en) * | 1989-07-31 | 1992-06-09 | Merck & Co., Inc. | Substituted aromatic sulfonamides as antiglaucoma agents |
IL96507A0 (en) * | 1989-12-08 | 1991-08-16 | Merck & Co Inc | Nitrogen-containing spirocycles and pharmaceutical compositions containing them |
-
1991
- 1991-04-09 IE IE119291A patent/IE911192A1/en unknown
- 1991-04-10 NZ NZ237783A patent/NZ237783A/en unknown
- 1991-04-11 NO NO911420A patent/NO180680C/no not_active IP Right Cessation
- 1991-04-11 FI FI911747A patent/FI98371C/fi not_active IP Right Cessation
- 1991-04-11 IL IL9782891A patent/IL97828A/xx not_active IP Right Cessation
- 1991-04-11 ZA ZA912703A patent/ZA912703B/xx unknown
- 1991-04-11 AU AU74343/91A patent/AU645075B2/en not_active Ceased
- 1991-04-12 PT PT97359A patent/PT97359B/pt not_active IP Right Cessation
- 1991-04-12 KR KR1019910005824A patent/KR0182610B1/ko not_active IP Right Cessation
- 1991-04-12 CA CA002040312A patent/CA2040312C/en not_active Expired - Fee Related
- 1991-04-12 DK DK91303269.4T patent/DK0452151T3/da active
- 1991-04-12 DE DE69126814T patent/DE69126814T2/de not_active Expired - Fee Related
- 1991-04-12 EP EP91303269A patent/EP0452151B1/en not_active Expired - Lifetime
- 1991-04-12 AT AT91303269T patent/ATE155468T1/de not_active IP Right Cessation
- 1991-04-12 ES ES91303269T patent/ES2104663T3/es not_active Expired - Lifetime
-
1997
- 1997-09-24 GR GR970402452T patent/GR3024818T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
AU645075B2 (en) | 1994-01-06 |
FI911747A (fi) | 1991-10-13 |
FI911747A0 (fi) | 1991-04-11 |
DE69126814D1 (de) | 1997-08-21 |
IE911192A1 (en) | 1991-10-23 |
NO180680C (no) | 1997-05-28 |
FI98371B (fi) | 1997-02-28 |
CA2040312C (en) | 2001-06-12 |
NZ237783A (en) | 1994-05-26 |
AU7434391A (en) | 1991-10-17 |
FI98371C (fi) | 1997-06-10 |
IL97828A0 (en) | 1992-06-21 |
KR0182610B1 (ko) | 1999-05-01 |
PT97359B (pt) | 1998-08-31 |
IL97828A (en) | 2000-06-01 |
NO911420D0 (no) | 1991-04-11 |
DK0452151T3 (da) | 1997-09-08 |
EP0452151A1 (en) | 1991-10-16 |
ATE155468T1 (de) | 1997-08-15 |
ZA912703B (en) | 1991-12-24 |
PT97359A (pt) | 1991-12-31 |
NO911420L (no) | 1991-10-14 |
GR3024818T3 (en) | 1998-01-30 |
KR910018386A (ko) | 1991-11-30 |
DE69126814T2 (de) | 1998-02-12 |
NO180680B (no) | 1997-02-17 |
CA2040312A1 (en) | 1991-10-13 |
EP0452151B1 (en) | 1997-07-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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