IL95085A - Benzoxazolones 4,5,6,7-Tetraforms are converted into anti-allergy and anti-allergy pharmaceuticals - Google Patents

Benzoxazolones 4,5,6,7-Tetraforms are converted into anti-allergy and anti-allergy pharmaceuticals

Info

Publication number
IL95085A
IL95085A IL9508590A IL9508590A IL95085A IL 95085 A IL95085 A IL 95085A IL 9508590 A IL9508590 A IL 9508590A IL 9508590 A IL9508590 A IL 9508590A IL 95085 A IL95085 A IL 95085A
Authority
IL
Israel
Prior art keywords
fluoro
compound
hydrogen
formula
benzoxazolone
Prior art date
Application number
IL9508590A
Other languages
English (en)
Hebrew (he)
Other versions
IL95085A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL95085A0 publication Critical patent/IL95085A0/xx
Publication of IL95085A publication Critical patent/IL95085A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Non-Silver Salt Photosensitive Materials And Non-Silver Salt Photography (AREA)
IL9508590A 1989-07-20 1990-07-13 Benzoxazolones 4,5,6,7-Tetraforms are converted into anti-allergy and anti-allergy pharmaceuticals IL95085A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP1188683A JPH0678327B2 (ja) 1989-07-20 1989-07-20 ４，５，６，７，―四置換ベンゾオキサゾロン類

Publications (2)

Publication Number Publication Date
IL95085A0 IL95085A0 (en) 1991-06-10
IL95085A true IL95085A (en) 1994-10-21

Family

ID=16228012

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9508590A IL95085A (en) 1989-07-20 1990-07-13 Benzoxazolones 4,5,6,7-Tetraforms are converted into anti-allergy and anti-allergy pharmaceuticals

Country Status (18)

Country Link
US (1) US5071863A (ko)
EP (1) EP0409484B1 (ko)
JP (1) JPH0678327B2 (ko)
KR (1) KR930002099B1 (ko)
AT (1) ATE106877T1 (ko)
AU (1) AU616608B2 (ko)
CA (1) CA2021421A1 (ko)
DE (1) DE69009607T2 (ko)
DK (1) DK0409484T3 (ko)
ES (1) ES2055332T3 (ko)
FI (1) FI95378C (ko)
HU (1) HU206101B (ko)
IE (1) IE63203B1 (ko)
IL (1) IL95085A (ko)
NO (1) NO903230L (ko)
NZ (1) NZ234583A (ko)
PT (1) PT94750A (ko)
ZA (1) ZA905677B (ko)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2674524B1 (fr) * 1991-03-25 1993-05-21 Adir Nouveaux amides alkyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US20040192669A1 (en) * 2000-04-13 2004-09-30 Rosenfeld Mark J. Novel compounds for use in weight loss and appetite suppression in humans
US7794761B2 (en) * 2000-04-13 2010-09-14 Seroctin Research & Technology, Inc. Methods for inducing anti-anxiety and calming effects in animals and humans
US7524877B2 (en) 2003-11-20 2009-04-28 Seroctin Research & Technology, Inc. Compounds for use in weight loss and appetite suppression in humans
JP4695012B2 (ja) * 2006-04-21 2011-06-08 セイコークロック株式会社 アラーム時計
NZ590688A (en) 2008-08-05 2012-09-28 Daiichi Sankyo Co Ltd imidazo[4,5-b]pyridin-2-one derivatives

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3256293A (en) * 1964-02-05 1966-06-14 Monsanto Co 3-(phenylcarbamoyl) benzoxazolinones-2
US3657265A (en) * 1968-06-21 1972-04-18 Olin Corp Process for preparing benzoxazolones from aromatic nitro compounds
CA1048035A (en) * 1971-09-28 1979-02-06 Jozef Drabek Dithiophosphoric acid esters
US4227915A (en) * 1978-05-18 1980-10-14 Monsanto Company N-Substituted oxobenzothiazoline and oxobenzoxazoline derivatives and their use as plant growth regulants
JPS57123103A (en) * 1981-01-26 1982-07-31 Hokko Chem Ind Co Ltd Agricultural and horticultural fungicide
GB8325370D0 (en) * 1983-09-22 1983-10-26 Fujisawa Pharmaceutical Co Benzoxazoline and benzothiazoline derivatives
JPS6293283A (ja) * 1985-10-18 1987-04-28 Idemitsu Kosan Co Ltd ベンゾオキサゾロン誘導体，その製造方法およびそれを有効成分とする農園芸用殺菌剤
DK288287A (da) * 1986-06-09 1987-12-10 Pfizer Heterocycliske forbindelser samt farmaceutiske praeparater til behandling af allergiske eller inflammatoriske tilstande
US4835166A (en) * 1986-06-09 1989-05-30 Pfizer Inc. Antiallergy and antiinflammatory agents
IL93473A0 (en) * 1989-02-28 1990-11-29 Pfizer Antiinflammatory benzoxazolones

Also Published As

Publication number Publication date
FI95378C (fi) 1996-01-25
IL95085A0 (en) 1991-06-10
JPH0352875A (ja) 1991-03-07
NZ234583A (en) 1991-12-23
NO903230D0 (no) 1990-07-19
IE902630A1 (en) 1991-02-27
PT94750A (pt) 1991-03-20
AU616608B2 (en) 1991-10-31
FI903655A0 (fi) 1990-07-19
HUT57745A (en) 1991-12-30
KR910002818A (ko) 1991-02-26
ES2055332T3 (es) 1994-08-16
HU904565D0 (en) 1990-12-28
JPH0678327B2 (ja) 1994-10-05
CA2021421A1 (en) 1991-01-21
EP0409484A2 (en) 1991-01-23
HU206101B (en) 1992-08-28
KR930002099B1 (ko) 1993-03-26
DE69009607D1 (de) 1994-07-14
US5071863A (en) 1991-12-10
AU5919390A (en) 1991-01-24
EP0409484B1 (en) 1994-06-08
DE69009607T2 (de) 1994-09-22
IE63203B1 (en) 1995-04-05
ZA905677B (en) 1992-02-26
DK0409484T3 (da) 1994-07-04
ATE106877T1 (de) 1994-06-15
EP0409484A3 (en) 1991-05-15
NO903230L (no) 1991-01-21
FI95378B (fi) 1995-10-13

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Legal Events

Date Code Title Description
KB Patent renewed
RH Patent void