IL88573A - 2-plasmin inhibitor depressant, urokinase secretion accelerator or thrombolytic composition comprising trihydroxypiperidine derivatives, nojirimycin or castanospermine - Google Patents

2-plasmin inhibitor depressant, urokinase secretion accelerator or thrombolytic composition comprising trihydroxypiperidine derivatives, nojirimycin or castanospermine

Info

Publication number
IL88573A
IL88573A IL8857388A IL8857388A IL88573A IL 88573 A IL88573 A IL 88573A IL 8857388 A IL8857388 A IL 8857388A IL 8857388 A IL8857388 A IL 8857388A IL 88573 A IL88573 A IL 88573A
Authority
IL
Israel
Prior art keywords
acid addition
physiologically acceptable
acceptable acid
addition salt
nojirimycin
Prior art date
Application number
IL8857388A
Other languages
English (en)
Original Assignee
Nippon Shinyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Shinyaku Co Ltd filed Critical Nippon Shinyaku Co Ltd
Publication of IL88573A publication Critical patent/IL88573A/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7004Monosaccharides having only carbon, hydrogen and oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
IL8857388A 1987-12-09 1988-12-04 2-plasmin inhibitor depressant, urokinase secretion accelerator or thrombolytic composition comprising trihydroxypiperidine derivatives, nojirimycin or castanospermine IL88573A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP31134887 1987-12-09

Publications (1)

Publication Number Publication Date
IL88573A true IL88573A (en) 1994-05-30

Family

ID=18016066

Family Applications (1)

Application Number Title Priority Date Filing Date
IL8857388A IL88573A (en) 1987-12-09 1988-12-04 2-plasmin inhibitor depressant, urokinase secretion accelerator or thrombolytic composition comprising trihydroxypiperidine derivatives, nojirimycin or castanospermine

Country Status (11)

Country Link
EP (1) EP0319986B1 (fr)
KR (1) KR960009417B1 (fr)
AT (1) ATE149836T1 (fr)
BE (1) BE1004874A4 (fr)
CA (1) CA1316831C (fr)
CH (1) CH677610A5 (fr)
DE (1) DE3855824T2 (fr)
FR (1) FR2626470B1 (fr)
GB (2) GB8827701D0 (fr)
IL (1) IL88573A (fr)
SE (1) SE502110C2 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990001319A1 (fr) * 1988-08-10 1990-02-22 The Australian National University Utilisation de castanospermine comme agent anti-inflammatoire et immunosuppresseur
WO1998006264A1 (fr) * 1996-08-14 1998-02-19 Myung Hee Chun Therapie par appauvrissement de la plasmine
EP1903034A1 (fr) * 2006-09-19 2008-03-26 Technische Universität Graz Iminosucres glycoconjugués

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54106477A (en) * 1978-02-03 1979-08-21 Nippon Shinyaku Co Ltd Moranoline derivative
JPS5943946B2 (ja) * 1978-04-28 1984-10-25 日本新薬株式会社 N−アルケニルモラノリン誘導体
JPS5943947B2 (ja) * 1978-05-03 1984-10-25 日本新薬株式会社 N−置換モラノリン誘導体
GB2020278B (en) * 1978-05-03 1983-02-23 Nippon Shinyaku Co Ltd Moranoline dervitives
JPS6026387B2 (ja) * 1979-01-20 1985-06-24 日本新薬株式会社 シンナミルモラノリン誘導体
JPS5943949B2 (ja) * 1978-09-29 1984-10-25 日本新薬株式会社 モラノリンのn−置換誘導体
DE2925943A1 (de) * 1979-06-27 1981-01-29 Bayer Ag 1-alkadien-2,4-yl-2-hydroxymethyl3,4,5-trihydroxypiperidine, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
JPS56108767A (en) * 1980-01-28 1981-08-28 Nippon Shinyaku Co Ltd Bismoranoline derivative
DE3007078A1 (de) * 1980-02-26 1981-09-10 Bayer Ag, 5090 Leverkusen Neue derivate von 3,4,5-trihydroxypiperidin, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel sowie in der tierernaehrung
JPS60224675A (ja) * 1984-04-24 1985-11-09 Meiji Seika Kaisha Ltd 新規1−デオキシノジリマイシン誘導体およびそれを含有する血中脂質低下剤
CA1327970C (fr) * 1985-05-24 1994-03-22 Paul S. Liu Isolement de la castanospermine et son usage comme agent antidiabetique
DE3650377T2 (de) * 1985-12-23 1996-02-22 Hutchinson Fred Cancer Res Regulierung der retroviralen replikation, infektion und pathogenese.
ZA883925B (en) * 1987-06-08 1989-02-22 Merrell Dow Pharma Inhibitors of glycoprotein processing having anti-retroviral activity

Also Published As

Publication number Publication date
GB2213374B (en) 1992-01-29
CH677610A5 (fr) 1991-06-14
EP0319986A3 (fr) 1992-09-30
BE1004874A4 (fr) 1993-02-16
KR890009399A (ko) 1989-08-01
FR2626470B1 (fr) 1994-12-09
ATE149836T1 (de) 1997-03-15
CA1316831C (fr) 1993-04-27
GB8827927D0 (en) 1989-01-05
GB8827701D0 (en) 1988-12-29
DE3855824T2 (de) 1997-10-16
SE8804436D0 (sv) 1988-12-08
KR960009417B1 (ko) 1996-07-19
FR2626470A1 (fr) 1989-08-04
SE8804436L (sv) 1989-06-10
SE502110C2 (sv) 1995-08-21
DE3855824D1 (de) 1997-04-17
EP0319986A2 (fr) 1989-06-14
GB2213374A (en) 1989-08-16
EP0319986B1 (fr) 1997-03-12

Similar Documents

Publication Publication Date Title
CA2113229A1 (fr) Compositions anti-fibreuses contenant de la quinazolinone et methodes d'utilisation correspondantes
GR3005315T3 (fr)
HU9500240D0 (en) New prolin-amide derivatives and pharmaceutical compositions containing them as active component
HUT52770A (en) Process for producing new 2-amino-pyrimidinone derivatives and pharmaceutical compositions containing them
HK1003708A1 (en) Peripheral vasodilating agent containing n-acylated 4-amino piperidine derivatives as active ingredients
HU895609D0 (en) Process for the preparation of novel 1,4-diazepine derivatives and pharmaceutical compositions containing such compounds
HUT52059A (en) Process for producing pharmaceutical compositions and new quinoline derivatives as a group of active components
AU1433588A (en) 1-phenyl-3-naphthalenyloxypropanamines
ES8802421A1 (es) Un procedimiento para la preparacion de un derivado de acido 5-imidazolcarboxilico
ES542125A0 (es) Un procedimiento para preparar un derivado de 1,5-benzotiazepina.
IL88573A (en) 2-plasmin inhibitor depressant, urokinase secretion accelerator or thrombolytic composition comprising trihydroxypiperidine derivatives, nojirimycin or castanospermine
EP0123962A3 (en) Novel benzimidazole derivative, process for the preparation thereof and pharmaceutical composition
EP0335979A4 (en) Thienopyrimidine derivatives
CA1264753C (fr) 2-pyridylcarboxamides
CA2118425A1 (fr) Derive du benzothiazolesulfamide, son mode de preparation et son utilisation
ES8801615A1 (es) Un procedimiento para preparar esteres de acidos ciclopropanocarboxolico que contienen fluor.
ATE50248T1 (de) Ein imidazolidintrion-derivat oder ein seiner pharmazeutisch akzeptierbaren salze enthaltende pharmazeutische zusammenstellung.
GR3007219T3 (fr)
EP0414903A4 (en) New thioproline derivative
AU8835291A (en) 5-amino-5,6,7,8-tetrahydroquinolines and related compounds and pharmaceutical use
EP0376162A3 (fr) Produit inhibant la formation de plaque dentaire
WO2001035938A3 (fr) Derives tetrahydrothiopyran-4-ol pharmacologiquement actifs, leur procede de fabrication et leur utilisation
ATE131480T1 (de) Pyrimidoindolderivate und verfahren zu ihrer herstellung
AU657423B2 (en) Novel piperidine derivatives and process for preparation thereof
ES8604210A1 (es) Procedimiento para preparar 2- (fenetil) -5- (3,4-metilen- dioxi)-x-hidroxibencil) -pirrolidina

Legal Events

Date Code Title Description
RH Patent void