IL81010A - 4-(4,5-dihydro-2-(imidazolyl,oxazolyl or thiazolyl))-amino benzamides,their preparation and pharmaceutical compositions containing them - Google Patents
4-(4,5-dihydro-2-(imidazolyl,oxazolyl or thiazolyl))-amino benzamides,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL81010A IL81010A IL81010A IL8101086A IL81010A IL 81010 A IL81010 A IL 81010A IL 81010 A IL81010 A IL 81010A IL 8101086 A IL8101086 A IL 8101086A IL 81010 A IL81010 A IL 81010A
- Authority
- IL
- Israel
- Prior art keywords
- oxazolyl
- thiazolyl
- imidazolyl
- dihydro
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/28—Nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/18—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IL95681A IL95681A (en) | 1985-12-19 | 1986-12-17 | Substituted alkyl 4-(4,5-dihydro-2-(imidazolyl,oxazolyl or thiazolyl)amino)benzoates and their preparation |
IL95681A IL95681A0 (en) | 1985-12-19 | 1990-09-13 | Substituted benzoic acid esters and their preparation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8518829A FR2592042B1 (fr) | 1985-12-19 | 1985-12-19 | Nouveaux ortho-anisamides, leur procede d'obtention, et leurs applications therapeutiques |
Publications (2)
Publication Number | Publication Date |
---|---|
IL81010A0 IL81010A0 (en) | 1987-03-31 |
IL81010A true IL81010A (en) | 1991-06-30 |
Family
ID=9325965
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL81010A IL81010A (en) | 1985-12-19 | 1986-12-17 | 4-(4,5-dihydro-2-(imidazolyl,oxazolyl or thiazolyl))-amino benzamides,their preparation and pharmaceutical compositions containing them |
Country Status (37)
Country | Link |
---|---|
US (2) | US4835172A (de) |
EP (1) | EP0236646B1 (de) |
JP (1) | JPS62246553A (de) |
KR (1) | KR930004653B1 (de) |
CN (1) | CN1018454B (de) |
AR (1) | AR242193A1 (de) |
AT (1) | ATE57376T1 (de) |
AU (1) | AU586057B2 (de) |
CA (2) | CA1298301C (de) |
CH (1) | CH671396A5 (de) |
CS (1) | CS274285B2 (de) |
DD (1) | DD260495A5 (de) |
DE (2) | DE3674916D1 (de) |
DK (1) | DK612886A (de) |
ES (1) | ES2036178T3 (de) |
FI (1) | FI865190A (de) |
FR (1) | FR2592042B1 (de) |
GB (1) | GB2184723B (de) |
GR (1) | GR3002524T3 (de) |
HU (1) | HU196794B (de) |
IE (1) | IE59212B1 (de) |
IL (1) | IL81010A (de) |
IN (1) | IN163130B (de) |
IS (1) | IS1448B6 (de) |
MA (1) | MA20835A1 (de) |
NO (1) | NO168176C (de) |
NZ (1) | NZ218675A (de) |
OA (1) | OA08564A (de) |
PH (2) | PH24365A (de) |
PL (1) | PL148408B1 (de) |
PT (1) | PT83982B (de) |
SU (1) | SU1496632A3 (de) |
TN (1) | TNSN86165A1 (de) |
YU (1) | YU44796B (de) |
ZA (1) | ZA869560B (de) |
ZM (1) | ZM10686A1 (de) |
ZW (1) | ZW24886A1 (de) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3782651T2 (de) * | 1987-06-17 | 1993-03-25 | Delagrange Lab | Anwendung von n-(2-(diaethylamino)aethyl)-2-methoxy-4((1-h-4,5-dihydro-2-imidazolyl)amino)-5-chlorobenzamid als anxiolytisches und antipsychotisches mittel. |
FR2640139A1 (fr) * | 1988-12-14 | 1990-06-15 | Delagrange Laboratoires | Application de benzamides substitues comme gastromoteurs |
FR2640507A1 (fr) * | 1988-12-20 | 1990-06-22 | Delagrange Laboratoires | Application de benzamides substitues comme anxiolytiques et anti-psychotiques |
FR2645742A1 (fr) * | 1989-04-12 | 1990-10-19 | Delagrange Laboratoires | Application de derives de 2-methoxy 4-(4,5-dihydro 2-imidazolyl (ou 2-oxazolyl) amino) 5-chloro benzamide dans le traitement des troubles de la fonction cognitive |
US5401851A (en) * | 1992-06-03 | 1995-03-28 | Eli Lilly And Company | Angiotensin II antagonists |
US20050140688A1 (en) * | 2003-12-29 | 2005-06-30 | Kim Pallister | Method and mechanism for programmable filtering of texture map data in 3D graphics subsystems |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3342826A (en) * | 1964-01-13 | 1967-09-19 | Ile De France | Heterocyclic aminoalkyl benzamides |
FR1539104A (fr) * | 1967-07-31 | 1968-09-13 | Ile De France | Nouveaux benzamides et leur procédé de préparation |
US3682968A (en) * | 1969-06-25 | 1972-08-08 | Merck & Co Inc | Anti-inflammatory salicylic acid derivatives |
DE1963193A1 (de) * | 1969-12-17 | 1971-06-24 | Bayer Ag | N-substituierte 2-Arylimino-oxazolidine,Verfahren zu ihrer Herstellung und ihre Verwendung als Ektoparasiticide |
FR2432513A1 (fr) * | 1977-10-24 | 1980-02-29 | Merieux Inst | Nouveaux derives de la thiazoline et leur application comme medicaments |
DE2905883A1 (de) * | 1979-02-16 | 1980-08-28 | Boehringer Sohn Ingelheim | Radioimmuntest fuer clonidin |
US4461904A (en) * | 1981-11-20 | 1984-07-24 | Alcon Laboratories, Inc. | 2-(Trisubstituted phenylimino)-imidazolines |
CA1201066A (en) * | 1981-11-20 | 1986-02-25 | Alcon Laboratories, Inc. | N-¬3,5-dichloro-4-(2-imidazolidinylideneamino)- phenyl|-acetamide solutions for lowering intraocular pressure |
DE3514351A1 (de) * | 1985-04-20 | 1986-11-06 | Boehringer Ingelheim KG, 6507 Ingelheim | Neue substituierte 2-(n-alkinyl-n-phenyl)amino)-imidazolinderivate, deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zu deren herstellung |
JPS6341471A (ja) * | 1986-08-08 | 1988-02-22 | Nippon Soda Co Ltd | オキサ(チア)ゾリジン誘導体、その製造法及び殺ダニ剤 |
US4826990A (en) * | 1987-09-30 | 1989-05-02 | American Home Products Corporation | 2-aryl substituted heterocyclic compounds as antiallergic and antiinflammatory agents |
-
1985
- 1985-12-19 FR FR8518829A patent/FR2592042B1/fr not_active Expired
-
1986
- 1986-12-15 ES ES198686402796T patent/ES2036178T3/es not_active Expired - Lifetime
- 1986-12-15 IE IE327086A patent/IE59212B1/en not_active IP Right Cessation
- 1986-12-15 AT AT86402796T patent/ATE57376T1/de active
- 1986-12-15 EP EP86402796A patent/EP0236646B1/de not_active Expired - Lifetime
- 1986-12-15 DE DE8686402796T patent/DE3674916D1/de not_active Expired - Lifetime
- 1986-12-16 CH CH4997/86A patent/CH671396A5/fr not_active IP Right Cessation
- 1986-12-16 IN IN983/MAS/86A patent/IN163130B/en unknown
- 1986-12-17 NZ NZ218675A patent/NZ218675A/xx unknown
- 1986-12-17 IL IL81010A patent/IL81010A/xx not_active IP Right Cessation
- 1986-12-17 DD DD86297795A patent/DD260495A5/de not_active IP Right Cessation
- 1986-12-17 DE DE19863643103 patent/DE3643103A1/de not_active Withdrawn
- 1986-12-17 PH PH34606A patent/PH24365A/en unknown
- 1986-12-17 GB GB8630143A patent/GB2184723B/en not_active Expired
- 1986-12-17 HU HU865271A patent/HU196794B/hu not_active IP Right Cessation
- 1986-12-17 MA MA21067A patent/MA20835A1/fr unknown
- 1986-12-17 IS IS3178A patent/IS1448B6/is unknown
- 1986-12-17 AR AR86306202A patent/AR242193A1/es active
- 1986-12-18 ZM ZM106/86A patent/ZM10686A1/xx unknown
- 1986-12-18 FI FI865190A patent/FI865190A/fi not_active Application Discontinuation
- 1986-12-18 AU AU66687/86A patent/AU586057B2/en not_active Ceased
- 1986-12-18 CN CN86108972A patent/CN1018454B/zh not_active Expired
- 1986-12-18 SU SU864028722A patent/SU1496632A3/ru active
- 1986-12-18 OA OA59022A patent/OA08564A/xx unknown
- 1986-12-18 NO NO865148A patent/NO168176C/no unknown
- 1986-12-18 YU YU2179/86A patent/YU44796B/xx unknown
- 1986-12-18 PL PL1986263078A patent/PL148408B1/pl unknown
- 1986-12-18 KR KR1019860010868A patent/KR930004653B1/ko not_active IP Right Cessation
- 1986-12-18 CA CA000525719A patent/CA1298301C/fr not_active Expired - Lifetime
- 1986-12-18 DK DK612886A patent/DK612886A/da not_active Application Discontinuation
- 1986-12-19 TN TNTNSN86165A patent/TNSN86165A1/fr unknown
- 1986-12-19 PT PT83982A patent/PT83982B/pt not_active IP Right Cessation
- 1986-12-19 US US06/943,708 patent/US4835172A/en not_active Expired - Fee Related
- 1986-12-19 CS CS960386A patent/CS274285B2/cs unknown
- 1986-12-19 JP JP61305136A patent/JPS62246553A/ja active Pending
- 1986-12-19 ZW ZW248/86A patent/ZW24886A1/xx unknown
- 1986-12-19 ZA ZA869560A patent/ZA869560B/xx unknown
-
1988
- 1988-02-17 PH PH36522A patent/PH24469A/en unknown
-
1989
- 1989-03-13 US US07/322,122 patent/US4914117A/en not_active Expired - Fee Related
-
1990
- 1990-10-22 CA CA000615908A patent/CA1299579C/fr not_active Expired - Lifetime
- 1990-11-13 GR GR90400910T patent/GR3002524T3/el unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NZ222977A (en) | Aminotetralins and pharmaceutical compositions; 8-substituted-2-aminotetralins and pharmaceutical compositions thereof | |
PT84737A (en) | N-(2(-aminophenyl)-benzamide derivatives process for the preparation thereof and pharmaceutical compositions containing them | |
PH24049A (en) | Substituted benzamide derivatives and pharmaceutical compositions containing the same | |
IL87080A (en) | 4-amino-5-halo 2,n-disubstituted benzamides,their preparation and pharmaceutical compositions containing them | |
IL85704A0 (en) | Thiazole derivatives,their preparation and pharmaceutical compositions containing them | |
IL88670A0 (en) | 2,5-diaryl-tetrahydrofurans and analogs thereof and pharmaceutical compositions containing them | |
NZ223875A (en) | 9-aminotetrahydroacridines and related homologues and pharmaceutical compositions | |
AR242574A1 (es) | Nuevas (indolil-(hexa- o tetra-)hidropiridin-1-il-alquil)-tiazol y procedimiento para la preparacion de los mismos. | |
IL80339A (en) | 2-(2-(2-pyridyl)- phenylsulphinyl) -benzimidazoles, their preparation and pharmaceutical compositions containing them | |
IL65097A0 (en) | N-(4-(indolyl)-piperidino-alkyl)-benzimidazolones,their preparation and pharmaceutical compositions containing them | |
IL71185A (en) | Pharmaceutical compositions comprising n-(piperidinyl-alkyl))carboxamides,some such novel compounds and their preparation | |
IL81874A0 (en) | Substituted thiazoles and oxazoles,their preparation and pharmaceutical compositions containing them | |
IL85223A0 (en) | N-(aryl-,aryloxy-,arylthio-,arylsulfinyl-and arylsulfonyl-)alkyl-n,n-(or n',n')alkylaminoalkyl ureas,thioureas and cyanoguanidines and pharmaceutical compositions containing them | |
DE3568333D1 (en) | Novel 4,5-bis(4-methoxyphenyl)-2-(pyrrol-2-yl)thiazoles, process for the preparation thereof and pharmaceutical composition containing the same | |
AU1706788A (en) | 2-(3,4-dihydroxyphenyl)ethylamines, and their use pharmaceutical compositions | |
IL80835A0 (en) | N-(pyrrol-1-yl)pyridinamines,a process for their preparation and pharmaceutical compositions containing them | |
IL81010A (en) | 4-(4,5-dihydro-2-(imidazolyl,oxazolyl or thiazolyl))-amino benzamides,their preparation and pharmaceutical compositions containing them | |
PT85360B (en) | Process for the preparation of a fungicidal composition containing n-(2-cyano-2-oxyminoacetyl)-aminonitriles and intermediate products | |
NZ219719A (en) | Endo-4-amino-5-chloro-2-methoxy-n-cl-azabicyclo -(3,3,1)-non-4-yl)-benzamide and pharmaceutical compositions | |
IL63217A0 (en) | N-(1-allyl-2-pyrrolidinyl-methyl)2-methoxy-4-amino-5-methylsulfamoyl benzamide,its preparation and pharmaceutical compositions containing it | |
IL80733A0 (en) | 2,2'-bi-1h-imidazoles and pharmaceutical compositions containing same | |
IL67647A (en) | 6-aminoalkylpenicillanic acid 1,1-dioxides and derivatives thereof and pharmaceutical compositions containing them | |
IL79241A (en) | N-((2-imidazolin-2-yl)alkyl)-4-amino-5-halo benzamide derivatives,their preparation and pharmaceutical compositions containing them | |
NZ214231A (en) | 1,3,4-thiadiazole derivatives and pharmaceutical compositions | |
KR900700471A (ko) | 신규의 2,3-티오모르폴린디온-2-옥심유도체, 이들을 함유하는 약제학적 조성물 및 제법 |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
RH | Patent void |