IL76020A - 3-(acylaminomethyl)-2-phenyl imidazo(1,2-a)pyridine derivatives,their preparation and pharmaceutical compositions containing them - Google Patents
3-(acylaminomethyl)-2-phenyl imidazo(1,2-a)pyridine derivatives,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL76020A IL76020A IL76020A IL7602085A IL76020A IL 76020 A IL76020 A IL 76020A IL 76020 A IL76020 A IL 76020A IL 7602085 A IL7602085 A IL 7602085A IL 76020 A IL76020 A IL 76020A
- Authority
- IL
- Israel
- Prior art keywords
- acylaminomethyl
- preparation
- pharmaceutical compositions
- compositions containing
- pyridine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8412447A FR2568880B1 (fr) | 1984-08-07 | 1984-08-07 | Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
IL76020A0 IL76020A0 (en) | 1985-12-31 |
IL76020A true IL76020A (en) | 1989-01-31 |
Family
ID=9306856
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL76020A IL76020A (en) | 1984-08-07 | 1985-08-06 | 3-(acylaminomethyl)-2-phenyl imidazo(1,2-a)pyridine derivatives,their preparation and pharmaceutical compositions containing them |
Country Status (23)
Country | Link |
---|---|
US (1) | US4650796A (fi) |
EP (1) | EP0172096B1 (fi) |
JP (1) | JPS6147485A (fi) |
KR (1) | KR910004450B1 (fi) |
AR (1) | AR241185A1 (fi) |
AT (1) | ATE40365T1 (fi) |
AU (1) | AU575190B2 (fi) |
CA (1) | CA1261830A (fi) |
CZ (1) | CZ357691A3 (fi) |
DE (1) | DE3567867D1 (fi) |
DK (1) | DK163923C (fi) |
ES (1) | ES8604592A1 (fi) |
FI (1) | FI80696C (fi) |
FR (1) | FR2568880B1 (fi) |
GR (1) | GR851928B (fi) |
HU (1) | HU193799B (fi) |
IE (1) | IE58347B1 (fi) |
IL (1) | IL76020A (fi) |
MX (1) | MX160845A (fi) |
NO (1) | NO162189C (fi) |
NZ (1) | NZ213013A (fi) |
PT (1) | PT80921B (fi) |
ZA (1) | ZA855939B (fi) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE62687T1 (de) * | 1986-01-22 | 1991-05-15 | Synthelabo | Acylaminomethylimidazo(1,2-a>pyrimidinderivate, ihre herstellung und therapeutische verwendung. |
FR2593818B1 (fr) * | 1986-02-05 | 1988-04-29 | Synthelabo | Derives d'acylaminomethyl-3 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique |
FR2593180B1 (fr) * | 1986-01-22 | 1990-10-26 | Synthelabo | Derives d'acylaminomethyl-1 imidazo (1,2-a)quinoleines, leur preparation et leur application en therapeutique |
US4990506A (en) * | 1986-02-05 | 1991-02-05 | Synthelabo | 3-(acylaminomethyl)imidazo[1,2-a]pyridine derivatives and their application in therapy |
FR2606409B1 (fr) * | 1986-11-07 | 1989-05-05 | Synthelabo | Derives d'imidazopyridine, leur preparation et leur application en therapeutique |
ES2026666T3 (es) * | 1987-03-27 | 1992-05-01 | Synthelabo | Procedimiento para preparar derivados de imidazopiridinas. |
FR2615513B1 (fr) * | 1987-05-21 | 1989-07-13 | Synthelabo | Derives d'acylaminomethyl-3 tetrahydro-5,6,7,8 imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique |
FR2654933B1 (fr) * | 1989-11-30 | 1994-06-10 | Synthelabo | Utilisation d'une imidazopyridine pour la fabrication de medicaments anesthesiques. |
KR910011852A (ko) * | 1989-12-04 | 1991-08-07 | 폴 디. 매튜카이티스 | 신경독 장해 치료용 이미다조[1,2-a]피리디닐알킬 화합물 |
IE904346A1 (en) * | 1989-12-04 | 1991-06-05 | Searle & Co | IMIDAZO[1,2-a]PYRIDINYLALKYL COMPOUNDS FOR TREATMENT OF¹NEUROTOXIC INJURY |
US5716964A (en) * | 1989-12-04 | 1998-02-10 | G.D. Searle & Co. | Tetrazolyl substituted imidazo 1,2-a!pyridinylalkyl compounds for treatment of neurotoxic injury |
US5464843A (en) * | 1992-06-23 | 1995-11-07 | G.D. Searle & Co. | Imidazo[1,2-a]pyridinyldiacid compounds for cognitive enhancement and for treatment of cognitive disorders and neutrotoxic injury |
AUPP278498A0 (en) * | 1998-04-03 | 1998-04-30 | Australian Nuclear Science & Technology Organisation | Peripheral benzodiazepine receptor binding agents |
DE10019714A1 (de) * | 2000-04-20 | 2002-01-10 | Gruenenthal Gmbh | Salze von bicyclischen, N-acylierten Imidazo-3-aminen und Imidazo-5-aminen |
WO2002002557A2 (en) * | 2000-06-30 | 2002-01-10 | Neurogen Corporation | 2-phenylimidazo[1,2-a]pyridine derivatives: a new class of gaba brain receptor ligands |
US6596731B2 (en) | 2001-03-27 | 2003-07-22 | Hoffmann-La Roche Inc. | Substituted imidazo[1,2-A] pyridine derivatives |
DE10247269A1 (de) | 2002-10-10 | 2004-04-22 | Grünenthal GmbH | Substituierte C-Imidazo[1,2-a]pyridin-3-yl-methylamine |
AU2004287847A1 (en) * | 2003-10-28 | 2005-05-19 | Sepracor Inc. | Imidazo(1,2-a)pyridine anxiolytics |
WO2005081749A2 (en) * | 2004-01-23 | 2005-09-09 | Avanir Pharmaceuticals, Inc. | Neutralizing human antibodies to anthraxtoxin |
FR2874611B1 (fr) * | 2004-08-31 | 2006-11-17 | Servier Lab | Nouveaux derives d'imidazopyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
PT1814880E (pt) * | 2004-11-11 | 2009-04-23 | Ferrer Int | Compostos imidazo[1,2-a]piridina, composições, utilizações e métodos a eles relacionados |
US8178533B2 (en) * | 2005-06-01 | 2012-05-15 | Ucb Pharma, S.A. | 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses |
WO2008132142A2 (en) * | 2007-04-27 | 2008-11-06 | Ucb Pharma S.A. | New heterocyclic derivatives useful for the treatment of cns disorders |
CA2724842A1 (en) * | 2008-05-19 | 2009-11-26 | Sunovion Pharmaceuticals Inc. | Imidazo[1,2-a]pyridine compounds |
WO2010064020A1 (en) * | 2008-12-04 | 2010-06-10 | Proximagen Ltd. | Imidazopyridine compounds |
WO2014187922A1 (en) | 2013-05-24 | 2014-11-27 | Iomet Pharma Ltd. | Slc2a transporter inhibitors |
US20230121497A1 (en) * | 2020-01-29 | 2023-04-20 | Foghorn Therapeutics Inc. | Compounds and uses thereof |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB991589A (en) * | 1963-04-30 | 1965-05-12 | Selvi & C Lab Bioterapico | Novel [1,2-ª‡]imidazopyridines and a process for the manufacture thereof |
GB1076089A (en) * | 1965-11-09 | 1967-07-19 | Selvi & C Lab Bioterapico | New derivatives of imidazo [1,2-a]-pyridine and a process for the manufacture thereof |
-
1984
- 1984-08-07 FR FR8412447A patent/FR2568880B1/fr not_active Expired
-
1985
- 1985-07-30 DE DE8585401554T patent/DE3567867D1/de not_active Expired
- 1985-07-30 EP EP85401554A patent/EP0172096B1/fr not_active Expired
- 1985-07-30 AT AT85401554T patent/ATE40365T1/de not_active IP Right Cessation
- 1985-08-06 IL IL76020A patent/IL76020A/xx not_active IP Right Cessation
- 1985-08-06 JP JP60173977A patent/JPS6147485A/ja active Granted
- 1985-08-06 FI FI853026A patent/FI80696C/fi not_active IP Right Cessation
- 1985-08-06 GR GR851928A patent/GR851928B/el unknown
- 1985-08-06 ES ES545928A patent/ES8604592A1/es not_active Expired
- 1985-08-06 ZA ZA855939A patent/ZA855939B/xx unknown
- 1985-08-06 NO NO853100A patent/NO162189C/no unknown
- 1985-08-06 AR AR85301203A patent/AR241185A1/es active
- 1985-08-06 DK DK356885A patent/DK163923C/da not_active IP Right Cessation
- 1985-08-06 MX MX206217A patent/MX160845A/es unknown
- 1985-08-06 NZ NZ213013A patent/NZ213013A/en unknown
- 1985-08-06 KR KR1019850005660A patent/KR910004450B1/ko not_active IP Right Cessation
- 1985-08-06 AU AU45809/85A patent/AU575190B2/en not_active Ceased
- 1985-08-06 HU HU852991A patent/HU193799B/hu not_active IP Right Cessation
- 1985-08-06 CA CA000488165A patent/CA1261830A/en not_active Expired
- 1985-08-06 IE IE193785A patent/IE58347B1/en not_active IP Right Cessation
- 1985-08-06 PT PT80921A patent/PT80921B/pt not_active IP Right Cessation
-
1986
- 1986-02-07 US US06/826,966 patent/US4650796A/en not_active Expired - Lifetime
-
1991
- 1991-11-25 CZ CS913576A patent/CZ357691A3/cs unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IL76020A (en) | 3-(acylaminomethyl)-2-phenyl imidazo(1,2-a)pyridine derivatives,their preparation and pharmaceutical compositions containing them | |
IL62494A0 (en) | 3-(1-piperidinylalkyl)-4h-pyrido(1,2-a)pyrimidin-4-one derivatives,their preparation and pharmaceutical compositions containing them | |
DE3166531D1 (en) | Imidazo(1,2-a)pyridines, processes for their preparation and pharmaceutical compositions containing them | |
IL64759A0 (en) | Furo-(3,4-c)pyridine derivatives,their preparation and pharmaceutical compositions containing them | |
IL76133A (en) | Mercaptomethyl-octahydro-oxo-pyridazino(1,2-a)(1,2)diazepine-,diazocine-and(1,2,5)triazepinecarboxylic acid derivatives,their preparation and pharmaceutical compositions containing them and certain intermediates therefor | |
IL76405A0 (en) | 1,3-diacyl-2-oxyindole derivatives,their preparation and pharmaceutical compositions containing them | |
IL86798A0 (en) | 2,2-dimethylchroman-3-ol derivatives,their preparation and pharmaceutical compositions containing them | |
IL71243A0 (en) | Furo-(3,4-c)-pyridine derivatives,their preparation and pharmaceutical compositions containing them | |
ZA848130B (en) | New 6-vinyl-furo-(3,4-c)-pyridine derivatives,their preparation and pharmaceutical compositions containing them | |
IL62246A (en) | 2(1h)-pyridinone derivatives,their preparation and pharmaceutical compositions containing them | |
IL68442A0 (en) | Imidazo(1,2-a)pyridine derivatives,their preparation and pharmaceutical compositions containing them | |
IL81209A (en) | Substituted 6h-indolo(2,3-b)-quinoxalines,their preparation and pharmaceutical compositions comprising them | |
IL63982A (en) | 6-hydroxy-2-phenyl-imidazo(4,5-b)pyridines,their preparation and pharmaceutical compositions containing them | |
NZ211424A (en) | Pharmaceutical compositions comprising 3-isobutyryl-2-isopropylpyrazolo(1,5-a)pyridine | |
IL70485A (en) | Imidazo(1,5-a)pyridine derivatives,their preparation and pharmaceutical compositions containing them | |
IL88002A0 (en) | 2,2-dimethylchromene derivatives,their preparation and pharmaceutical compositions containing them | |
IL80658A0 (en) | 6,7,8,9-tetrahydro-10-methyl-pyrido(1,2-a)indol-9-amines and derivatives thereof,their preparation and pharmaceutical compositions containing them | |
NZ224032A (en) | Imidazo(1,2-a)pyridine derivatives and pharmaceutical compositions | |
IL66101A (en) | Substituted imidazo(1,5-a)pyridines,their manufacture and pharmaceutical compositions containing them | |
IL75603A0 (en) | 1,3-dioxanylheptenoic acid derivatives,their preparation and pharmaceutical compositions containing them | |
IL76019A0 (en) | Imidazo(1,2-a)quinoline derivatives,their preparation and pharmaceutical compositions containing them | |
IL73810A (en) | 4,5,6,7-tetrahydrothiazolo-(5,4-c)pyridine derivatives,their preparation and pharmaceutical compositions containing them | |
IL88658A0 (en) | 8,9-annelated beta-carbolines and 3,4-dihydro-beta-carbolines,their preparation and pharmaceutical compositions containing them | |
IL70651A0 (en) | Carboxy-thiazolo(3,2-a)pyrimidine derivatives,their preparation and pharmaceutical compositions containing them | |
IL65555A (en) | 5-pyridyl-1h-pyrazolo(3,4-b)pyridin-3-amine derivatives,their preparation and pharmaceutical compositions containing them |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
KB | Patent renewed | ||
KB | Patent renewed | ||
EXP | Patent expired |