IL65977A - 1,4,9,10-tetrahydropyrazolo(4,3-e)pyrido(3,2-b)(1,4)diazepin-10-one derivatives,their preparation and pharmaceutical compositions containing them - Google Patents
1,4,9,10-tetrahydropyrazolo(4,3-e)pyrido(3,2-b)(1,4)diazepin-10-one derivatives,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL65977A IL65977A IL65977A IL6597782A IL65977A IL 65977 A IL65977 A IL 65977A IL 65977 A IL65977 A IL 65977A IL 6597782 A IL6597782 A IL 6597782A IL 65977 A IL65977 A IL 65977A
- Authority
- IL
- Israel
- Prior art keywords
- tetrahydropyrazolo
- diazepin
- pyrido
- derivatives
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19813122670 DE3122670A1 (de) | 1981-06-06 | 1981-06-06 | "neue 1,4,9,10-tetrahydro-pyrazolo(4,3-e) pyrido(3,2-b)(1,4)diazepin-10-one, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von pharmazeutischen wirkstoffen" |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL65977A0 IL65977A0 (en) | 1982-09-30 |
| IL65977A true IL65977A (en) | 1984-12-31 |
Family
ID=6134176
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL65977A IL65977A (en) | 1981-06-06 | 1982-06-04 | 1,4,9,10-tetrahydropyrazolo(4,3-e)pyrido(3,2-b)(1,4)diazepin-10-one derivatives,their preparation and pharmaceutical compositions containing them |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US4381303A (ko) |
| EP (1) | EP0066774B1 (ko) |
| JP (1) | JPS57212182A (ko) |
| KR (1) | KR880001719B1 (ko) |
| AR (1) | AR229124A1 (ko) |
| AT (1) | ATE10744T1 (ko) |
| AU (1) | AU552765B2 (ko) |
| CA (1) | CA1167440A (ko) |
| CS (1) | CS226743B2 (ko) |
| DD (1) | DD202574A5 (ko) |
| DE (2) | DE3122670A1 (ko) |
| DK (1) | DK253382A (ko) |
| ES (1) | ES512846A0 (ko) |
| FI (1) | FI71560C (ko) |
| GB (1) | GB2117755B (ko) |
| GR (1) | GR76438B (ko) |
| HU (1) | HU186067B (ko) |
| IE (1) | IE53067B1 (ko) |
| IL (1) | IL65977A (ko) |
| NO (1) | NO158063C (ko) |
| NZ (1) | NZ200859A (ko) |
| PH (1) | PH17719A (ko) |
| PL (1) | PL135845B1 (ko) |
| PT (1) | PT75016B (ko) |
| SU (1) | SU1103795A3 (ko) |
| YU (1) | YU118282A (ko) |
| ZA (1) | ZA823919B (ko) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3643666A1 (de) * | 1986-12-20 | 1988-06-30 | Thomae Gmbh Dr K | Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| US4749788A (en) * | 1987-04-13 | 1988-06-07 | A. H. Robins Company, Incorporated | Process for the preparation of aryl-pyrido(1,4) benzodiazepines |
| US5366972A (en) * | 1989-04-20 | 1994-11-22 | Boehringer Ingelheim Pharmaceuticals, Inc. | 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection |
| ATE103918T1 (de) * | 1989-06-28 | 1994-04-15 | Boehringer Ingelheim Pharma | 5,11-dihydro-6h-dipyrido(3,2-b:2',3'e>(1,4>diazepin-6-one und -thione und ihre verwendung bei der aids-vorbeugung oder behandlung. |
| CA2052946A1 (en) * | 1990-10-19 | 1992-04-20 | Karl G. Grozinger | Method for the preparation of 5,11-dihydro-6h-dipyrido ¬3,2-b:2', 3'-e| ¬1,4|diazepines |
| ES2137113B1 (es) | 1997-07-29 | 2000-09-16 | Almirall Prodesfarma Sa | Nuevos derivados de triazolo-piridazinas heterociclicos. |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3450694A (en) * | 1966-02-23 | 1969-06-17 | Abbott Lab | Substituted benzoxazepines and benzothiazepines |
| DE2707269A1 (de) * | 1977-02-19 | 1978-08-24 | Hoechst Ag | Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung |
| DK334580A (da) * | 1979-08-03 | 1981-02-04 | Byk Gulden Lomberg Chem Fab | Fremgangsmaade til fremstilling af substituerede tetraazatricycler |
-
1981
- 1981-06-06 DE DE19813122670 patent/DE3122670A1/de not_active Withdrawn
-
1982
- 1982-05-13 US US06/377,911 patent/US4381303A/en not_active Expired - Fee Related
- 1982-05-25 DE DE8282104549T patent/DE3261530D1/de not_active Expired
- 1982-05-25 EP EP82104549A patent/EP0066774B1/de not_active Expired
- 1982-05-25 AT AT82104549T patent/ATE10744T1/de not_active IP Right Cessation
- 1982-05-25 SU SU823441915A patent/SU1103795A3/ru active
- 1982-06-01 AR AR289564A patent/AR229124A1/es active
- 1982-06-02 GR GR68322A patent/GR76438B/el unknown
- 1982-06-03 YU YU01182/82A patent/YU118282A/xx unknown
- 1982-06-03 PL PL1982236742A patent/PL135845B1/pl unknown
- 1982-06-03 KR KR8202494A patent/KR880001719B1/ko active
- 1982-06-03 CS CS824137A patent/CS226743B2/cs unknown
- 1982-06-03 DD DD82240437A patent/DD202574A5/de unknown
- 1982-06-04 NZ NZ200859A patent/NZ200859A/en unknown
- 1982-06-04 PH PH27402A patent/PH17719A/en unknown
- 1982-06-04 IL IL65977A patent/IL65977A/xx unknown
- 1982-06-04 GB GB08216381A patent/GB2117755B/en not_active Expired
- 1982-06-04 AU AU84605/82A patent/AU552765B2/en not_active Ceased
- 1982-06-04 CA CA000404541A patent/CA1167440A/en not_active Expired
- 1982-06-04 NO NO821882A patent/NO158063C/no unknown
- 1982-06-04 IE IE1350/82A patent/IE53067B1/en unknown
- 1982-06-04 FI FI821992A patent/FI71560C/fi not_active IP Right Cessation
- 1982-06-04 PT PT75016A patent/PT75016B/pt unknown
- 1982-06-04 ZA ZA823919A patent/ZA823919B/xx unknown
- 1982-06-04 ES ES512846A patent/ES512846A0/es active Granted
- 1982-06-04 DK DK253382A patent/DK253382A/da not_active Application Discontinuation
- 1982-06-04 JP JP57096080A patent/JPS57212182A/ja active Pending
- 1982-06-04 HU HU821823A patent/HU186067B/hu unknown
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